FI960332A0 - Menetelmä substituoitujan 4,6-diamino-5-syanopyrinidiinien valmistamiseksi - Google Patents

Menetelmä substituoitujan 4,6-diamino-5-syanopyrinidiinien valmistamiseksi

Info

Publication number
FI960332A0
FI960332A0 FI960332A FI960332A FI960332A0 FI 960332 A0 FI960332 A0 FI 960332A0 FI 960332 A FI960332 A FI 960332A FI 960332 A FI960332 A FI 960332A FI 960332 A0 FI960332 A0 FI 960332A0
Authority
FI
Finland
Prior art keywords
pyrimidines
diamino
cyano
preparing substituted
substituted
Prior art date
Application number
FI960332A
Other languages
English (en)
Swedish (sv)
Other versions
FI960332A (fi
Inventor
Jean-Marie Asserco
Heinz Peter Schwemlein
Jeffrey William Perine
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Publication of FI960332A0 publication Critical patent/FI960332A0/fi
Publication of FI960332A publication Critical patent/FI960332A/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/50Three nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
FI960332A 1993-07-26 1996-01-24 Menetelmä substituoitujan 4,6-diamino-5-syanopyrinidiinien valmistamiseksi FI960332A (fi)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US9714193A 1993-07-26 1993-07-26
US21098094A 1994-03-21 1994-03-21
PCT/EP1994/002312 WO1995003282A2 (en) 1993-07-26 1994-07-14 Process for the preparation of substituted 4,6-diamino-5-cyanopyrimidines

Publications (2)

Publication Number Publication Date
FI960332A0 true FI960332A0 (fi) 1996-01-24
FI960332A FI960332A (fi) 1996-01-24

Family

ID=26792702

Family Applications (1)

Application Number Title Priority Date Filing Date
FI960332A FI960332A (fi) 1993-07-26 1996-01-24 Menetelmä substituoitujan 4,6-diamino-5-syanopyrinidiinien valmistamiseksi

Country Status (15)

Country Link
EP (1) EP0711285A1 (fi)
JP (1) JPH09500632A (fi)
CN (1) CN1128024A (fi)
AU (1) AU7385994A (fi)
BG (1) BG100366A (fi)
BR (1) BR9407024A (fi)
CA (1) CA2166989A1 (fi)
CZ (1) CZ22496A3 (fi)
FI (1) FI960332A (fi)
HU (1) HUT73357A (fi)
IL (1) IL110425A0 (fi)
LV (1) LV11463B (fi)
NO (1) NO960307D0 (fi)
SK (1) SK10396A3 (fi)
WO (1) WO1995003282A2 (fi)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR9811920A (pt) * 1997-08-27 2000-08-15 Novartis Ag Formas polimorfas de cristais de diciclanil e hidratos dos mesmos e sua preparação
KR101132590B1 (ko) 2007-04-19 2012-04-10 닛뽕소다 가부시키가이샤 N-(2-아미노-1,2-디시아노비닐)이미데이트류의 제조 방법
CN102250017A (zh) * 2011-06-15 2011-11-23 扬州天和药业有限公司 地昔尼尔的一种合成方法
CN102399193A (zh) * 2011-12-15 2012-04-04 连云港市亚晖医药化工有限公司 4,6-二氨基-2-环丙胺基-5-腈基嘧啶的制备方法
CN104130197A (zh) * 2014-07-29 2014-11-05 华中农业大学 2,4,6-三氨基-5-氰基嘧啶的化学合成方法
CN104649982B (zh) * 2015-02-26 2016-12-07 齐鲁晟华制药有限公司 一种地昔尼尔的制备方法
CN107056655B (zh) * 2017-01-22 2018-12-04 营口三征新科技化工有限公司 一种1-氨基-1-氰氨基-2,2-二氰乙烯钠盐的制备方法
CN106966922B (zh) * 2017-03-28 2020-10-27 中国科学院大学 一种功能化取代的二氰基乙烯类化合物的合成方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1135913B (de) * 1960-11-08 1962-09-06 Bayer Ag Verfahren zur Herstellung von 2-Methyl-4-amino-5-cyanpyrimidin
US3226424A (en) * 1962-10-03 1965-12-28 Hoffmann La Roche Process for preparing 2-lower alkoxy-1,1-dicyanoethylene and 2-amino-1,1-dicyanoethylene
US4783468A (en) * 1986-04-30 1988-11-08 Ciba-Geigy Corporation Insecticidal 5-pyrimidine carbonitriles

Also Published As

Publication number Publication date
LV11463B (en) 1996-12-20
CN1128024A (zh) 1996-07-31
CA2166989A1 (en) 1995-02-02
HU9503959D0 (en) 1996-03-28
WO1995003282A2 (en) 1995-02-02
HUT73357A (en) 1996-07-29
NO960307L (no) 1996-01-25
NO960307D0 (no) 1996-01-25
BG100366A (en) 1996-07-31
FI960332A (fi) 1996-01-24
EP0711285A1 (en) 1996-05-15
CZ22496A3 (en) 1996-04-17
SK10396A3 (en) 1996-09-04
AU7385994A (en) 1995-02-20
IL110425A0 (en) 1994-10-21
WO1995003282A3 (en) 1995-04-13
BR9407024A (pt) 1996-09-10
LV11463A (lv) 1996-08-20
JPH09500632A (ja) 1997-01-21

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Legal Events

Date Code Title Description
FD Application lapsed