IL100502A - תכשירי רוקחות המכילים סיס-4- אמינו-1- )2-הידרוקסימתיל- 1,3- אוקסאתיולן-5-איל(- h1- פירימיד -2-און נוקלאוסיד או תולדות שלהן - Google Patents

תכשירי רוקחות המכילים סיס-4- אמינו-1- )2-הידרוקסימתיל- 1,3- אוקסאתיולן-5-איל(- h1- פירימיד -2-און נוקלאוסיד או תולדות שלהן

Info

Publication number
IL100502A
IL100502A IL10050291A IL10050291A IL100502A IL 100502 A IL100502 A IL 100502A IL 10050291 A IL10050291 A IL 10050291A IL 10050291 A IL10050291 A IL 10050291A IL 100502 A IL100502 A IL 100502A
Authority
IL
Israel
Prior art keywords
compound
formula
hepatitis
amino
oxathiolan
Prior art date
Application number
IL10050291A
Other languages
English (en)
Other versions
IL100502A0 (en
Original Assignee
Iaf Biochem Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26298202&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL100502(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GB919100039A external-priority patent/GB9100039D0/en
Priority claimed from GB919109913A external-priority patent/GB9109913D0/en
Application filed by Iaf Biochem Int filed Critical Iaf Biochem Int
Publication of IL100502A0 publication Critical patent/IL100502A0/xx
Publication of IL100502A publication Critical patent/IL100502A/he

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
IL10050291A 1991-01-03 1991-12-25 תכשירי רוקחות המכילים סיס-4- אמינו-1- )2-הידרוקסימתיל- 1,3- אוקסאתיולן-5-איל(- h1- פירימיד -2-און נוקלאוסיד או תולדות שלהן IL100502A (he)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB919100039A GB9100039D0 (en) 1991-01-03 1991-01-03 Medicaments
GB919109913A GB9109913D0 (en) 1991-05-07 1991-05-07 Medicaments

Publications (2)

Publication Number Publication Date
IL100502A0 IL100502A0 (en) 1992-09-06
IL100502A true IL100502A (he) 1995-12-08

Family

ID=26298202

Family Applications (1)

Application Number Title Priority Date Filing Date
IL10050291A IL100502A (he) 1991-01-03 1991-12-25 תכשירי רוקחות המכילים סיס-4- אמינו-1- )2-הידרוקסימתיל- 1,3- אוקסאתיולן-5-איל(- h1- פירימיד -2-און נוקלאוסיד או תולדות שלהן

Country Status (23)

Country Link
US (2) US5532246A (he)
EP (2) EP0565549B1 (he)
JP (1) JP2659863B2 (he)
KR (1) KR0156747B1 (he)
AT (1) ATE120644T1 (he)
AU (1) AU660650B2 (he)
CA (2) CA2100269C (he)
CY (1) CY2047B1 (he)
DE (1) DE69201948T2 (he)
DK (1) DK0565549T3 (he)
EE (1) EE02995B1 (he)
ES (1) ES2070628T3 (he)
GE (1) GEP19981482B (he)
GR (1) GR3015694T3 (he)
HK (1) HK159395A (he)
IE (1) IE73642B1 (he)
IL (1) IL100502A (he)
MD (1) MD1224C2 (he)
NO (1) NO180407C (he)
PH (1) PH31397A (he)
TJ (1) TJ249B (he)
TW (1) TW202385B (he)
WO (1) WO1992011852A1 (he)

