IL110994A - Process for preparing a history of 2-transformed-H3-imidazo [B-4,5] pyridine - Google Patents
Process for preparing a history of 2-transformed-H3-imidazo [B-4,5] pyridineInfo
- Publication number
- IL110994A IL110994A IL110994A IL11099494A IL110994A IL 110994 A IL110994 A IL 110994A IL 110994 A IL110994 A IL 110994A IL 11099494 A IL11099494 A IL 11099494A IL 110994 A IL110994 A IL 110994A
- Authority
- IL
- Israel
- Prior art keywords
- general formula
- alkyl
- aryl
- groups
- preparing
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CH281693 | 1993-09-17 |
Publications (2)
Publication Number | Publication Date |
---|---|
IL110994A0 IL110994A0 (en) | 1994-11-28 |
IL110994A true IL110994A (en) | 1998-02-08 |
Family
ID=4242236
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL110994A IL110994A (en) | 1993-09-17 | 1994-09-18 | Process for preparing a history of 2-transformed-H3-imidazo [B-4,5] pyridine |
Country Status (22)
Country | Link |
---|---|
US (1) | US5446160A (fr) |
EP (1) | EP0645389B1 (fr) |
JP (1) | JP3713724B2 (fr) |
KR (1) | KR950008512A (fr) |
AT (1) | ATE148702T1 (fr) |
AU (1) | AU680025B2 (fr) |
BR (1) | BR9403594A (fr) |
CA (1) | CA2131680C (fr) |
CZ (1) | CZ285489B6 (fr) |
DE (1) | DE59401760D1 (fr) |
DK (1) | DK0645389T3 (fr) |
ES (1) | ES2098089T3 (fr) |
GR (1) | GR3022500T3 (fr) |
HU (1) | HU218488B (fr) |
IL (1) | IL110994A (fr) |
PL (1) | PL305067A1 (fr) |
RU (1) | RU94033473A (fr) |
SI (1) | SI0645389T1 (fr) |
SK (1) | SK111494A3 (fr) |
TR (1) | TR27788A (fr) |
TW (1) | TW410225B (fr) |
ZA (1) | ZA947189B (fr) |
Families Citing this family (34)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9312853D0 (en) | 1993-06-22 | 1993-08-04 | Euro Celtique Sa | Chemical compounds |
US5591776A (en) | 1994-06-24 | 1997-01-07 | Euro-Celtique, S.A. | Pheynl or benzyl-substituted rolipram-based compounds for and method of inhibiting phosphodiesterase IV |
US5922751A (en) | 1994-06-24 | 1999-07-13 | Euro-Celtique, S.A. | Aryl pyrazole compound for inhibiting phosphodiesterase IV and methods of using same |
US6166041A (en) | 1995-10-11 | 2000-12-26 | Euro-Celtique, S.A. | 2-heteroaryl and 2-heterocyclic benzoxazoles as PDE IV inhibitors for the treatment of asthma |
US6075016A (en) | 1996-04-10 | 2000-06-13 | Euro-Celtique S.A. | 6,5-fused aromatic ring systems having enhanced phosphodiesterase IV inhibitory activity |
HRP980375A2 (en) | 1997-07-03 | 1999-04-30 | Argyrios Georgios Arvanitis | Imidazopyrimidines and imidazopyridines for the treatment of neurological disorders |
US6365589B1 (en) | 1998-07-02 | 2002-04-02 | Bristol-Myers Squibb Pharma Company | Imidazo-pyridines, -pyridazines, and -triazines as corticotropin releasing factor antagonists |
US6124463A (en) * | 1998-07-02 | 2000-09-26 | Dupont Pharmaceuticals | Benzimidazoles as corticotropin release factor antagonists |
US7045529B2 (en) * | 1999-12-17 | 2006-05-16 | Bristol-Myers Squibb Company | Imidazopyrimidinyl and imidazopyri dinyl derivatives |
MXPA06001669A (es) | 2003-08-12 | 2006-04-28 | 3M Innovative Properties Co | Compuestos que contienen imidazo-oxima sustituidos. |
US7897597B2 (en) | 2003-08-27 | 2011-03-01 | 3M Innovative Properties Company | Aryloxy and arylalkyleneoxy substituted imidazoquinolines |
WO2005023190A2 (fr) | 2003-09-05 | 2005-03-17 | 3M Innovative Properties Company | Traitement pour le lymphome a cellules b cd5+ |
US7544697B2 (en) | 2003-10-03 | 2009-06-09 | Coley Pharmaceutical Group, Inc. | Pyrazolopyridines and analogs thereof |
US8871782B2 (en) | 2003-10-03 | 2014-10-28 | 3M Innovative Properties Company | Alkoxy substituted imidazoquinolines |
