ATE220670T1 - Herstellung von thiazolen - Google Patents
Herstellung von thiazolenInfo
- Publication number
- ATE220670T1 ATE220670T1 AT97954817T AT97954817T ATE220670T1 AT E220670 T1 ATE220670 T1 AT E220670T1 AT 97954817 T AT97954817 T AT 97954817T AT 97954817 T AT97954817 T AT 97954817T AT E220670 T1 ATE220670 T1 AT E220670T1
- Authority
- AT
- Austria
- Prior art keywords
- alkyl
- halogen
- formula
- phenyl
- compound
- Prior art date
Links
- FZWLAAWBMGSTSO-UHFFFAOYSA-N Thiazole Chemical compound C1=CSC=N1 FZWLAAWBMGSTSO-UHFFFAOYSA-N 0.000 title 1
- 125000000217 alkyl group Chemical group 0.000 abstract 7
- 150000001875 compounds Chemical class 0.000 abstract 3
- 125000001997 phenyl group Chemical class [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 3
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 abstract 2
- 125000003342 alkenyl group Chemical group 0.000 abstract 2
- 125000001797 benzyl group Chemical class [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 2
- 229910052799 carbon Inorganic materials 0.000 abstract 2
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical group [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 abstract 1
- AFVFQIVMOAPDHO-UHFFFAOYSA-M Methanesulfonate Chemical group CS([O-])(=O)=O AFVFQIVMOAPDHO-UHFFFAOYSA-M 0.000 abstract 1
- 125000000304 alkynyl group Chemical group 0.000 abstract 1
- -1 benzothilzolyl Chemical class 0.000 abstract 1
- 125000000113 cyclohexyl group Chemical class [H]C1([H])C([H])([H])C([H])([H])C([H])(*)C([H])([H])C1([H])[H] 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 150000002367 halogens Chemical class 0.000 abstract 1
- 125000005842 heteroatom Chemical group 0.000 abstract 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
- 229910052757 nitrogen Inorganic materials 0.000 abstract 1
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 1
- 229910052760 oxygen Inorganic materials 0.000 abstract 1
- 125000004076 pyridyl group Chemical class 0.000 abstract 1
- 125000000714 pyrimidinyl group Chemical class 0.000 abstract 1
- 229910052717 sulfur Inorganic materials 0.000 abstract 1
- 125000000335 thiazolyl group Chemical class 0.000 abstract 1
- JOXIMZWYDAKGHI-UHFFFAOYSA-N toluene-4-sulfonic acid Chemical compound CC1=CC=C(S(O)(=O)=O)C=C1 JOXIMZWYDAKGHI-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/08—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D277/12—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/16—Sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/36—Sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/70—Sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/70—Sulfur atoms
- C07D277/74—Sulfur atoms substituted by carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH312596 | 1996-12-19 | ||
| PCT/EP1997/007088 WO1998027075A1 (en) | 1996-12-19 | 1997-12-17 | Preparation of thiazoles |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE220670T1 true ATE220670T1 (de) | 2002-08-15 |
Family
ID=4249152
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT01129478T ATE307807T1 (de) | 1996-12-19 | 1997-12-17 | Herstellung von thiazolen |
| AT97954817T ATE220670T1 (de) | 1996-12-19 | 1997-12-17 | Herstellung von thiazolen |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT01129478T ATE307807T1 (de) | 1996-12-19 | 1997-12-17 | Herstellung von thiazolen |
Country Status (11)
| Country | Link |
|---|---|
| US (5) | US6548676B1 (de) |
| EP (3) | EP0946532B1 (de) |
| JP (1) | JP4354533B2 (de) |
| KR (1) | KR100521067B1 (de) |
| AT (2) | ATE307807T1 (de) |
| AU (1) | AU6205698A (de) |
| DE (2) | DE69734479T2 (de) |
| DK (2) | DK1201662T3 (de) |
| ES (2) | ES2246985T3 (de) |
| IL (1) | IL130293A0 (de) |
