HUT73357A - Process for the preparation of substituted 4,6-diamino-5-cyanopyrimidine derivatives - Google Patents

Process for the preparation of substituted 4,6-diamino-5-cyanopyrimidine derivatives Download PDF

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Publication number
HUT73357A
HUT73357A HU9503959A HU9503959A HUT73357A HU T73357 A HUT73357 A HU T73357A HU 9503959 A HU9503959 A HU 9503959A HU 9503959 A HU9503959 A HU 9503959A HU T73357 A HUT73357 A HU T73357A
Authority
HU
Hungary
Prior art keywords
formula
alkali metal
amino
dicyanoethylene
water
Prior art date
Application number
HU9503959A
Other languages
English (en)
Hungarian (hu)
Other versions
HU9503959D0 (en
Inventor
Jean-Marie Assercq
Jeffrey William Perine
Heinz Peter Schwemlein
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Publication of HU9503959D0 publication Critical patent/HU9503959D0/hu
Publication of HUT73357A publication Critical patent/HUT73357A/hu

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/50Three nitrogen atoms

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
HU9503959A 1993-07-26 1994-07-14 Process for the preparation of substituted 4,6-diamino-5-cyanopyrimidine derivatives HUT73357A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US9714193A 1993-07-26 1993-07-26
US21098094A 1994-03-21 1994-03-21

Publications (2)

Publication Number Publication Date
HU9503959D0 HU9503959D0 (en) 1996-03-28
HUT73357A true HUT73357A (en) 1996-07-29

Family

ID=26792702

Family Applications (1)

Application Number Title Priority Date Filing Date
HU9503959A HUT73357A (en) 1993-07-26 1994-07-14 Process for the preparation of substituted 4,6-diamino-5-cyanopyrimidine derivatives

Country Status (15)

Country Link
EP (1) EP0711285A1 (sk)
JP (1) JPH09500632A (sk)
CN (1) CN1128024A (sk)
AU (1) AU7385994A (sk)
BG (1) BG100366A (sk)
BR (1) BR9407024A (sk)
CA (1) CA2166989A1 (sk)
CZ (1) CZ22496A3 (sk)
FI (1) FI960332A (sk)
HU (1) HUT73357A (sk)
IL (1) IL110425A0 (sk)
LV (1) LV11463B (sk)
NO (1) NO960307D0 (sk)
SK (1) SK10396A3 (sk)
WO (1) WO1995003282A2 (sk)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT1007516E (pt) * 1997-08-27 2004-11-30 Novartis Ag Polimorfos e hidratos de diciclanilo e sua preparacao
ATE528283T1 (de) 2007-04-19 2011-10-15 Nippon Soda Co Verfahren zur herstellung von n-(2-amino-1,2- dicyanovinyl)imidaten und verfahren zur herstellung von aminoimidazolderivaten
CN102250017A (zh) * 2011-06-15 2011-11-23 扬州天和药业有限公司 地昔尼尔的一种合成方法
CN102399193A (zh) * 2011-12-15 2012-04-04 连云港市亚晖医药化工有限公司 4,6-二氨基-2-环丙胺基-5-腈基嘧啶的制备方法
CN104130197A (zh) * 2014-07-29 2014-11-05 华中农业大学 2,4,6-三氨基-5-氰基嘧啶的化学合成方法
CN104649982B (zh) * 2015-02-26 2016-12-07 齐鲁晟华制药有限公司 一种地昔尼尔的制备方法
CN107056655B (zh) * 2017-01-22 2018-12-04 营口三征新科技化工有限公司 一种1-氨基-1-氰氨基-2,2-二氰乙烯钠盐的制备方法
CN106966922B (zh) * 2017-03-28 2020-10-27 中国科学院大学 一种功能化取代的二氰基乙烯类化合物的合成方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1135913B (de) * 1960-11-08 1962-09-06 Bayer Ag Verfahren zur Herstellung von 2-Methyl-4-amino-5-cyanpyrimidin
US3226424A (en) * 1962-10-03 1965-12-28 Hoffmann La Roche Process for preparing 2-lower alkoxy-1,1-dicyanoethylene and 2-amino-1,1-dicyanoethylene
US4783468A (en) * 1986-04-30 1988-11-08 Ciba-Geigy Corporation Insecticidal 5-pyrimidine carbonitriles

Also Published As

Publication number Publication date
BG100366A (en) 1996-07-31
NO960307L (no) 1996-01-25
AU7385994A (en) 1995-02-20
WO1995003282A2 (en) 1995-02-02
BR9407024A (pt) 1996-09-10
JPH09500632A (ja) 1997-01-21
LV11463A (lv) 1996-08-20
FI960332A0 (fi) 1996-01-24
SK10396A3 (en) 1996-09-04
WO1995003282A3 (en) 1995-04-13
HU9503959D0 (en) 1996-03-28
NO960307D0 (no) 1996-01-25
CN1128024A (zh) 1996-07-31
FI960332A (fi) 1996-01-24
IL110425A0 (en) 1994-10-21
EP0711285A1 (en) 1996-05-15
CZ22496A3 (en) 1996-04-17
CA2166989A1 (en) 1995-02-02
LV11463B (en) 1996-12-20

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Legal Events

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DFC4 Cancellation of temporary protection due to refusal