CA2545825A1 (fr) | 2003-11-14 | 2005-06-02 | 3M Innovative Properties Company | Composes d'un anneau d'imidazo substitue par hydroxylamine |
CA2545774A1 (fr) | 2003-11-14 | 2005-06-02 | 3M Innovative Properties Company | Composes d'un anneau d'imidazo substitues par oxime |
AU2004293078B2 (en) | 2003-11-25 | 2012-01-19 | 3M Innovative Properties Company | Substituted imidazo ring systems and methods |
EP1701955A1 (fr) | 2003-12-29 | 2006-09-20 | 3M Innovative Properties Company | Imidazoquinolines a substitution arylalcenyle et arylalkynyle |
CA2551399A1 (fr) | 2003-12-30 | 2005-07-21 | 3M Innovative Properties Company | Sulfonamides d'imidazoquinolinyle, d'imidazopyridinyle et d'imidazonaphtyridinyle |
EP1730143A2 (fr) | 2004-03-24 | 2006-12-13 | 3M Innovative Properties Company | Imidazopyridines, imidazoquinolines, et imidazonaphthyridines a substitution amide |
WO2005123080A2 (fr) | 2004-06-15 | 2005-12-29 | 3M Innovative Properties Company | Imidazoquinolines et imidazonaphthyridines substituees par un heterocyclyle contenant un azote |
WO2006038923A2 (fr) | 2004-06-18 | 2006-04-13 | 3M Innovative Properties Company | Imidazonaphthyridines substituees par aryle |
WO2006009826A1 (fr) | 2004-06-18 | 2006-01-26 | 3M Innovative Properties Company | Thiazoloquinolines et thiazolonaphtyridines substitues par aryloxy et arylalkyleneoxy |
US7915281B2 (en) | 2004-06-18 | 2011-03-29 | 3M Innovative Properties Company | Isoxazole, dihydroisoxazole, and oxadiazole substituted imidazo ring compounds and method |
JP5313502B2 (ja) | 2004-12-30 | 2013-10-09 | スリーエム イノベイティブ プロパティズ カンパニー | 置換キラル縮合[1,2]イミダゾ[4,5−c]環状化合物 |
AU2005322898B2 (en) | 2004-12-30 | 2011-11-24 | 3M Innovative Properties Company | Chiral fused (1,2)imidazo(4,5-c) ring compounds |
AU2006210392A1 (en) | 2005-02-04 | 2006-08-10 | Coley Pharmaceutical Group, Inc. | Aqueous gel formulations containing immune response modifiers |
JP2008530113A (ja) | 2005-02-11 | 2008-08-07 | コーリー ファーマシューティカル グループ,インコーポレイテッド | オキシムおよびヒドロキシラミン置換イミダゾ[4,5−c]環化合物および方法 |
WO2006121528A2 (fr) | 2005-04-01 | 2006-11-16 | Coley Pharmaceutical Group, Inc. | Fermeture de cycle et procedes et produits intermediaires associes |
AU2006232377A1 (en) | 2005-04-01 | 2006-10-12 | Coley Pharmaceutical Group, Inc. | Pyrazolopyridine-1,4-diamines and analogs thereof |
WO2006107851A1 (fr) | 2005-04-01 | 2006-10-12 | Coley Pharmaceutical Group, Inc. | Composes cycliques 1-pyrazolo[3,4-c] substitues comme modulateurs de la biosynthese de cytokine destines au traitement d'infections virales et de maladies neoplastiques |
EP1937683A4 (fr) * | 2005-09-23 | 2010-08-25 | Coley Pharm Group Inc | Procede de preparation de 1h-imidazoý4,5-c¨pyridines et d'analogues de ceux-ci |
US7906506B2 (en) | 2006-07-12 | 2011-03-15 | 3M Innovative Properties Company | Substituted chiral fused [1,2] imidazo [4,5-c] ring compounds and methods |
US20080139608A1 (en) * | 2006-12-06 | 2008-06-12 | Universiteit Leiden | 2,6,8, Trisubstituted 1-deazapurines and their different uses |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3324115A1 (de) * | 1983-07-05 | 1985-01-17 | Dr. Karl Thomae Gmbh, 7950 Biberach | Neue imidazole, ihre herstellung und diese verbindungen enthaltende arzneimittel |
FR2643903A1 (fr) * | 1989-03-03 | 1990-09-07 | Union Pharma Scient Appl | Nouveaux derives de benzimidazole, leurs procedes de preparation, intermediaires de synthese, compositions pharmaceutiques les contenant, utiles notamment pour le traitement des maladies cardiovasculaires, et des ulceres duodenaux |