| WO (1) | WO1998027075A1 (de) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI359810B (en) * | 2004-11-04 | 2012-03-11 | Mitsubishi Tanabe Pharma Corp | Carboxylic acid derivative containing thiazole rin |
| US10118890B2 (en) | 2014-10-10 | 2018-11-06 | The Research Foundation For The State University Of New York | Trifluoromethoxylation of arenes via intramolecular trifluoromethoxy group migration |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US546167A (en) * | 1895-09-10 | Mills | ||
| EP0192060B1 (de) | 1985-02-04 | 1991-09-18 | Nihon Bayer Agrochem K.K. | Heterocyclische Verbindungen |
| US5180833A (en) * | 1990-03-16 | 1993-01-19 | Takeda Chemical Industries, Ltd. | Process for the preparation of chlorothiazole derivatives |
| CA2044755A1 (en) * | 1990-06-18 | 1991-12-19 | Bunji Natsume | Pyrazolecarboxamide, insecticidal and miticidal composition, and fungicidal composition for use in agriculture and horticulture |
| ZA9610046B (en) * | 1995-12-01 | 1997-07-10 | Ciba Geigy | Process for preparing 2-chlorothiazole compounds |
-
1997
- 1997-12-17 EP EP97954817A patent/EP0946532B1/de not_active Expired - Lifetime
- 1997-12-17 ES ES01129478T patent/ES2246985T3/es not_active Expired - Lifetime
- 1997-12-17 DE DE69734479T patent/DE69734479T2/de not_active Expired - Lifetime
- 1997-12-17 EP EP05013434A patent/EP1577307A3/de not_active Withdrawn
- 1997-12-17 AT AT01129478T patent/ATE307807T1/de active
- 1997-12-17 DK DK01129478T patent/DK1201662T3/da active
- 1997-12-17 KR KR10-1999-7005612A patent/KR100521067B1/ko not_active Expired - Fee Related
- 1997-12-17 AT AT97954817T patent/ATE220670T1/de active
- 1997-12-17 DE DE69714076T patent/DE69714076T2/de not_active Expired - Lifetime
- 1997-12-17 JP JP52732398A patent/JP4354533B2/ja not_active Expired - Fee Related
- 1997-12-17 US US09/331,433 patent/US6548676B1/en not_active Expired - Fee Related
- 1997-12-17 WO PCT/EP1997/007088 patent/WO1998027075A1/en not_active Ceased
- 1997-12-17 ES ES97954817T patent/ES2181059T3/es not_active Expired - Lifetime
- 1997-12-17 EP EP01129478A patent/EP1201662B1/de not_active Expired - Lifetime
- 1997-12-17 AU AU62056/98A patent/AU6205698A/en not_active Abandoned
- 1997-12-17 DK DK97954817T patent/DK0946532T3/da active
- 1997-12-17 IL IL13029397A patent/IL130293A0/xx not_active IP Right Cessation
-
2003
- 2003-03-27 US US10/400,826 patent/US7161011B2/en not_active Expired - Fee Related
-
2006
- 2006-10-24 US US11/552,255 patent/US7323564B2/en not_active Expired - Fee Related
-
2007
- 2007-11-30 US US11/947,891 patent/US7538229B2/en not_active Expired - Fee Related
-
2009
- 2009-04-16 US US12/424,594 patent/US7795442B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| ES2246985T3 (es) | 2006-03-01 |
| DK1201662T3 (da) | 2006-02-13 |
| EP1577307A2 (de) | 2005-09-21 |
| US7161011B2 (en) | 2007-01-09 |
| JP4354533B2 (ja) | 2009-10-28 |
| EP0946532B1 (de) | 2002-07-17 |
| KR100521067B1 (ko) | 2005-10-14 |
| DE69714076D1 (de) | 2002-08-22 |
| US7323564B2 (en) | 2008-01-29 |
| AU6205698A (en) | 1998-07-15 |
| WO1998027075A1 (en) | 1998-06-25 |
| EP1577307A3 (de) | 2009-04-29 |
| ES2181059T3 (es) | 2003-02-16 |
| DE69734479T2 (de) | 2006-06-29 |
| IL130293A0 (en) | 2000-06-01 |
| EP1201662B1 (de) | 2005-10-26 |
| US20080076920A1 (en) | 2008-03-27 |
| US20030216579A1 (en) | 2003-11-20 |
| US20070055063A1 (en) | 2007-03-08 |
| US6548676B1 (en) | 2003-04-15 |
| DE69714076T2 (de) | 2003-03-06 |
| JP2001506255A (ja) | 2001-05-15 |
| US7795442B2 (en) | 2010-09-14 |
| US7538229B2 (en) | 2009-05-26 |
| EP0946532A1 (de) | 1999-10-06 |
| DK0946532T3 (da) | 2002-11-11 |
| US20090198054A1 (en) | 2009-08-06 |
| KR20000069614A (ko) | 2000-11-25 |
| DE69734479D1 (de) | 2005-12-01 |
| EP1201662A1 (de) | 2002-05-02 |
| ATE307807T1 (de) | 2005-11-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification |