IL109750A - Substituted 2-hydroxy-3- £1-(1h-imidazol-4-yl) alkyl|- benzenecarboximidamides, their preparation and ophthalmic conpositions containing them - Google Patents

Substituted 2-hydroxy-3- £1-(1h-imidazol-4-yl) alkyl|- benzenecarboximidamides, their preparation and ophthalmic conpositions containing them

Info

Publication number
IL109750A
IL109750A IL109750A IL10975094A IL109750A IL 109750 A IL109750 A IL 109750A IL 109750 A IL109750 A IL 109750A IL 10975094 A IL10975094 A IL 10975094A IL 109750 A IL109750 A IL 109750A
Authority
IL
Israel
Prior art keywords
imidazol
hydroxy
alkyl
benzenecarboximidamide
formula
Prior art date
Application number
IL109750A
Other languages
English (en)
Other versions
IL109750A0 (en
Original Assignee
Ucb Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ucb Sa filed Critical Ucb Sa
Publication of IL109750A0 publication Critical patent/IL109750A0/xx
Publication of IL109750A publication Critical patent/IL109750A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Treatments For Attaching Organic Compounds To Fibrous Goods (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
IL109750A 1993-05-27 1994-05-24 Substituted 2-hydroxy-3- £1-(1h-imidazol-4-yl) alkyl|- benzenecarboximidamides, their preparation and ophthalmic conpositions containing them IL109750A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB939310965A GB9310965D0 (en) 1993-05-27 1993-05-27 2-hydroxy-3-(1h-imidazol-4-yl)alkyl)benzenecarboximidamides

Publications (2)

Publication Number Publication Date
IL109750A0 IL109750A0 (en) 1994-08-26
IL109750A true IL109750A (en) 1998-06-15

Family

ID=10736226

Family Applications (1)

Application Number Title Priority Date Filing Date
IL109750A IL109750A (en) 1993-05-27 1994-05-24 Substituted 2-hydroxy-3- £1-(1h-imidazol-4-yl) alkyl|- benzenecarboximidamides, their preparation and ophthalmic conpositions containing them

Country Status (21)

Country Link
US (1) US5385927A (xx)
EP (1) EP0626372B1 (xx)
JP (1) JPH0770082A (xx)
AT (1) ATE198196T1 (xx)
AU (1) AU673422B2 (xx)
CA (1) CA2124289A1 (xx)
CZ (1) CZ287136B6 (xx)
DE (1) DE69426433D1 (xx)
FI (1) FI942390A (xx)
GB (1) GB9310965D0 (xx)
HU (1) HUT67813A (xx)
IL (1) IL109750A (xx)
MY (1) MY111216A (xx)
NO (1) NO303824B1 (xx)
NZ (1) NZ260588A (xx)
PL (1) PL175970B1 (xx)
RU (1) RU2125557C1 (xx)
SG (1) SG42791A1 (xx)
SK (1) SK60394A3 (xx)
TW (1) TW263500B (xx)
ZA (1) ZA943651B (xx)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9521680D0 (en) * 1995-10-23 1996-01-03 Orion Yhtymo Oy New use of imidazole derivatives
AU3496297A (en) * 1996-06-25 1998-01-14 Eli Lilly And Company Anticoagulant agents
US6200967B1 (en) 1996-06-25 2001-03-13 Eli Lilly And Company Anticoagulant agents
US7902247B2 (en) * 2008-01-09 2011-03-08 Allergan, Inc. Substituted-aryl-2-phenylethyl-1H-imidazole compounds as subtype selective modulators of alpha 2B and/or alpha 2C adrenergic receptors
EP2196461A1 (de) 2008-12-15 2010-06-16 Bayer CropScience AG 4-Amino-1,2,3-benzoxathiazin-Derivate als Pestizide

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8626287D0 (en) * 1986-11-04 1986-12-03 Ucb Sa Substituted 1h-imidazoles
GB8810067D0 (en) * 1988-04-28 1988-06-02 Ucb Sa Substituted 1-(1h-imidazol-4-yl)alkyl-benzamides
FI98815C (fi) * 1990-11-30 1997-08-25 Santen Oy Menetelmä uusien, farmakologisesti käyttökelpoisten bispilokarpiinihapon esterijohdannaisten valmistamiseksi

Also Published As

Publication number Publication date
HUT67813A (en) 1995-05-29
NO303824B1 (no) 1998-09-07
NO941932D0 (no) 1994-05-25
NZ260588A (en) 1995-09-26
US5385927A (en) 1995-01-31
IL109750A0 (en) 1994-08-26
GB9310965D0 (en) 1993-07-14
DE69426433D1 (de) 2001-01-25
FI942390A0 (fi) 1994-05-24
EP0626372B1 (fr) 2000-12-20
TW263500B (xx) 1995-11-21
AU673422B2 (en) 1996-11-07
CA2124289A1 (en) 1994-11-28
CZ124794A3 (en) 1994-12-15
FI942390A (fi) 1994-11-28
RU2125557C1 (ru) 1999-01-27
EP0626372A1 (fr) 1994-11-30
MY111216A (en) 1999-09-30
ATE198196T1 (de) 2001-01-15
JPH0770082A (ja) 1995-03-14
SK60394A3 (en) 1995-07-11
PL175970B1 (pl) 1999-03-31
SG42791A1 (en) 1997-10-17
HU9401574D0 (en) 1994-08-29
ZA943651B (en) 1995-01-26
CZ287136B6 (en) 2000-09-13
AU6330394A (en) 1994-12-01
NO941932L (no) 1994-11-28

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Legal Events

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MM9K Patent not in force due to non-payment of renewal fees