IE45613L - Cephalosporins. - Google Patents
Cephalosporins.Info
- Publication number
- IE45613L IE45613L IE771969A IE196977A IE45613L IE 45613 L IE45613 L IE 45613L IE 771969 A IE771969 A IE 771969A IE 196977 A IE196977 A IE 196977A IE 45613 L IE45613 L IE 45613L
- Authority
- IE
- Ireland
- Prior art keywords
- formula
- compound
- gb1572201a
- ylthiomethyl
- cephem
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
- C07D217/24—Oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/24—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Cephalosporin Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
New amino-3-(2-carboxyalkyl-2,3-dihydro-3-oxo-s-triazolo[4,3-b]pyridazin-6 -ylthiomethyl)-3-cephem-4-carboxylic acids of formula I, their salts and their easily hydrolysed esters of the 4-carboxyl group are prepared. The synthesis consists in reacting a compound of formula III with a compound of formula IV and then treating the product obtained with an acylating agent R<2>-X. The compounds of the invention are powerful antibacterial agents which have a good solubility in water. <IMAGE>
[GB1572201A]
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IE269/81A IE45614B1 (en) | 1977-04-05 | 1977-09-27 | Cephalosporins |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US05/784,885 US4082912A (en) | 1976-06-30 | 1977-04-05 | Certain 7-acylamido-3-(2-carboxyalkyl-2,3-dihydro-s-triazolo[4,3-b]pyridazin-3-on-6-ylmethyl)-3-cephem-4-carboxylic acids their salts and easily hydrolyzed esters |
Publications (2)
Publication Number | Publication Date |
---|---|
IE45613L true IE45613L (en) | 1978-10-05 |
IE45613B1 IE45613B1 (en) | 1982-10-06 |
Family
ID=25133827
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IE1969/77A IE45613B1 (en) | 1977-04-05 | 1977-09-27 | Cephalosporins |
Country Status (17)
Country | Link |
---|---|
JP (1) | JPS53124290A (en) |
AU (1) | AU517919B2 (en) |
BE (1) | BE859774A (en) |
CA (1) | CA1113455A (en) |
CH (1) | CH627184A5 (en) |
DE (1) | DE2807847A1 (en) |
DK (1) | DK145497C (en) |
FI (1) | FI60869C (en) |
FR (1) | FR2408614A1 (en) |
GB (1) | GB1572201A (en) |
GR (1) | GR73550B (en) |
IE (1) | IE45613B1 (en) |
LU (1) | LU78323A1 (en) |
NL (1) | NL7711644A (en) |
SE (1) | SE425491B (en) |
YU (1) | YU247977A (en) |
ZA (1) | ZA775781B (en) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3000377A1 (en) * | 1980-01-07 | 1981-07-09 | Boehringer Mannheim Gmbh, 6800 Mannheim | NEW SULPHONAMIDES, METHOD FOR THE PRODUCTION THEREOF AND MEDICINAL PRODUCTS CONTAINING THESE COMPOUNDS |
CN114940665B (en) * | 2022-06-10 | 2024-05-07 | 河南省科学院高新技术研究中心 | Benzisothiazolinone compound serving as bactericide and preparation method thereof |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3907786A (en) * | 1973-09-04 | 1975-09-23 | Bristol Myers Co | 7-{8 {60 -(2-aminomethyl-1,4-cyclohexadienyl)acetamido{9 -3-heterocyclic-thiomethyl-3-cephem-4-carboxylic acids and salts |
US3946000A (en) * | 1973-10-31 | 1976-03-23 | Bristol-Myers Company | 7-[α-(2-Aminomethyl-1-cyclohexenyl)-acetamido]-3-heterocyclic thiomethyl-3-cephem-4-carboxylic acids |
-
1977
- 1977-09-26 GB GB39951/77A patent/GB1572201A/en not_active Expired
- 1977-09-27 CA CA287,569A patent/CA1113455A/en not_active Expired
- 1977-09-27 ZA ZA00775781A patent/ZA775781B/en unknown
- 1977-09-27 IE IE1969/77A patent/IE45613B1/en unknown
- 1977-09-28 DK DK429577A patent/DK145497C/en not_active IP Right Cessation
