HUP9601261A3 - Process for preparation of 2-fluor-pirimidine-derivatives - Google Patents

Process for preparation of 2-fluor-pirimidine-derivatives

Info

Publication number
HUP9601261A3
HUP9601261A3 HU9601261A HUP9601261A HUP9601261A3 HU P9601261 A3 HUP9601261 A3 HU P9601261A3 HU 9601261 A HU9601261 A HU 9601261A HU P9601261 A HUP9601261 A HU P9601261A HU P9601261 A3 HUP9601261 A3 HU P9601261A3
Authority
HU
Hungary
Prior art keywords
pirimidine
fluor
derivatives
preparation
Prior art date
Application number
HU9601261A
Other languages
English (en)
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of HU9601261D0 publication Critical patent/HU9601261D0/hu
Publication of HUP9601261A2 publication Critical patent/HUP9601261A2/hu
Publication of HUP9601261A3 publication Critical patent/HUP9601261A3/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/52—Two oxygen atoms
    • C07D239/54—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals
    • C07D239/545—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals with other hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/553—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals with other hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms with halogen atoms or nitro radicals directly attached to ring carbon atoms, e.g. fluorouracil
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/30—Halogen atoms or nitro radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
HU9601261A 1995-05-11 1996-05-10 Process for preparation of 2-fluor-pirimidine-derivatives HUP9601261A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19517186A DE19517186A1 (de) 1995-05-11 1995-05-11 Verfahren zur Herstellung substituierter 2-Fluor-pyrimidine

Publications (3)

Publication Number Publication Date
HU9601261D0 HU9601261D0 (en) 1996-07-29
HUP9601261A2 HUP9601261A2 (en) 1997-02-28
HUP9601261A3 true HUP9601261A3 (en) 1999-03-01

Family

ID=7761586

Family Applications (1)

Application Number Title Priority Date Filing Date
HU9601261A HUP9601261A3 (en) 1995-05-11 1996-05-10 Process for preparation of 2-fluor-pirimidine-derivatives

Country Status (7)

Country Link
US (1) US5681957A (hu)
EP (1) EP0742212A1 (hu)
JP (1) JPH08301855A (hu)
CZ (1) CZ137496A3 (hu)
DE (1) DE19517186A1 (hu)
HU (1) HUP9601261A3 (hu)
IL (1) IL118200A0 (hu)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2001019801A1 (fr) * 1999-09-16 2001-03-22 Rimma Iliinichna Ashkinazi Substance bioactive a base de derives des 2-amino-6-aryloxypyrimidines et de produits de synthese intermediaires de ces derniers
BR0211072A (pt) 2001-07-13 2004-12-14 Astrazeneca Uk Ltd Processo para preparar um composto, composto, e, método para a preparação de um composto
US7524955B2 (en) * 2002-12-16 2009-04-28 Astrazeneca Uk Limited Process for the preparation of pyrimidine compounds
BRPI0509394A (pt) * 2004-04-02 2007-09-18 Hoffmann La Roche derivados de diazina, sua manufatura e uso como agentes farmacêuticos
GB0428328D0 (en) * 2004-12-24 2005-02-02 Astrazeneca Uk Ltd Chemical process
US8030529B2 (en) * 2005-02-09 2011-10-04 Syngenta Crop Protection, Inc. Process for the preparation of intermediates
TW200904437A (en) * 2007-02-14 2009-02-01 Janssen Pharmaceutica Nv 2-aminopyrimidine modulators of the histamine H4 receptor
CN102134240A (zh) * 2010-06-29 2011-07-27 嘉兴宜博生物医药科技有限公司 一种6-氟-7-氮杂吲哚的合成方法
CN102161607B (zh) * 2011-03-11 2014-07-30 华南农业大学 一种含氟芳香化合物的制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS54157575A (en) * 1978-05-31 1979-12-12 Expansia Sa Manufacture of 22chloropyrimidine
WO1992009584A1 (fr) * 1990-11-30 1992-06-11 Kumiai Chemical Industry Co., Ltd. Derive d'alcanamide, son sel, son procede de production associe et herbicide
KR100233068B1 (ko) * 1991-11-26 1999-12-01 하인즈 모제르 2-치환된 4,6-디알콕시피리미딘의 제조방법
JP3269192B2 (ja) * 1992-08-05 2002-03-25 ロンザ リミテッド ２−ハロゲン−４，６−ジアルコキシ−ピリミジンの製造方法

Also Published As

Publication number Publication date
HUP9601261A2 (en) 1997-02-28
IL118200A0 (en) 1996-09-12
EP0742212A1 (de) 1996-11-13
HU9601261D0 (en) 1996-07-29
JPH08301855A (ja) 1996-11-19
US5681957A (en) 1997-10-28
CZ137496A3 (en) 1996-11-13
DE19517186A1 (de) 1996-11-14

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