FR2207719A2 - Triazolobenzodiazepine prepns - with antidepressant and anxiolytic activity - Google Patents

Triazolobenzodiazepine prepns - with antidepressant and anxiolytic activity

Info

Publication number
FR2207719A2
FR2207719A2 FR7341861A FR7341861A FR2207719A2 FR 2207719 A2 FR2207719 A2 FR 2207719A2 FR 7341861 A FR7341861 A FR 7341861A FR 7341861 A FR7341861 A FR 7341861A FR 2207719 A2 FR2207719 A2 FR 2207719A2
Authority
FR
France
Prior art keywords
antidepressant
prepns
anxiolytic activity
triazolobenzodiazepine
pharm
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7341861A
Other languages
French (fr)
Other versions
FR2207719B2 (en
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pharmacia and Upjohn Co
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of FR2207719A2 publication Critical patent/FR2207719A2/en
Application granted granted Critical
Publication of FR2207719B2 publication Critical patent/FR2207719B2/fr
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Pharmaceutical prepns contain >=1 triazolobenzodiazepines of formula (I): (where R1 and R2 are H, CH3 or C2H5 and R3 is H, F, Cl, Br, CN NO2, CF3 or 1-3C alkylthio) or their pharm. acceptable acid addn salts of N-oxides, opt. together with usual pharm. carriers, have antidepressant and anxiolytic activity and can be used in the treatment of depression, anxiety, and mixed anxiety/depression states such as occur with certain neuroses.
FR7341861A 1972-11-24 1973-11-23 Triazolobenzodiazepine prepns - with antidepressant and anxiolytic activity Granted FR2207719A2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US30921372A 1972-11-24 1972-11-24
US32047573A 1973-01-02 1973-01-02

Publications (2)

Publication Number Publication Date
FR2207719A2 true FR2207719A2 (en) 1974-06-21
FR2207719B2 FR2207719B2 (en) 1977-09-02

Family

ID=26976672

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7341861A Granted FR2207719A2 (en) 1972-11-24 1973-11-23 Triazolobenzodiazepine prepns - with antidepressant and anxiolytic activity

Country Status (2)

Country Link
DE (1) DE2356369C2 (en)
FR (1) FR2207719A2 (en)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2375233A1 (en) * 1976-03-15 1978-07-21 Upjohn Co NEW BENZODIAZEPINES, THEIR PREPARATION PROCESS AND THE MEDICINAL PRODUCT CONTAINING THEM

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2122485A1 (en) * 1971-01-21 1972-09-01 Ciba Geigy Ag

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI50981C (en) * 1968-11-05 1976-09-10 Takeda Chemical Industries Ltd Process for the preparation of s-triat solo- (4,3-a) (1,4) -benzodiazepines acting as hypnotics and sedatives.

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2122485A1 (en) * 1971-01-21 1972-09-01 Ciba Geigy Ag

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2375233A1 (en) * 1976-03-15 1978-07-21 Upjohn Co NEW BENZODIAZEPINES, THEIR PREPARATION PROCESS AND THE MEDICINAL PRODUCT CONTAINING THEM

Also Published As

Publication number Publication date
DE2356369A1 (en) 1974-05-30
AU6207073A (en) 1975-05-01
DE2356369C2 (en) 1984-08-23
FR2207719B2 (en) 1977-09-02

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