IL111216A - Heteroarylpiperidines their preparation and pharmaceutical compositions containing them - Google Patents
Heteroarylpiperidines their preparation and pharmaceutical compositions containing themInfo
- Publication number
- IL111216A IL111216A IL11121694A IL11121694A IL111216A IL 111216 A IL111216 A IL 111216A IL 11121694 A IL11121694 A IL 11121694A IL 11121694 A IL11121694 A IL 11121694A IL 111216 A IL111216 A IL 111216A
- Authority
- IL
- Israel
- Prior art keywords
- formula
- alk
- group
- methylpiperidine
- amino
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP93402498 | 1993-10-11 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IL111216A0 IL111216A0 (en) | 1994-12-29 |
| IL111216A true IL111216A (en) | 1999-03-12 |
Family
ID=8214753
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL11121694A IL111216A (en) | 1993-10-11 | 1994-10-10 | Heteroarylpiperidines their preparation and pharmaceutical compositions containing them |
Country Status (15)
| Country | Link |
|---|---|
| US (3) | US5502063A (OSRAM) |
| JP (1) | JPH07165754A (OSRAM) |
| KR (1) | KR950011436A (OSRAM) |
| CN (1) | CN1106400A (OSRAM) |
| AU (2) | AU687090B2 (OSRAM) |
| CA (1) | CA2133855A1 (OSRAM) |
| FI (1) | FI944751L (OSRAM) |
| HU (1) | HUT71349A (OSRAM) |
| IL (1) | IL111216A (OSRAM) |
| NO (1) | NO943826L (OSRAM) |
| NZ (1) | NZ264634A (OSRAM) |
| RU (1) | RU94036762A (OSRAM) |
| SG (1) | SG47476A1 (OSRAM) |
| TW (1) | TW274548B (OSRAM) |
| ZA (1) | ZA947924B (OSRAM) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5502063A (en) * | 1993-10-11 | 1996-03-26 | Sanofi | 1-halopyridin-4-amino-4-alkylpiperidines |
| AU3463497A (en) * | 1996-07-23 | 1998-02-10 | Yamanouchi Pharmaceutical Co., Ltd. | Novel medicinal compositions for therapeutic use |
| FR2780057B1 (fr) * | 1998-06-18 | 2002-09-13 | Sanofi Sa | Phenoxypropanolamines, procede pour leur preparation et compositions pharmaceutiques les contenant |
| US6242473B1 (en) * | 1999-01-08 | 2001-06-05 | Maxim Pharmaceuticals, Inc. | Treatment and prevention of reactive oxygen metabolite-mediated cellular damage |
| HU225894B1 (en) * | 1999-05-21 | 2007-12-28 | Abbott Lab | Heterocyclic substituted aminoazacycles useful as central nervous system agents |
| RU2168506C1 (ru) * | 1999-10-26 | 2001-06-10 | Институт нефтехимии и катализа АН РБ и УНЦ РАН | 2-(n-пиперидил)-3,5-диметилпиридин в качестве ингибитора кислотной коррозии стали |
| CA2587749A1 (en) * | 2004-12-08 | 2006-06-15 | Astellas Pharma Inc. | Piperidine derivative and process for producing the same |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4302455A (en) * | 1980-04-14 | 1981-11-24 | Merck & Co., Inc. | 2-(4-Aminopiperidino)pyrazines |
| US5001125A (en) * | 1984-03-26 | 1991-03-19 | Janssen Pharmaceutica N.V. | Anti-virally active pyridazinamines |
| US5196439A (en) * | 1987-11-27 | 1993-03-23 | Eisai Co., Ltd. | Piperidine compounds useful to treat cerebrovascular diseases |
| DE69228017D1 (de) * | 1991-03-27 | 1999-02-11 | Sanofi Sa | Verwendung von 4-Amino-1-(2-Pyridyl)Piperidinen als 5-HT3-Agonisten zur Behandlung und Verhütung von serotoninergen Dysfunktionen |
| JPH0665203A (ja) * | 1992-06-25 | 1994-03-08 | Elf Sanofi | ピペラジンのヘテロ環誘導体 |
| US5502063A (en) * | 1993-10-11 | 1996-03-26 | Sanofi | 1-halopyridin-4-amino-4-alkylpiperidines |
-
1994
- 1994-10-07 US US08/319,595 patent/US5502063A/en not_active Expired - Fee Related
- 1994-10-07 CA CA002133855A patent/CA2133855A1/en not_active Abandoned
- 1994-10-07 NZ NZ264634A patent/NZ264634A/en unknown
- 1994-10-10 FI FI944751A patent/FI944751L/fi unknown
- 1994-10-10 HU HU9402919A patent/HUT71349A/hu unknown
- 1994-10-10 IL IL11121694A patent/IL111216A/en not_active IP Right Cessation
- 1994-10-10 SG SG1996002107A patent/SG47476A1/en unknown
- 1994-10-10 RU RU94036762/04A patent/RU94036762A/ru unknown
