IL117815A - Ascomycin-phenylaminocarbonyloxy derivatives substituted by carboxy or physiologically hydrolysable and acceptable oxycarbonyl moieties their preparation and pharmaceutical compositions containing them - Google Patents
Ascomycin-phenylaminocarbonyloxy derivatives substituted by carboxy or physiologically hydrolysable and acceptable oxycarbonyl moieties their preparation and pharmaceutical compositions containing themInfo
- Publication number
- IL117815A IL117815A IL11781596A IL11781596A IL117815A IL 117815 A IL117815 A IL 117815A IL 11781596 A IL11781596 A IL 11781596A IL 11781596 A IL11781596 A IL 11781596A IL 117815 A IL117815 A IL 117815A
- Authority
- IL
- Israel
- Prior art keywords
- phenylaminocarbonyloxy
- ascomycin
- carboxy
- preparation
- pharmaceutical compositions
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D498/18—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Immunology (AREA)
- Pulmonology (AREA)
- Genetics & Genomics (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- Molecular Biology (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Transplantation (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB9507128.8A GB9507128D0 (en) | 1995-04-06 | 1995-04-06 | Organic compounds |
GBGB9526049.3A GB9526049D0 (en) | 1995-12-20 | 1995-12-20 | Organic compounds |
GBGB9526050.1A GB9526050D0 (en) | 1995-12-20 | 1995-12-20 | Organic compounds |
Publications (2)
Publication Number | Publication Date |
---|---|
IL117815A0 IL117815A0 (en) | 1996-08-04 |
IL117815A true IL117815A (en) | 2000-07-16 |
Family
ID=27267660
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL11781596A IL117815A (en) | 1995-04-06 | 1996-04-03 | Ascomycin-phenylaminocarbonyloxy derivatives substituted by carboxy or physiologically hydrolysable and acceptable oxycarbonyl moieties their preparation and pharmaceutical compositions containing them |
Country Status (21)
Country | Link |
---|---|
US (1) | US5925649A (pt) |
EP (1) | EP0819130A1 (pt) |
JP (1) | JP2000505044A (pt) |
KR (1) | KR19980703583A (pt) |
CN (1) | CN1088068C (pt) |
AR (1) | AR004480A1 (pt) |
AU (1) | AU703523B2 (pt) |
BR (1) | BR9604808A (pt) |
CA (1) | CA2216562A1 (pt) |
CO (1) | CO4750668A1 (pt) |
CZ (1) | CZ312397A3 (pt) |
FI (1) | FI973529A (pt) |
HU (1) | HUP9801993A3 (pt) |
IL (1) | IL117815A (pt) |
MX (1) | MX9707636A (pt) |
NO (1) | NO309273B1 (pt) |
NZ (1) | NZ307170A (pt) |
PL (1) | PL322553A1 (pt) |
SK (1) | SK133997A3 (pt) |
TR (1) | TR199700999T1 (pt) |
WO (1) | WO1996031514A1 (pt) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BRPI9909201B8 (pt) | 1998-03-26 | 2021-05-25 | Astellas Pharma Inc | formulação de composto de macrolídeo de liberação controlada |
GB9826656D0 (en) | 1998-12-03 | 1999-01-27 | Novartis Ag | Organic compounds |
US6121257A (en) * | 1999-03-31 | 2000-09-19 | Abbott Laboratories | Sulfamate containing macrocyclic immunomodulators |
US7063857B1 (en) | 1999-04-30 | 2006-06-20 | Sucampo Ag | Use of macrolide compounds for the treatment of dry eye |
CA2372448A1 (en) * | 1999-04-30 | 2000-11-09 | Sucampo Ag | Use of macrolide compounds for the treatment of dry eye |
