IL118200A0 - Process for the preparation of substituted 2-fluoro-pyrimidines - Google Patents

Process for the preparation of substituted 2-fluoro-pyrimidines

Info

Publication number
IL118200A0
IL118200A0 IL11820096A IL11820096A IL118200A0 IL 118200 A0 IL118200 A0 IL 118200A0 IL 11820096 A IL11820096 A IL 11820096A IL 11820096 A IL11820096 A IL 11820096A IL 118200 A0 IL118200 A0 IL 118200A0
Authority
IL
Israel
Prior art keywords
pyrimidines
fluoro
substituted
preparation
Prior art date
Application number
IL11820096A
Other languages
English (en)
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of IL118200A0 publication Critical patent/IL118200A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/52—Two oxygen atoms
    • C07D239/54—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals
    • C07D239/545—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals with other hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/553—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals with other hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms with halogen atoms or nitro radicals directly attached to ring carbon atoms, e.g. fluorouracil
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/30—Halogen atoms or nitro radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL11820096A 1995-05-11 1996-05-09 Process for the preparation of substituted 2-fluoro-pyrimidines IL118200A0 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19517186A DE19517186A1 (de) 1995-05-11 1995-05-11 Verfahren zur Herstellung substituierter 2-Fluor-pyrimidine

Publications (1)

Publication Number Publication Date
IL118200A0 true IL118200A0 (en) 1996-09-12

Family

ID=7761586

Family Applications (1)

Application Number Title Priority Date Filing Date
IL11820096A IL118200A0 (en) 1995-05-11 1996-05-09 Process for the preparation of substituted 2-fluoro-pyrimidines

Country Status (7)

Country Link
US (1) US5681957A (xx)
EP (1) EP0742212A1 (xx)
JP (1) JPH08301855A (xx)
CZ (1) CZ137496A3 (xx)
DE (1) DE19517186A1 (xx)
HU (1) HUP9601261A3 (xx)
IL (1) IL118200A0 (xx)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2582600A (en) * 1999-09-16 2001-04-17 Rimma Iliinichna Ashkinazi Bioactive substance containing derivatives of 2-amino-6-aryloxypyrimidines and intermediary products of synthesis thereof
WO2003006439A1 (en) 2001-07-13 2003-01-23 Astrazeneca Uk Limited Preparation of aminopyrimidine compounds
DK1578731T3 (da) * 2002-12-16 2010-02-15 Astrazeneca Uk Ltd Fremgangsmåde til fremstilling af pyrimidinforbindelser
EP1758897A1 (en) * 2004-04-02 2007-03-07 F.Hoffmann-La Roche Ag Novel diazine derivatives, their manufacture and use as pharmaceutical agents
GB0428328D0 (en) * 2004-12-24 2005-02-02 Astrazeneca Uk Ltd Chemical process
DK1848678T3 (en) * 2005-02-09 2015-09-21 Syngenta Participations Ag METHOD OF MANUFACTURING INTERMEDIATES
CL2008000467A1 (es) * 2007-02-14 2008-08-22 Janssen Pharmaceutica Nv Compuestos derivados de 2-aminopirimidina, moduladores del receptor histamina h4; su procedimiento de preparacion; composicion farmaceutica que comprende a dichos compuestos; y su uso para tratar un trastorno inflamatorio seleccionado de alegia, asma
CN102134240A (zh) * 2010-06-29 2011-07-27 嘉兴宜博生物医药科技有限公司 一种6-氟-7-氮杂吲哚的合成方法
CN102161607B (zh) * 2011-03-11 2014-07-30 华南农业大学 一种含氟芳香化合物的制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS54157575A (en) * 1978-05-31 1979-12-12 Expansia Sa Manufacture of 22chloropyrimidine
CA2074812A1 (en) * 1990-11-30 1992-05-31 Takumi Yoshimura Alkanoic acid amide derivative or its salt, process for producing the same and herbicidal composition
KR100233068B1 (ko) * 1991-11-26 1999-12-01 하인즈 모제르 2-치환된 4,6-디알콕시피리미딘의 제조방법
JP3269192B2 (ja) * 1992-08-05 2002-03-25 ロンザ リミテッド ２−ハロゲン−４，６−ジアルコキシ−ピリミジンの製造方法

Also Published As

Publication number Publication date
HU9601261D0 (en) 1996-07-29
HUP9601261A3 (en) 1999-03-01
HUP9601261A2 (en) 1997-02-28
DE19517186A1 (de) 1996-11-14
CZ137496A3 (en) 1996-11-13
US5681957A (en) 1997-10-28
JPH08301855A (ja) 1996-11-19
EP0742212A1 (de) 1996-11-13

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