SI0645389T1 - Process for the production of imidazopyridines - Google Patents

Process for the production of imidazopyridines

Info

Publication number
SI0645389T1
SI0645389T1 SI9430048T SI9430048T SI0645389T1 SI 0645389 T1 SI0645389 T1 SI 0645389T1 SI 9430048 T SI9430048 T SI 9430048T SI 9430048 T SI9430048 T SI 9430048T SI 0645389 T1 SI0645389 T1 SI 0645389T1
Authority
SI
Slovenia
Prior art keywords
imidazopyridines
image
production
preparation
general formula
Prior art date
Application number
SI9430048T
Other languages
English (en)
Inventor
Gerhard Dr Stucky
Renu Dr Imwinkelried
Original Assignee
Lonza Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lonza Ag filed Critical Lonza Ag
Publication of SI0645389T1 publication Critical patent/SI0645389T1/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
SI9430048T 1993-09-17 1994-09-15 Process for the production of imidazopyridines SI0645389T1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH281693 1993-09-17
EP94114551A EP0645389B1 (fr) 1993-09-17 1994-09-15 Procédé pour la préparation de derivés des imidazopyridines

Publications (1)

Publication Number Publication Date
SI0645389T1 true SI0645389T1 (en) 1997-10-31

Family

ID=4242236

Family Applications (1)

Application Number Title Priority Date Filing Date
SI9430048T SI0645389T1 (en) 1993-09-17 1994-09-15 Process for the production of imidazopyridines

Country Status (22)

Country Link
US (1) US5446160A (fr)
EP (1) EP0645389B1 (fr)
JP (1) JP3713724B2 (fr)
KR (1) KR950008512A (fr)
AT (1) ATE148702T1 (fr)
AU (1) AU680025B2 (fr)
BR (1) BR9403594A (fr)
CA (1) CA2131680C (fr)
CZ (1) CZ285489B6 (fr)
DE (1) DE59401760D1 (fr)
DK (1) DK0645389T3 (fr)
ES (1) ES2098089T3 (fr)
GR (1) GR3022500T3 (fr)
HU (1) HU218488B (fr)
IL (1) IL110994A (fr)
PL (1) PL305067A1 (fr)
RU (1) RU94033473A (fr)
SI (1) SI0645389T1 (fr)
SK (1) SK111494A3 (fr)
TR (1) TR27788A (fr)
TW (1) TW410225B (fr)
ZA (1) ZA947189B (fr)

Families Citing this family (34)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9312853D0 (en) 1993-06-22 1993-08-04 Euro Celtique Sa Chemical compounds
US5591776A (en) 1994-06-24 1997-01-07 Euro-Celtique, S.A. Pheynl or benzyl-substituted rolipram-based compounds for and method of inhibiting phosphodiesterase IV
US5922751A (en) 1994-06-24 1999-07-13 Euro-Celtique, S.A. Aryl pyrazole compound for inhibiting phosphodiesterase IV and methods of using same
US6166041A (en) 1995-10-11 2000-12-26 Euro-Celtique, S.A. 2-heteroaryl and 2-heterocyclic benzoxazoles as PDE IV inhibitors for the treatment of asthma
US6075016A (en) 1996-04-10 2000-06-13 Euro-Celtique S.A. 6,5-fused aromatic ring systems having enhanced phosphodiesterase IV inhibitory activity
US6143743A (en) 1997-07-03 2000-11-07 Dupont Pharmaceuticals Company Imidazopyrimidines and imidazopyridines for the treatment of neurological disorders
US6365589B1 (en) 1998-07-02 2002-04-02 Bristol-Myers Squibb Pharma Company Imidazo-pyridines, -pyridazines, and -triazines as corticotropin releasing factor antagonists
US6124463A (en) * 1998-07-02 2000-09-26 Dupont Pharmaceuticals Benzimidazoles as corticotropin release factor antagonists
EP1244666A1 (fr) * 1999-12-17 2002-10-02 Bristol-Myers Squibb Pharma Company Derives imidazopyrimidinyles et imidazopyridinyles
EP1653914A4 (fr) 2003-08-12 2008-10-29 3M Innovative Properties Co Composes contenant une structure imidazo a substitution oxime
NZ545412A (en) 2003-08-27 2008-12-24 Coley Pharm Group Inc Aryloxy and arylalkyleneoxy substituted imidazoquinolines
CA2537763A1 (fr) 2003-09-05 2005-03-17 3M Innovative Properties Company Traitement pour le lymphome a cellules b cd5<sp>+</sp>
BRPI0414856A (pt) 2003-10-03 2006-11-21 3M Innovative Properties Co imidazoquinolinas alcóxi-substituìdas
US7544697B2 (en) 2003-10-03 2009-06-09 Coley Pharmaceutical Group, Inc. Pyrazolopyridines and analogs thereof
CN1906193A (zh) 2003-11-14 2007-01-31 3M创新有限公司 肟取代的咪唑环化合物
CA2545825A1 (fr) 2003-11-14 2005-06-02 3M Innovative Properties Company Composes d'un anneau d'imidazo substitue par hydroxylamine
MXPA06005910A (es) 2003-11-25 2006-08-23 3M Innovative Properties Co Sistemas de anillo imidazo sustituido y metodos.
WO2005066170A1 (fr) 2003-12-29 2005-07-21 3M Innovative Properties Company Imidazoquinolines a substitution arylalcenyle et arylalkynyle
JP2007517044A (ja) 2003-12-30 2007-06-28 スリーエム イノベイティブ プロパティズ カンパニー イミダゾキノリニル、イミダゾピリジニル、およびイミダゾナフチリジニルスルホンアミド
AU2005228150A1 (en) 2004-03-24 2005-10-13 3M Innovative Properties Company Amide substituted imidazopyridines, imidazoquinolines, and imidazonaphthyridines
US8017779B2 (en) 2004-06-15 2011-09-13 3M Innovative Properties Company Nitrogen containing heterocyclyl substituted imidazoquinolines and imidazonaphthyridines
US7897609B2 (en) 2004-06-18 2011-03-01 3M Innovative Properties Company Aryl substituted imidazonaphthyridines
WO2006065280A2 (fr) 2004-06-18 2006-06-22 3M Innovative Properties Company Composes a noyau imidazo a substitutif d'isoxazole, de dihydroisoxazole et d'oxadiazole
US8026366B2 (en) 2004-06-18 2011-09-27 3M Innovative Properties Company Aryloxy and arylalkyleneoxy substituted thiazoloquinolines and thiazolonaphthyridines
EP1831226B1 (fr) 2004-12-30 2012-08-08 3M Innovative Properties Company Composes chiraux tetracycliques incitant la biosynthese d'interferon
JP5313502B2 (ja) 2004-12-30 2013-10-09 スリーエム イノベイティブ プロパティズ カンパニー 置換キラル縮合[1,2]イミダゾ[4,5−c]環状化合物
US9248127B2 (en) 2005-02-04 2016-02-02 3M Innovative Properties Company Aqueous gel formulations containing immune response modifiers
CA2597587A1 (fr) 2005-02-11 2006-08-17 Coley Pharmaceutical Group, Inc. Composes cycliques imidazo[4,5-c] substitues par oxime et hydroxylamine et procedes associes
JP2008538550A (ja) 2005-04-01 2008-10-30 コーリー ファーマシューティカル グループ,インコーポレイテッド ウイルス感染および腫瘍性疾患を処置するためのサイトカイン生合成の調節因子としての1−置換ピラゾロ(3,4−c)環状化合物
AU2006232377A1 (en) 2005-04-01 2006-10-12 Coley Pharmaceutical Group, Inc. Pyrazolopyridine-1,4-diamines and analogs thereof
AU2006244635A1 (en) * 2005-04-01 2006-11-16 Coley Pharmaceutical Group, Inc. Ring closing and related methods and intermediates
CA2623541A1 (fr) * 2005-09-23 2007-03-29 Coley Pharmaceutical Group, Inc. Procede de preparation de 1h-imidazo[4,5-c]pyridines et d'analogues de ceux-ci
US7906506B2 (en) 2006-07-12 2011-03-15 3M Innovative Properties Company Substituted chiral fused [1,2] imidazo [4,5-c] ring compounds and methods
US20080139608A1 (en) * 2006-12-06 2008-06-12 Universiteit Leiden 2,6,8, Trisubstituted 1-deazapurines and their different uses

