JPS56122383A - Novel cephalosporin compound and its preparation - Google Patents
Novel cephalosporin compound and its preparationInfo
- Publication number
- JPS56122383A JPS56122383A JP2699280A JP2699280A JPS56122383A JP S56122383 A JPS56122383 A JP S56122383A JP 2699280 A JP2699280 A JP 2699280A JP 2699280 A JP2699280 A JP 2699280A JP S56122383 A JPS56122383 A JP S56122383A
- Authority
- JP
- Japan
- Prior art keywords
- formula
- carboxylic acid
- gram
- give
- cephalosporin compound
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Classifications
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Cephalosporin Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
NEW MATERIAL:A cephalosporin compound shown by the formula I (R1 is phenyl which may be substituted by hydroxyl group, etc.; one of R2 and R3 is carboxyl which may be esterified or amino which may be acylated by a nitrogen-containing heterocyclic carboxylic acid and the other is H, both form substituted imino; R4 is lower alkyl).
EXAMPLE: 7-( α-Carboxyphenylacetamide )-3-[ 2-(1-methyl-1H-tetrazole-5-yl )vinyl]-Δ3-cephem-4-carboxylic acid.
USE: An antibacterial agent. Having antibacterial action on Gram-positive and Gram- negative bacteria.
PROCESS: A 7-aminocephalosporin derivative shown by the formula II is reacted with a carboxylic acid derivative shown by the formula III, and, if necessary, a protecting group is removed, to give a reaction product, which is converted into a salt or ester, to give a compound shown by the formula I.
COPYRIGHT: (C)1981,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2699280A JPS56122383A (en) | 1980-03-04 | 1980-03-04 | Novel cephalosporin compound and its preparation |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2699280A JPS56122383A (en) | 1980-03-04 | 1980-03-04 | Novel cephalosporin compound and its preparation |
Publications (1)
Publication Number | Publication Date |
---|---|
JPS56122383A true JPS56122383A (en) | 1981-09-25 |
Family
ID=12208649
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2699280A Pending JPS56122383A (en) | 1980-03-04 | 1980-03-04 | Novel cephalosporin compound and its preparation |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS56122383A (en) |
-
1980
- 1980-03-04 JP JP2699280A patent/JPS56122383A/en active Pending
Similar Documents
Publication | Publication Date | Title |
---|---|---|
JPS5452096A (en) | Cephem compound, its preparation and bacteriostatic agent containing the same | |
JPS5543011A (en) | 7-halothiazolylalkoxyiminoacetamido-3-cephem compound | |
JPS565487A (en) | Cephalosporin compound, its preparation, and antimicrobial comprising it | |
JPS5547688A (en) | Novel cephem compound and its preparation | |
JPS56118085A (en) | 2-methylcephalosporin derivative and its preparation | |
JPS5799592A (en) | Novel cephalosporins | |
JPS56122383A (en) | Novel cephalosporin compound and its preparation | |
JPS54117493A (en) | 3,7-disubstituted-3-cephem-4-carboxylic acid compound, its salt, its preparation, and preventives and remedies for microbism consisting mainly of them | |
JPS5515454A (en) | Novel cephalosporin derivative | |
JPS57165389A (en) | Novel penicillin and cephalosporin compound | |
JPS5780390A (en) | Novel cephalosporin derivative | |
JPS5549384A (en) | Novel antibacterial compound | |
JPS5732289A (en) | Alpha-substituted ureidobenzylpenicillin | |
JPS56115788A (en) | Azetidinone derivative and its preparation | |
JPS5673087A (en) | Cephalosporin derivative, its preparation and antimicrobial agent consisting of the same | |
JPS57165390A (en) | Novel penicillin and cephalosporin derivative | |
JPS57163386A (en) | Cephalosporin derivative and its production | |
JPS57167993A (en) | Novel 3-((4-carboxy-3-hydroxyisothiazole-5-yl) thiomethyl)-delta3-cephem derivative | |
JPS55100391A (en) | Cephalosporin analog | |
JPS5770897A (en) | Aminoethylphosphonic acid derivative | |
JPS56142283A (en) | Penem-3-carboxylic acid derivative and its preparation | |
JPS56133260A (en) | Azetidine derivative and its preparation | |
JPS5585594A (en) | Cephem compound and their preparation | |
JPS5645461A (en) | Alpha-amino acid derivative | |
JPS55136292A (en) | Cephalosporin derivative, its preparation, and antibacterial comprising it |