US5223499A (en) * | 1989-05-30 | 1993-06-29 | Merck & Co., Inc. | 6-amino substituted imidazo[4,5-bipyridines as angiotensin II antagonists |
US5240938A (en) * | 1991-02-13 | 1993-08-31 | Merck & Co., Inc. | Angiotensin II antagonists incorporating a substituted pyridoimidazolyl ring |
US5066654A (en) * | 1990-10-22 | 1991-11-19 | A. H. Robins Company, Incorporated | 2-aryl-3-heterocyclicmethyl-3H-imidazo[4,5-b]pyridines as anxiolytics and anticonvulsants |
US5128327A (en) * | 1991-03-25 | 1992-07-07 | Merck & Co., Inc. | Angiotensin II antagonists incorporating a nitrogen containing six membered ring heterocycle |
-
1994
- 1994-09-08 CA CA002131680A patent/CA2131680C/fr not_active Expired - Fee Related
- 1994-09-13 JP JP21837194A patent/JP3713724B2/ja not_active Expired - Fee Related
- 1994-09-15 DK DK94114551.8T patent/DK0645389T3/da active
- 1994-09-15 TR TR00943/94A patent/TR27788A/xx unknown
- 1994-09-15 SI SI9430048T patent/SI0645389T1/xx not_active IP Right Cessation
- 1994-09-15 EP EP94114551A patent/EP0645389B1/fr not_active Expired - Lifetime
- 1994-09-15 KR KR1019940023449A patent/KR950008512A/ko not_active Application Discontinuation
- 1994-09-15 ES ES94114551T patent/ES2098089T3/es not_active Expired - Lifetime
- 1994-09-15 AT AT94114551T patent/ATE148702T1/de not_active IP Right Cessation
- 1994-09-15 DE DE59401760T patent/DE59401760D1/de not_active Expired - Fee Related
- 1994-09-16 PL PL94305067A patent/PL305067A1/xx unknown
- 1994-09-16 HU HU9402662A patent/HU218488B/hu not_active IP Right Cessation
- 1994-09-16 ZA ZA947189A patent/ZA947189B/xx unknown
- 1994-09-16 BR BR9403594A patent/BR9403594A/pt not_active Application Discontinuation
- 1994-09-16 CZ CZ942266A patent/CZ285489B6/cs not_active IP Right Cessation
- 1994-09-16 AU AU73058/94A patent/AU680025B2/en not_active Ceased
- 1994-09-16 SK SK1114-94A patent/SK111494A3/sk unknown
- 1994-09-16 RU RU94033473/04A patent/RU94033473A/ru unknown
- 1994-09-18 IL IL110994A patent/IL110994A/en not_active IP Right Cessation
- 1994-09-19 US US08/308,448 patent/US5446160A/en not_active Expired - Lifetime
- 1994-10-08 TW TW083109361A patent/TW410225B/zh not_active IP Right Cessation
-
1997
- 1997-02-06 GR GR970400075T patent/GR3022500T3/el unknown
Also Published As
Publication number | Publication date |
---|---|
SK111494A3 (en) | 1995-06-07 |
JP3713724B2 (ja) | 2005-11-09 |
TR27788A (tr) | 1995-08-29 |
DK0645389T3 (da) | 1997-03-10 |
GR3022500T3 (en) | 1997-05-31 |
AU680025B2 (en) | 1997-07-17 |
SI0645389T1 (en) | 1997-10-31 |
HU9402662D0 (en) | 1994-11-28 |
HUT68250A (en) | 1995-06-28 |
US5446160A (en) | 1995-08-29 |
BR9403594A (pt) | 1995-05-16 |
AU7305894A (en) | 1995-03-30 |
CA2131680C (fr) | 2006-11-07 |
RU94033473A (ru) | 1996-08-10 |
KR950008512A (ko) | 1995-04-17 |
DE59401760D1 (de) | 1997-03-20 |
EP0645389B1 (fr) | 1997-02-05 |
ES2098089T3 (es) | 1997-04-16 |
HU218488B (hu) | 2000-09-28 |
EP0645389A1 (fr) | 1995-03-29 |
JPH07179465A (ja) | 1995-07-18 |
ZA947189B (en) | 1995-05-12 |
CA2131680A1 (fr) | 1995-03-18 |
TW410225B (en) | 2000-11-01 |
CZ285489B6 (cs) | 1999-08-11 |
ATE148702T1 (de) | 1997-02-15 |
PL305067A1 (en) | 1995-03-20 |
CZ226694A3 (en) | 1995-04-12 |
IL110994A0 (en) | 1994-11-28 |
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Legal Events
Date | Code | Title | Description |
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FF | Patent granted | ||
KB | Patent renewed | ||
KB | Patent renewed | ||
KB | Patent renewed | ||
KB | Patent renewed | ||
MM9K | Patent not in force due to non-payment of renewal fees |