IL110964A - כלורידים של 4,3,2,1- טלרהידרוקינולין -8-חומצה סולפונית וחומצותיהם, הכנתם ושימושם כמתווכים סינטיים - Google Patents

כלורידים של 4,3,2,1- טלרהידרוקינולין -8-חומצה סולפונית וחומצותיהם, הכנתם ושימושם כמתווכים סינטיים

Info

Publication number
IL110964A
IL110964A IL11096494A IL11096494A IL110964A IL 110964 A IL110964 A IL 110964A IL 11096494 A IL11096494 A IL 11096494A IL 11096494 A IL11096494 A IL 11096494A IL 110964 A IL110964 A IL 110964A
Authority
IL
Israel
Prior art keywords
methyl
formula
tetrahydroquinoline
mixture
compound
Prior art date
Application number
IL11096494A
Other languages
English (en)
Other versions
IL110964A0 (en
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Publication of IL110964A0 publication Critical patent/IL110964A0/xx
Publication of IL110964A publication Critical patent/IL110964A/he

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/04—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to the ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/36—Sulfur atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Quinoline Compounds (AREA)
IL11096494A 1993-09-14 1994-09-13 כלורידים של 4,3,2,1- טלרהידרוקינולין -8-חומצה סולפונית וחומצותיהם, הכנתם ושימושם כמתווכים סינטיים IL110964A (he)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9310905A FR2710061B1 (fr) 1993-09-14 1993-09-14 Acides et chlorures d'acides 1,2,3, 4-tétrahydroquinoléine-8-sulfoniques, et leur utilisation comme intermédiaires de synthèse.

Publications (2)

Publication Number Publication Date
IL110964A0 IL110964A0 (en) 1994-11-28
IL110964A true IL110964A (he) 1998-09-24

Family

ID=9450828

Family Applications (1)

Application Number Title Priority Date Filing Date
IL11096494A IL110964A (he) 1993-09-14 1994-09-13 כלורידים של 4,3,2,1- טלרהידרוקינולין -8-חומצה סולפונית וחומצותיהם, הכנתם ושימושם כמתווכים סינטיים

Country Status (8)

Country Link
US (1) US5552410A (he)
EP (1) EP0643046A1 (he)
JP (1) JPH07149729A (he)
KR (1) KR950008482A (he)
CA (1) CA2131764A1 (he)
FI (1) FI944227A (he)
FR (1) FR2710061B1 (he)
IL (1) IL110964A (he)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5840733A (en) * 1996-07-01 1998-11-24 Redcell, Canada, Inc. Methods and compositions for producing novel conjugates of thrombin inhibitors and endogenous carriers resulting in anti-thrombins with extended lifetimes
BRPI0512236A (pt) 2004-06-18 2008-02-19 Wyeth Corp processos para a preparação de 6-alquil-5-arilsulfonil-diidrofenantridinas
EP2824187A1 (en) * 2013-07-09 2015-01-14 Euticals S.P.A. Biocatalyzed synthesis of the optically pure (R) and (S) 3-methyl-1,2,3,4-tetrahydroquinoline and their use as chiral synthons for the preparation of the antithrombotic (21R)- and (21S)-argatroban

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE48623B1 (en) * 1978-08-31 1985-03-20 Mitsubishi Chem Ind Alpha-(n-arylsulfonyl-l-argininamides,processes for their preparation and pharmaceutical compositions containing these substances
DE3337569A1 (de) * 1983-10-15 1985-04-25 Basf Ag, 6700 Ludwigshafen Verfahren zur herstellung von chinolinen
FR2689130B1 (fr) * 1992-03-30 1994-05-27 Synthelabo Derives de 1-[2 (arylsulfonylamino)ethyl-1-oxo] piperidine, leur preparation et leur application en therapeutique.

Also Published As

Publication number Publication date
FR2710061A1 (fr) 1995-03-24
FI944227A (fi) 1995-03-15
IL110964A0 (en) 1994-11-28
FI944227A0 (fi) 1994-09-13
CA2131764A1 (fr) 1995-03-15
US5552410A (en) 1996-09-03
FR2710061B1 (fr) 1995-12-29
EP0643046A1 (fr) 1995-03-15
JPH07149729A (ja) 1995-06-13
KR950008482A (ko) 1995-04-17

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