IL120343A0 - Epimers of (22RS)-N-(1,1,1-trifluoro-2-phenylprop-2-YL)-3-oxo-4-aza-5alpha-androst-1-ene-17beta-carboxamide - Google Patents

Epimers of (22RS)-N-(1,1,1-trifluoro-2-phenylprop-2-YL)-3-oxo-4-aza-5alpha-androst-1-ene-17beta-carboxamide

Info

Publication number
IL120343A0
IL120343A0 IL12034396A IL12034396A IL120343A0 IL 120343 A0 IL120343 A0 IL 120343A0 IL 12034396 A IL12034396 A IL 12034396A IL 12034396 A IL12034396 A IL 12034396A IL 120343 A0 IL120343 A0 IL 120343A0
Authority
IL
Israel
Prior art keywords
5alpha
17beta
androst
phenylprop
epimers
Prior art date
Application number
IL12034396A
Other languages
English (en)
Original Assignee
Pharmacia & Upjohn Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia & Upjohn Spa filed Critical Pharmacia & Upjohn Spa
Publication of IL120343A0 publication Critical patent/IL120343A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • C07J73/001—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
    • C07J73/005—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by nitrogen as hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
IL12034396A 1995-07-21 1996-06-28 Epimers of (22RS)-N-(1,1,1-trifluoro-2-phenylprop-2-YL)-3-oxo-4-aza-5alpha-androst-1-ene-17beta-carboxamide IL120343A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT95MI001587A IT1275594B1 (it) 1995-07-21 1995-07-21 Epimeri del (22rs)-n-(1,1,1-trifluoro-2-fenilprop-2-il)-3-osso -4-aza-5alfa-androst-1-ene-17beta-carbossammide
PCT/EP1996/002830 WO1997004002A1 (en) 1995-07-21 1996-06-28 EPIMERS OF (22RS)-N-(1,1,1-TRIFLUORO-2-PHENYLPROP-2-YL)-3-OXO-4-AZA-5α-ANDROST-1-ENE-17β-CARBOXAMIDE

Publications (1)

Publication Number Publication Date
IL120343A0 true IL120343A0 (en) 1997-06-10

Family

ID=11372032

Family Applications (1)

Application Number Title Priority Date Filing Date
IL12034396A IL120343A0 (en) 1995-07-21 1996-06-28 Epimers of (22RS)-N-(1,1,1-trifluoro-2-phenylprop-2-YL)-3-oxo-4-aza-5alpha-androst-1-ene-17beta-carboxamide

Country Status (17)

Country Link
EP (1) EP0782582A1 (no)
JP (1) JPH10506411A (no)
KR (1) KR970706298A (no)
CN (1) CN1159195A (no)
AR (1) AR003967A1 (no)
AU (1) AU6418396A (no)
BR (1) BR9606527A (no)
CA (1) CA2199273A1 (no)
EA (1) EA199700045A1 (no)
HU (1) HUP9702465A3 (no)
IL (1) IL120343A0 (no)
IT (1) IT1275594B1 (no)
MX (1) MX9701948A (no)
NO (1) NO971196L (no)
PL (1) PL319351A1 (no)
WO (1) WO1997004002A1 (no)
ZA (1) ZA965678B (no)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU6137399A (en) * 1998-09-09 2000-03-27 Merck & Co., Inc. Method of determining and reducing the risk of bph-related urologic events
DE60018707T2 (de) * 1999-01-25 2006-02-09 Smithkline Beecham Corp. Anti-androgene und verfahren zur behandlung von krankheiten
CN100355772C (zh) * 2005-12-28 2007-12-19 天津大学 具有5α－还原酶抑制活性的甾体化合物及其制备方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9216284D0 (en) * 1992-07-31 1992-09-16 Erba Carlo Spa Fluorinated 17beta-substituted 4-aza-5alpha-androstane-3-one derivatives

Also Published As

Publication number Publication date
NO971196D0 (no) 1997-03-14
AU6418396A (en) 1997-02-18
CA2199273A1 (en) 1997-02-06
PL319351A1 (en) 1997-08-04
WO1997004002A1 (en) 1997-02-06
ITMI951587A0 (it) 1995-07-21
ITMI951587A1 (it) 1997-01-21
HUP9702465A3 (en) 1998-11-30
NO971196L (no) 1997-03-14
HUP9702465A2 (hu) 1998-05-28
AR003967A1 (es) 1998-09-30
EA199700045A1 (ru) 1997-12-30
BR9606527A (pt) 1997-12-23
EP0782582A1 (en) 1997-07-09
MX9701948A (es) 1997-06-28
JPH10506411A (ja) 1998-06-23
CN1159195A (zh) 1997-09-10
IT1275594B1 (it) 1997-08-06
KR970706298A (ko) 1997-11-03
ZA965678B (en) 1997-01-24

Similar Documents

Publication Publication Date Title
GB2319250B (en) Derivatives of 6,8-Difluoro-7-Hydroxycoumarin
PL322277A1 (en) Derivatives of pyrazol-4-ylobenzoyl
PL324992A1 (en) Novel derivatives of 2,3-dioxotetrahydoquinoxaline
PL338563A1 (en) Substituted derivatives of 1,2,3,4-tetrahydronaphtalene
GR3033254T3 (en) 1 alpha, 26-dihydroxy-D-homo-vitamin D3
GB9526560D0 (en) Use of 2-Amino-Heterocycles
ZA969753B (en) Crystalline hydrochloride of (r)-(-)-2-än-4-(1,1-dioxido-3-oxo-2,3-dihydrobenzhisothiazol-2-yl)-aminomethylü-chroman
AU3284395A (en) Synthesis of 1,1,1,3,3,-pentafluoropropane
EP0754407A3 (en) Liquid compositions of 1,2-benzisothiazolin-3-one
PL324451A1 (en) Derivatives of diphenylmethylenepiperidine
AU4329396A (en) Use of 3,4-diphenylchromans
ZA969221B (en) Indolealkyl derivatives of benzodioxanmethylamine.
GB9512290D0 (en) Uses of polyhexanide
PL340372A1 (en) Novel 3,6x-hemiketals of 9a-azalydes class
ZA965922B (en) Preparation of N-substituted 3-hydroxypyrazoles.
ZA96725B (en) Use of phenyclyclohexylcarboxamides
GB9518692D0 (en) 'Spraymate'
PL322279A1 (en) Method of obtaining 1,2-benzoylthiazolin-3-ones
IL113057A0 (en) Compositions for the treatment of dandruff
PL327141A1 (en) Method of obtaining 9,11 beta-epoxysteroides
ZA965678B (en) Epimers of (22rs)-n-(1,1,1-trifluoro-2-phenylprop-2-yl)-3-oxo-4-aza-5alpha-androst-1-ene-17beta-carboxamide
IL119744A0 (en) Use of 8,9-dehydroestrone
IL118731A0 (en) Process for the preparation of 2,2-dialkyl-arylidene-cycloalkanones
ZA963356B (en) Novel uses of heptafluoropropane
HUP9600316A3 (en) Process for the preparation of n-(ortho-alkyl-phenyl)-imides