IE36231L - Triazolo diazepines - Google Patents

Triazolo diazepines

Info

Publication number
IE36231L
IE36231L IE720404A IE40472A IE36231L IE 36231 L IE36231 L IE 36231L IE 720404 A IE720404 A IE 720404A IE 40472 A IE40472 A IE 40472A IE 36231 L IE36231 L IE 36231L
Authority
IE
Ireland
Prior art keywords
oxides
alkyl
cpds
opt
diazepines
Prior art date
Application number
IE720404A
Other versions
IE36231B1 (en
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Publication of IE36231L publication Critical patent/IE36231L/en
Publication of IE36231B1 publication Critical patent/IE36231B1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C243/00—Compounds containing chains of nitrogen atoms singly-bound to each other, e.g. hydrazines, triazanes

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)

Abstract

Title cpds. of formula (I): (where R1 is H or 1-3C alkyl; R2 is 1-4C alkyl or R2--R2 is a satd. divalent 2-5C aliphatic hydrocarbon residue, and rings A and B can be substd. by F, Cl, Br, CF3, NO2 or 1-6C alkyl or alkoxy) and their 5-oxides and acid addn. salts, can be used as tranquillisers, sedatives, muscle relaxants and anti-epileptics; the 5-oxides are also of use as inters. for further pharmacologically active cpds. Cpds. (I) are e.g. prepd. by (a) reacting a 2-X-3-R1-5-phenyl-3H-1,4-benzodiazepine (where X is SH, lower alkoxy or alkylthio opt. activated by a substituent, or opt. mono- or disubstd. amino) with (R2O)2CHCONHNH2. The 5-oxides are obtd. by oxidn. [CH545302A]
IE404/72A 1971-04-08 1972-03-28 Triazolo diazepine derivatives and processes for the production thereof IE36231B1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH523371 1971-04-08

Publications (2)

Publication Number Publication Date
IE36231L true IE36231L (en) 1972-10-08
IE36231B1 IE36231B1 (en) 1976-09-15

Family

ID=4290168

Family Applications (1)

Application Number Title Priority Date Filing Date
IE404/72A IE36231B1 (en) 1971-04-08 1972-03-28 Triazolo diazepine derivatives and processes for the production thereof

Country Status (24)

Country Link
US (1) US3867536A (en)
JP (1) JPS5614671B1 (en)
AR (3) AR193382A1 (en)
AT (2) AT317222B (en)
AU (1) AU472767B2 (en)
BE (1) BE781816A (en)
CA (1) CA991639A (en)
CH (1) CH545302A (en)
CS (3) CS178406B2 (en)
DD (1) DD97655A5 (en)
DE (1) DE2215939A1 (en)
DK (1) DK141965B (en)
FI (1) FI52583C (en)
FR (1) FR2132767B1 (en)
GB (1) GB1392327A (en)
HU (1) HU165318B (en)
IE (1) IE36231B1 (en)
IL (1) IL39051A (en)
NL (1) NL7204700A (en)
NO (1) NO134839C (en)
PL (1) PL83566B1 (en)
SE (1) SE413408B (en)
SU (3) SU499808A3 (en)
ZA (1) ZA721896B (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH572056A5 (en) * 1972-11-28 1976-01-30 Ciba Geigy Ag

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3987052A (en) * 1969-03-17 1976-10-19 The Upjohn Company 6-Phenyl-4H-s-triazolo[4,3-a][1,4]benzodiazepines
BE759099A (en) * 1969-11-18 1971-04-30 Takeda Chemical Industries Ltd PROCESS FOR MANUFACTURING HETEROCYCLIC COMPOUNDS
US3681343A (en) * 1971-05-11 1972-08-01 Upjohn Co 6-phenyl-s-triazolo{8 4,3-a{9 {8 1,4{9 {0 benzodiazepines

Also Published As

Publication number Publication date
NO134839C (en) 1976-12-21
DK141965C (en) 1980-12-08
SU489332A3 (en) 1975-10-25
AT317230B (en) 1974-08-26
DE2215939A1 (en) 1972-10-19
IL39051A0 (en) 1972-05-30
AR194991A1 (en) 1973-08-30
AR193382A1 (en) 1973-04-23
FI52583C (en) 1977-10-10
DD97655A5 (en) 1973-05-12
SU499808A3 (en) 1976-01-15
NO134839B (en) 1976-09-13
FI52583B (en) 1977-06-30
AU4082072A (en) 1973-10-11
FR2132767B1 (en) 1975-06-20
CA991639A (en) 1976-06-22
SU482045A3 (en) 1975-08-25
AT317222B (en) 1974-08-26
US3867536A (en) 1975-02-18
CS178449B2 (en) 1977-09-15
IE36231B1 (en) 1976-09-15
IL39051A (en) 1975-02-10
SE413408B (en) 1980-05-27
DK141965B (en) 1980-07-28
FR2132767A1 (en) 1972-11-24
JPS5614671B1 (en) 1981-04-06
NL7204700A (en) 1972-10-10
HU165318B (en) 1974-08-28
GB1392327A (en) 1975-04-30
ZA721896B (en) 1972-12-27
CH545302A (en) 1974-01-13
BE781816A (en) 1972-10-09
CS178406B2 (en) 1977-09-15
PL83566B1 (en) 1975-12-31
AR193942A1 (en) 1973-05-31
AU472767B2 (en) 1973-10-11
CS178448B2 (en) 1977-09-15

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