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3324115A1 (de) * 1983-07-05 1985-01-17 Dr. Karl Thomae Gmbh, 7950 Biberach Neue imidazole, ihre herstellung und diese verbindungen enthaltende arzneimittel
FR2643903A1 (fr) * 1989-03-03 1990-09-07 Union Pharma Scient Appl Nouveaux derives de benzimidazole, leurs procedes de preparation, intermediaires de synthese, compositions pharmaceutiques les contenant, utiles notamment pour le traitement des maladies cardiovasculaires, et des ulceres duodenaux
US5223499A (en) * 1989-05-30 1993-06-29 Merck & Co., Inc. 6-amino substituted imidazo[4,5-bipyridines as angiotensin II antagonists
US5240938A (en) * 1991-02-13 1993-08-31 Merck & Co., Inc. Angiotensin II antagonists incorporating a substituted pyridoimidazolyl ring
US5066654A (en) * 1990-10-22 1991-11-19 A. H. Robins Company, Incorporated 2-aryl-3-heterocyclicmethyl-3H-imidazo[4,5-b]pyridines as anxiolytics and anticonvulsants
US5128327A (en) * 1991-03-25 1992-07-07 Merck & Co., Inc. Angiotensin II antagonists incorporating a nitrogen containing six membered ring heterocycle

Also Published As

Publication number Publication date
RU94033473A (ru) 1996-08-10
CA2131680A1 (fr) 1995-03-18
CZ285489B6 (cs) 1999-08-11
ES2098089T3 (es) 1997-04-16
CA2131680C (fr) 2006-11-07
TW410225B (en) 2000-11-01
TR27788A (tr) 1995-08-29
IL110994A (en) 1998-02-08
SK111494A3 (en) 1995-06-07
JP3713724B2 (ja) 2005-11-09
ZA947189B (en) 1995-05-12
US5446160A (en) 1995-08-29
HU218488B (hu) 2000-09-28
HUT68250A (en) 1995-06-28
JPH07179465A (ja) 1995-07-18
EP0645389B1 (fr) 1997-02-05
GR3022500T3 (en) 1997-05-31
KR950008512A (ko) 1995-04-17
HU9402662D0 (en) 1994-11-28
PL305067A1 (en) 1995-03-20
AU7305894A (en) 1995-03-30
DE59401760D1 (de) 1997-03-20
IL110994A0 (en) 1994-11-28
BR9403594A (pt) 1995-05-16
AU680025B2 (en) 1997-07-17
EP0645389A1 (fr) 1995-03-29
DK0645389T3 (da) 1997-03-10
CZ226694A3 (en) 1995-04-12
ATE148702T1 (de) 1997-02-15

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Effective date: 20100531