US6593292B1 (en) | 1999-08-24 | 2003-07-15 | Cellgate, Inc. | Compositions and methods for enhancing drug delivery across and into epithelial tissues |
AR033151A1 (es) * | 2001-04-12 | 2003-12-03 | Sucampo Pharmaceuticals Inc | Agente para el tratamiento oftalmico topico de las enfermedades inflamatorias oculares |
JP2005512946A (ja) * | 2001-05-09 | 2005-05-12 | ノバルティス アクチエンゲゼルシャフト | 選択的免疫調節法 |
KR20050086648A (ko) * | 2002-11-15 | 2005-08-30 | 노파르티스 아게 | 약물 전달 시스템 |
US20060115522A1 (en) * | 2003-02-17 | 2006-06-01 | Cipla Ltd | Pharmaceutical composition |
TWI324604B (en) | 2003-06-18 | 2010-05-11 | Novartis Ag | New use of staurosporine derivatives |
US7780973B2 (en) * | 2003-12-15 | 2010-08-24 | Ethicon Endo-Surgery, Inc. | Method and device for minimally invasive implantation of biomaterial |
CA2552305A1 (en) * | 2003-12-30 | 2005-07-14 | Astellas Pharma Inc. | Use of macrolides for treating or preventing airflow obstruction |
US20050142161A1 (en) * | 2003-12-30 | 2005-06-30 | Freeman Lynetta J. | Collagen matrix for soft tissue augmentation |
US20080233053A1 (en) * | 2005-02-07 | 2008-09-25 | Pharmalight Inc. | Method and Device for Ophthalmic Administration of Active Pharmaceutical Ingredients |
CN107106588B (zh) | 2014-10-28 | 2020-08-11 | 山口晃史 | 用于改善妊娠状态的药剂及其使用 |
CN112533599A (zh) | 2018-08-10 | 2021-03-19 | 山口晃史 | 与母体和胎儿的关系中的体液免疫相关的疾病的治疗药 |
AU2019401108A1 (en) | 2018-12-18 | 2021-07-01 | Koushi Yamaguchi | Agent for improving infertility, recurrent miscarriage, and state of pregnancy |
Family Cites Families (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3244592A (en) * | 1962-06-09 | 1966-04-05 | Arai Tadashi | Ascomycin and process for its production |
US4894366A (en) * | 1984-12-03 | 1990-01-16 | Fujisawa Pharmaceutical Company, Ltd. | Tricyclo compounds, a process for their production and a pharmaceutical composition containing the same |
JPS6317884A (ja) * | 1986-05-30 | 1988-01-25 | Fujisawa Pharmaceut Co Ltd | トリシクロ化合物 |
JPH01125394A (ja) * | 1987-11-10 | 1989-05-17 | Mect Corp | シアロシルグリセロリピッド類及びその製造方法 |
AU630866B2 (en) * | 1987-12-09 | 1992-11-12 | Fisons Plc | Macrocyclic compounds |
AU6286690A (en) * | 1989-08-18 | 1991-04-03 | Fisons Plc | Macrocyclic compounds |
KR0159766B1 (ko) * | 1989-10-16 | 1998-12-01 | 후지사와 토모키치로 | 양모제 조성물 |
DE69021833T2 (de) * | 1989-11-09 | 1996-03-21 | Sandoz Ag | Heteroatome enthaltende tricyclische Verbindungen. |
JPH05504956A (ja) * | 1990-03-12 | 1993-07-29 | 藤沢薬品工業株式会社 | トリシクロ化合物 |
JPH05507915A (ja) * | 1990-06-11 | 1993-11-11 | 藤沢薬品工業株式会社 | 特発性血小板減少性紫斑病およびバセドウ病治療薬製造のためのfk506等のマクロライド化合物の用途 |
MY110418A (en) * | 1990-07-02 | 1998-05-30 | Novartis Ag | Heteroatoms-containing tricyclic compounds. |
DE69125230T2 (de) * | 1990-09-04 | 1997-07-10 | Fujisawa Pharmaceutical Co | Tricyclische Verbindungen enthaltende Salben |
IE65341B1 (en) * | 1990-11-08 | 1995-10-18 | Fujisawa Pharmaceutical Co | Suspensions containing tricyclic compounds |
US5252732A (en) * | 1991-09-09 | 1993-10-12 | Merck & Co., Inc. | D-heteroaryl, O-alkylheteroaryl, O-alkenylheteroaryl and O-alkynylheteroarylmacrolides having immunosuppressive activity |