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US20020120130A1 (en) 1993-09-10 2002-08-29 Gilles Gosselin 2' or 3' -deoxy and 2', 3' -dideoxy-beta-L-pentofuranonucleo-side compounds, method of preparation and application in therapy, especially as anti- viral agents
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US5703058A (en) 1995-01-27 1997-12-30 Emory University Compositions containing 5-fluoro-2',3'-didehydro-2',3'-dideoxycytidine or a mono-, di-, or triphosphate thereof and a second antiviral agent
US6391859B1 (en) 1995-01-27 2002-05-21 Emory University [5-Carboxamido or 5-fluoro]-[2′,3′-unsaturated or 3′-modified]-pyrimidine nucleosides
US5808040A (en) * 1995-01-30 1998-09-15 Yale University L-nucleosides incorporated into polymeric structure for stabilization of oligonucleotides
US6689761B1 (en) 1995-02-01 2004-02-10 Merck & Co., Inc. Combination therapy for HIV infection
DE69636734T2 (de) 1995-06-07 2007-10-18 Emory University Nucleoside mit anti-hepatitis b virus wirksamkeit
GB9517022D0 (en) * 1995-08-19 1995-10-25 Glaxo Group Ltd Medicaments
GB9605293D0 (en) * 1996-03-13 1996-05-15 Glaxo Group Ltd Medicaments
EP0938321B1 (en) 1996-06-25 2004-01-14 Glaxo Group Limited Combinations comprising vx478, zidovudine and 3tc for use in the treatment of hiv
US5753789A (en) * 1996-07-26 1998-05-19 Yale University Oligonucleotides containing L-nucleosides
US6113920A (en) * 1996-10-31 2000-09-05 Glaxo Wellcome Inc. Pharmaceutical compositions
US20030100532A1 (en) * 1997-02-14 2003-05-29 Gary S. Jacob Use of n-substituted-1,5-dideoxy-1,5-imino-d-glucitol compounds in combination therapy for treating hepatitis virus infections
WO1998044913A2 (en) 1997-04-07 1998-10-15 Triangle Pharmaceuticals, Inc. Compositions containing mkc-442 in combination with other antiviral agents
MXPA01001507A (es) 1998-08-10 2003-09-10 Novirio Pharmaceuticals Ltd °l-2'desoxi-nucleosidos para el tratamiento de hepatitis b.
US6444652B1 (en) 1998-08-10 2002-09-03 Novirio Pharmaceuticals Limited β-L-2'-deoxy-nucleosides for the treatment of hepatitis B
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US6407077B1 (en) 1998-11-05 2002-06-18 Emory University β-L nucleosides for the treatment of HIV infection
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CN1315862C (zh) 2000-05-26 2007-05-16 艾登尼科斯（开曼）有限公司 处理黄病毒和瘟病毒的方法和组合物
US6787526B1 (en) 2000-05-26 2004-09-07 Idenix Pharmaceuticals, Inc. Methods of treating hepatitis delta virus infection with β-L-2′-deoxy-nucleosides
US6875751B2 (en) 2000-06-15 2005-04-05 Idenix Pharmaceuticals, Inc. 3′-prodrugs of 2′-deoxy-β-L-nucleosides
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Also Published As

Publication number Publication date
DE69201948T2 (de) 1995-08-03
EE02995B1 (et) 1997-06-16
DE69201948D1 (de) 1995-05-11
HK159395A (en) 1995-10-20
MD950086A (ro) 1997-01-31
NO932442L (no) 1993-08-26
CA2100269A1 (en) 1992-07-04
GR3015694T3 (en) 1995-07-31
NO932442D0 (no) 1993-07-05
IE920004A1 (en) 1992-07-15
EP0565549A1 (en) 1993-10-20
MD1224B2 (en) 1999-05-31
KR0156747B1 (en) 1998-11-16
CY2047B1 (en) 1998-04-30
TJ249B (en) 1999-12-23
USRE39155E1 (en) 2006-07-04
IL100502A0 (en) 1992-09-06
NO180407B (no) 1997-01-06
PH31397A (en) 1998-10-29
ES2070628T3 (es) 1995-06-01
AU1153492A (en) 1992-08-17
IE73642B1 (en) 1997-06-18
EP0494119A1 (en) 1992-07-08
JP2659863B2 (ja) 1997-09-30
TW202385B (he) 1993-03-21
AU660650B2 (en) 1995-07-06
DK0565549T3 (da) 1995-07-03
ATE120644T1 (de) 1995-04-15
CA2100269C (en) 1999-02-23
CA2254613A1 (en) 1992-07-04
WO1992011852A1 (en) 1992-07-23
NO180407C (no) 1997-04-16
JPH06507150A (ja) 1994-08-11
GEP19981482B (en) 1998-12-25
US5532246A (en) 1996-07-02
MD1224C2 (ro) 1999-11-30
EP0565549B1 (en) 1995-04-05

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