- 1994-10-10 NO NO943826A patent/NO943826L/no unknown
- 1994-10-11 ZA ZA947924A patent/ZA947924B/xx unknown
- 1994-10-11 TW TW083109398A patent/TW274548B/zh active
- 1994-10-11 CN CN94117118A patent/CN1106400A/zh active Pending
- 1994-10-11 AU AU75745/94A patent/AU687090B2/en not_active Ceased
- 1994-10-11 KR KR1019940026020A patent/KR950011436A/ko not_active Withdrawn
- 1994-10-11 JP JP6245145A patent/JPH07165754A/ja not_active Withdrawn
-
1995
- 1995-06-06 US US08/469,511 patent/US5595994A/en not_active Expired - Fee Related
- 1995-06-06 US US08/469,523 patent/US5723611A/en not_active Expired - Fee Related
-
1998
- 1998-05-13 AU AU64881/98A patent/AU6488198A/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| CN1106400A (zh) | 1995-08-09 |
| FI944751A7 (fi) | 1995-04-12 |
| FI944751A0 (fi) | 1994-10-10 |
| US5595994A (en) | 1997-01-21 |
| KR950011436A (ko) | 1995-05-15 |
| IL111216A0 (en) | 1994-12-29 |
| RU94036762A (ru) | 1996-09-10 |
| HU9402919D0 (en) | 1995-01-30 |
| US5502063A (en) | 1996-03-26 |
| ZA947924B (en) | 1995-05-26 |
| NO943826L (no) | 1995-04-12 |
| CA2133855A1 (en) | 1995-04-12 |
| AU687090B2 (en) | 1998-02-19 |
| HUT71349A (en) | 1995-11-28 |
| AU7574594A (en) | 1995-04-27 |
| NZ264634A (en) | 1995-12-21 |
| FI944751L (fi) | 1995-04-12 |
| TW274548B (OSRAM) | 1996-04-21 |
| SG47476A1 (en) | 1998-04-17 |
| AU6488198A (en) | 1998-07-02 |
| NO943826D0 (no) | 1994-10-10 |
| JPH07165754A (ja) | 1995-06-27 |
| US5723611A (en) | 1998-03-03 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| US6544997B1 (en) | 4-(aminomethyl)-piperidine benzamides for treating gastrointestinal disorders | |
| US4912219A (en) | 2-[4-pyrimidin-2-yl amino)piperidin-1-yl]benzimidazole compound | |
| JPH0739387B2 (ja) | 新規１−ベンジル−アミノアルキル−ピロリジノン化合物及びその製造方法 | |
| EP0863141A1 (en) | Substituted heteroaromatic derivatives | |
| US20070238878A1 (en) | Process for the synthesis of 4-(3-sulfonylphenyl)-piperidines | |
| NZ230956A (en) | Piperidinyl benzimidazole derivatives | |
| JPH0733384B2 (ja) | アミノ−チアゾ−ル及びオキサゾ−ル誘導体 | |
| KR20010015532A (ko) | 아제티디닐프로필피페리딘 유도체, 그의 중간체 및타키키닌 길항제로서의 용도 | |
| KR19990077027A (ko) | 타키키닌 길항제로서의 3-아제티디닐알킬피페리딘 또는 3-아제티디닐알킬피롤리딘 | |
| PL113999B1 (en) | Process for preparing novel derivatives of 5,11-dihydro-6h-pyrido/2,3-b//1,4/benzodiazepin-6-ones | |
| US5502063A (en) | 1-halopyridin-4-amino-4-alkylpiperidines | |
| US6858629B1 (en) | Heteroaryloxy propanolamines, preparation method and pharmaceutical compositions containing same | |
| US4224333A (en) | Antihypertensive 2H-indol-2-ones | |
| US4100291A (en) | Novel 1,4-benzodioxanes | |
| SK285557B6 (sk) | Tetrahydropyridíny, spôsob ich prípravy, farmaceutické kompozície obsahujúce tieto tetrahydropyridíny a ich použitie | |
| KR100485020B1 (ko) | 옥타하이드로-2Ｈ-피리도[1,2-ａ]피라진 화합물, 이들의 제조방법 및 이들을 함유하는 약제학적 조성물 | |
| NO136713B (OSRAM) | ||
| EP0647639A1 (fr) | Hétéroarylpipéridines, procédé pour leur préparation et compositions pharmaceutiques les contenant | |
| JP2003516992A (ja) | イミダゾピリミジニル誘導体およびイミダゾピリジニル誘導体 | |
| DE60033060T2 (de) | Lineare oder zyklische Harnstoffe, Verfahren zu ihrer Herstellung und sie enthaltende pharmazeutische Zusammensetzungen | |
| WO1997028157A1 (fr) | Nouveaux derives de la piperidine substitues en position 4 par un groupe imidazolidin-2-on-1-yl-ethyl, tetrahydropyrimidin-2-on-1-yl-ethyl, et 1,3-dia-zepin-2-on-1-yl-ethyl, et leurs applications comme antagonistes des recepteurs alpha-2 adrenergiques | |
| WO1988001270A1 (en) | Pyridopyrimidinediones | |
| EP0977740A1 (en) | Methods for synthesizing 2-substituted imidazoles | |
| KR0153530B1 (ko) | 락탐 유도체의 제조 방법 | |
| EP0746556B1 (en) | Tricyclic compounds having affinity for the 5-ht1a receptor |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FF | Patent granted | ||
| RH | Patent void |