US5208241A (en) * | 1991-09-09 | 1993-05-04 | Merck & Co., Inc. | N-heteroaryl, n-alkylheteroaryl, n-alkenylheteroaryl and n-alkynylheteroarylmacrolides having immunosuppressive activity |
US5247076A (en) * | 1991-09-09 | 1993-09-21 | Merck & Co., Inc. | Imidazolidyl macrolides having immunosuppressive activity |
US5457194A (en) * | 1993-03-17 | 1995-10-10 | Abbott Laboratories | Substituted aliphatic amine-containing macrocyclic immunomodulators |
CN1089233C (zh) * | 1994-10-26 | 2002-08-21 | 诺瓦蒂斯有限公司 | 药物组合物 |
-
1996
- 1996-04-02 AR ARP960102027A patent/AR004480A1/es unknown
- 1996-04-03 CO CO96016454A patent/CO4750668A1/es unknown
- 1996-04-03 IL IL11781596A patent/IL117815A/xx not_active IP Right Cessation
- 1996-04-04 AU AU56453/96A patent/AU703523B2/en not_active Ceased
- 1996-04-04 US US08/930,730 patent/US5925649A/en not_active Expired - Fee Related
- 1996-04-04 NZ NZ307170A patent/NZ307170A/xx unknown
- 1996-04-04 HU HU9801993A patent/HUP9801993A3/hu unknown
- 1996-04-04 JP JP8529996A patent/JP2000505044A/ja active Pending
- 1996-04-04 CZ CZ973123A patent/CZ312397A3/cs unknown
- 1996-04-04 CA CA002216562A patent/CA2216562A1/en not_active Abandoned
- 1996-04-04 KR KR1019970706988A patent/KR19980703583A/ko not_active Application Discontinuation
- 1996-04-04 SK SK1339-97A patent/SK133997A3/sk unknown
- 1996-04-04 WO PCT/EP1996/001492 patent/WO1996031514A1/en not_active Application Discontinuation
- 1996-04-04 PL PL96322553A patent/PL322553A1/xx unknown
- 1996-04-04 TR TR97/00999T patent/TR199700999T1/xx unknown
- 1996-04-04 CN CN96193091A patent/CN1088068C/zh not_active Expired - Fee Related
- 1996-04-04 BR BR9604808A patent/BR9604808A/pt active Search and Examination
- 1996-04-04 EP EP96913486A patent/EP0819130A1/en not_active Withdrawn
-
1997
- 1997-08-27 FI FI973529A patent/FI973529A/fi unknown
- 1997-10-01 NO NO974536A patent/NO309273B1/no not_active IP Right Cessation
- 1997-10-03 MX MX9707636A patent/MX9707636A/es not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
FI973529A (fi) | 1997-11-25 |
FI973529A0 (fi) | 1997-08-27 |
WO1996031514A1 (en) | 1996-10-10 |
US5925649A (en) | 1999-07-20 |
NO974536L (no) | 1997-10-01 |
CO4750668A1 (es) | 1999-03-31 |
CN1088068C (zh) | 2002-07-24 |
KR19980703583A (ko) | 1998-11-05 |
AR004480A1 (es) | 1998-12-16 |
AU5645396A (en) | 1996-10-23 |
CZ312397A3 (cs) | 1998-01-14 |
BR9604808A (pt) | 1998-06-09 |
PL322553A1 (en) | 1998-02-02 |
CA2216562A1 (en) | 1996-10-10 |
NZ307170A (en) | 1999-03-29 |
SK133997A3 (en) | 1998-05-06 |
HUP9801993A3 (en) | 2000-04-28 |
AU703523B2 (en) | 1999-03-25 |
CN1180359A (zh) | 1998-04-29 |
EP0819130A1 (en) | 1998-01-21 |
IL117815A0 (en) | 1996-08-04 |
MX9707636A (es) | 1998-06-30 |
NO309273B1 (no) | 2001-01-08 |
NO974536D0 (no) | 1997-10-01 |
JP2000505044A (ja) | 2000-04-25 |
HUP9801993A2 (hu) | 1998-12-28 |
TR199700999T1 (xx) | 1998-01-21 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FF | Patent granted | ||
KB | Patent renewed | ||
MM9K | Patent not in force due to non-payment of renewal fees |