IL102503A - History of Alkanamine of 6-Oxoazepino] CD-5,4,3 [Indole, their preparation and pharmaceutical preparations containing them - Google Patents

History of Alkanamine of 6-Oxoazepino] CD-5,4,3 [Indole, their preparation and pharmaceutical preparations containing them

Info

Publication number
IL102503A
IL102503A IL10250392A IL10250392A IL102503A IL 102503 A IL102503 A IL 102503A IL 10250392 A IL10250392 A IL 10250392A IL 10250392 A IL10250392 A IL 10250392A IL 102503 A IL102503 A IL 102503A
Authority
IL
Israel
Prior art keywords
compounds
group
lower alkyl
general formula
formula
Prior art date
Application number
IL10250392A
Other languages
English (en)
Hebrew (he)
Other versions
IL102503A0 (en
Original Assignee
Kali Chimie Pharma Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kali Chimie Pharma Gmbh filed Critical Kali Chimie Pharma Gmbh
Publication of IL102503A0 publication Critical patent/IL102503A0/xx
Publication of IL102503A publication Critical patent/IL102503A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/06Peri-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/06Antimigraine agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Nutrition Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
IL10250392A 1991-07-31 1992-07-15 History of Alkanamine of 6-Oxoazepino] CD-5,4,3 [Indole, their preparation and pharmaceutical preparations containing them IL102503A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4125292A DE4125292A1 (de) 1991-07-31 1991-07-31 6-oxo-azepinoindol-verbindungen sowie verfahren und zwischenprodukte zu ihrer herstellung und diese verbindungen enthaltende arzneimittel

Publications (2)

Publication Number Publication Date
IL102503A0 IL102503A0 (en) 1993-01-14
IL102503A true IL102503A (en) 1995-12-31

Family

ID=6437366

Family Applications (1)

Application Number Title Priority Date Filing Date
IL10250392A IL102503A (en) 1991-07-31 1992-07-15 History of Alkanamine of 6-Oxoazepino] CD-5,4,3 [Indole, their preparation and pharmaceutical preparations containing them

Country Status (21)

Country Link
US (1) US5272143A (no)
EP (1) EP0525584B1 (no)
JP (1) JP3174158B2 (no)
KR (1) KR930002353A (no)
CN (2) CN1069733A (no)
AT (1) ATE161012T1 (no)
AU (1) AU649153B2 (no)
CA (1) CA2075102A1 (no)
CZ (1) CZ239392A3 (no)
DE (2) DE4125292A1 (no)
ES (1) ES2110454T3 (no)
FI (1) FI923440A (no)
HU (2) HU211105B (no)
IE (1) IE922310A1 (no)
IL (1) IL102503A (no)
MX (1) MX9204457A (no)
NO (1) NO300375B1 (no)
NZ (1) NZ243715A (no)
RU (1) RU2078765C1 (no)
TW (1) TW207541B (no)
ZA (1) ZA925093B (no)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5414130A (en) * 1993-12-23 1995-05-09 The Dow Chemical Company Process for the preparation of diaminoresorcinol
EE05006B1 (et) 1999-01-11 2008-04-15 Agouron Pharmaceuticals, Inc. Polü(ADP-riboos)polümeraaside tritsüklilised inhibiitorid ja neid sisaldavad farmatseutilised kompositsioonid
ECSP003637A (es) 1999-08-31 2002-03-25 Agouron Pharma Inhibidores triciclicos de poli (adp-ribosa) polimerasas
JP5465241B2 (ja) 2008-05-29 2014-04-09 アルバニー モレキュラー リサーチ, インコーポレイテッド 5−ht3受容体調節物質ならびにその作製方法および使用
SG10201406805RA (en) * 2010-02-12 2014-11-27 Pfizer Salts and polymorphs of 8-fluoro-2-{4-[(methylamino}methyl]phenyl}-1,3,4,5-tetrahydro-6h-azepino[5,4,3-cd]indol-6-one
US10513515B2 (en) 2017-08-25 2019-12-24 Biotheryx, Inc. Ether compounds and uses thereof
US11236103B2 (en) 2018-07-27 2022-02-01 Biotheryx, Inc. Bifunctional compounds
US11897930B2 (en) 2020-04-28 2024-02-13 Anwita Biosciences, Inc. Interleukin-2 polypeptides and fusion proteins thereof, and their pharmaceutical compositions and therapeutic applications

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4910193A (en) * 1985-12-16 1990-03-20 Sandoz Ltd. Treatment of gastrointestinal disorders

Also Published As

Publication number Publication date
DE4125292A1 (de) 1993-02-04
HU210217A9 (en) 1995-02-28
JP3174158B2 (ja) 2001-06-11
AU649153B2 (en) 1994-05-12
JPH05202052A (ja) 1993-08-10
IL102503A0 (en) 1993-01-14
ATE161012T1 (de) 1997-12-15
MX9204457A (es) 1993-05-01
ZA925093B (en) 1993-04-28
HU211105B (en) 1995-10-30
NO300375B1 (no) 1997-05-20
HU9202430D0 (en) 1992-10-28
CN1069733A (zh) 1993-03-10
HUT65453A (en) 1994-06-28
FI923440A (fi) 1993-02-01
IE922310A1 (en) 1993-02-10
TW207541B (no) 1993-06-11
EP0525584B1 (de) 1997-12-10
CZ239392A3 (en) 1993-04-14
NO923004L (no) 1993-02-01
ES2110454T3 (es) 1998-02-16
NO923004D0 (no) 1992-07-30
RU2078765C1 (ru) 1997-05-10
NZ243715A (en) 1995-03-28
FI923440A0 (fi) 1992-07-30
DE59209055D1 (de) 1998-01-22
EP0525584A1 (de) 1993-02-03
KR930002353A (ko) 1993-02-23
AU2067792A (en) 1993-02-04
US5272143A (en) 1993-12-21
CA2075102A1 (en) 1993-02-01
CN1141773A (zh) 1997-02-05

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IL102503A (en) History of Alkanamine of 6-Oxoazepino] CD-5,4,3 [Indole, their preparation and pharmaceutical preparations containing them
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Legal Events

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FF Patent granted
RH Patent void