- 1977-09-28 SE SE7710823A patent/SE425491B/en unknown
- 1977-09-28 GR GR54448A patent/GR73550B/el unknown
- 1977-09-28 FI FI772860A patent/FI60869C/en not_active IP Right Cessation
- 1977-10-04 AU AU29328/77A patent/AU517919B2/en not_active Expired
- 1977-10-10 FR FR7730383A patent/FR2408614A1/en active Granted
- 1977-10-13 CH CH1249577A patent/CH627184A5/en not_active IP Right Cessation
- 1977-10-14 YU YU02479/77A patent/YU247977A/en unknown
- 1977-10-14 BE BE181787A patent/BE859774A/en not_active IP Right Cessation
- 1977-10-17 LU LU78323A patent/LU78323A1/xx unknown
- 1977-10-24 NL NL7711644A patent/NL7711644A/en not_active Application Discontinuation
- 1977-10-24 JP JP12688377A patent/JPS53124290A/en active Pending
-
1978
- 1978-02-23 DE DE19782807847 patent/DE2807847A1/en not_active Withdrawn
Also Published As
Publication number | Publication date |
---|---|
NL7711644A (en) | 1978-10-09 |
FI60869B (en) | 1981-12-31 |
SE7710823L (en) | 1978-10-06 |
CA1113455A (en) | 1981-12-01 |
ZA775781B (en) | 1978-08-30 |
FI772860A (en) | 1978-10-06 |
IE45613B1 (en) | 1982-10-06 |
CH627184A5 (en) | 1981-12-31 |
BE859774A (en) | 1978-04-14 |
FR2408614B1 (en) | 1980-12-05 |
GB1572201A (en) | 1980-07-23 |
JPS53124290A (en) | 1978-10-30 |
DK429577A (en) | 1978-10-06 |
FR2408614A1 (en) | 1979-06-08 |
DK145497C (en) | 1983-05-02 |
AU2932877A (en) | 1979-04-12 |
GR73550B (en) | 1984-03-13 |
LU78323A1 (en) | 1978-06-12 |
SE425491B (en) | 1982-10-04 |
DK145497B (en) | 1982-11-29 |
DE2807847A1 (en) | 1978-10-19 |
YU247977A (en) | 1982-10-31 |
AU517919B2 (en) | 1981-09-03 |
FI60869C (en) | 1982-04-13 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
IE802347L (en) | 7-acylamino-3-vinylcephalosporanic acid derivatives | |
JPS5452096A (en) | Cephem compound, its preparation and bacteriostatic agent containing the same | |
JPS55105689A (en) | Novel cephem and cepham compounds, their preparation and preventive and remedy for microbism | |
JPS5547688A (en) | Novel cephem compound and its preparation | |
IE45613L (en) | Cephalosporins. | |
IE45559L (en) | ß-LACTAM COMPOUNDS | |
ES482280A1 (en) | Imidazolylethoxy derivatives of pyrazolo{8 3,4-b{9 pyridine-5-methanols | |
JPS5511600A (en) | Cephem compound, its salt, their preparation and remedy and prophylactic for microbism containing mainly the same | |
IE42191L (en) | 7ó-methoxy cephalosporin compounds. | |
ES8504829A1 (en) | Alpha-hydroxy-beta-haloethylphosphinic acids and their salts, and their production and use. | |
JPS54117493A (en) | 3,7-disubstituted-3-cephem-4-carboxylic acid compound, its salt, its preparation, and preventives and remedies for microbism consisting mainly of them | |
IE772501L (en) | Clavulanic acid ethers | |
JPS56128787A (en) | Cephalosporin derivative and its preparation | |
IE43666L (en) | Cephalosporin derivatives. | |
JPS55100391A (en) | Cephalosporin analog | |
JPS565484A (en) | Cephalosporin derivative and its salt | |
JPS54144392A (en) | Cephalosporin derivative | |
JPS56122383A (en) | Novel cephalosporin compound and its preparation | |
JPS57163386A (en) | Cephalosporin derivative and its production | |
JPS56164194A (en) | Cephalosporin derivative | |
IE40122L (en) | Preparation of 7-acylamino cephalosporin derivatives | |
JPS5492986A (en) | Cephalosporin derivative | |
JPS5770893A (en) | Preparation of cephalosporin derivative | |
JPS6442490A (en) | Substituted oxycarbonylaminocephem compound | |
JPS5645461A (en) | Alpha-amino acid derivative |