HUP9901993A3 - Substituted aryl or heteroarylamides having retinoid-like biological activity - Google Patents
Substituted aryl or heteroarylamides having retinoid-like biological activityInfo
- Publication number
- HUP9901993A3 HUP9901993A3 HU9901993A HUP9901993A HUP9901993A3 HU P9901993 A3 HUP9901993 A3 HU P9901993A3 HU 9901993 A HU9901993 A HU 9901993A HU P9901993 A HUP9901993 A HU P9901993A HU P9901993 A3 HUP9901993 A3 HU P9901993A3
- Authority
- HU
- Hungary
- Prior art keywords
- heteroarylamides
- retinoid
- biological activity
- substituted aryl
- aryl
- Prior art date
Links
- 230000004071 biological effect Effects 0.000 title 1
- 125000003107 substituted aryl group Chemical group 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
- C07C235/42—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton
- C07C235/66—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton with carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings being part of condensed ring systems and singly-bound oxygen atoms, bound to the same carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/81—Amides; Imides
- C07D213/82—Amides; Imides in position 3
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C233/00—Carboxylic acid amides
- C07C233/64—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings
- C07C233/81—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
- C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
- C07D311/58—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US08/561,999 US5663357A (en) | 1995-11-22 | 1995-11-22 | Substituted heteroarylamides having retinoid-like biological activity |
Publications (2)
Publication Number | Publication Date |
---|---|
HUP9901993A2 HUP9901993A2 (hu) | 1999-10-28 |
HUP9901993A3 true HUP9901993A3 (en) | 2001-10-29 |
Family
ID=24244378
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HU9901993A HUP9901993A3 (en) | 1995-11-22 | 1996-11-19 | Substituted aryl or heteroarylamides having retinoid-like biological activity |
Country Status (16)
Country | Link |
---|---|
US (6) | US5663357A (hu) |
EP (1) | EP0862555B1 (hu) |
JP (1) | JP4125785B2 (hu) |
KR (1) | KR100483442B1 (hu) |
CN (1) | CN1207727A (hu) |
AT (1) | ATE280160T1 (hu) |
AU (1) | AU715624B2 (hu) |
BR (1) | BR9611615A (hu) |
CA (1) | CA2238310A1 (hu) |
DE (1) | DE69633679T2 (hu) |
HU (1) | HUP9901993A3 (hu) |
IL (3) | IL124593A (hu) |
MX (2) | MX230771B (hu) |
NZ (1) | NZ323574A (hu) |
PL (1) | PL326925A1 (hu) |
WO (1) | WO1997019062A1 (hu) |
Families Citing this family (62)
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US20030219832A1 (en) * | 1996-03-11 | 2003-11-27 | Klein Elliott S. | Synthesis and use of retinoid compounds having negative hormone and/or antagonist activities |
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-
1995
- 1995-11-22 US US08/561,999 patent/US5663357A/en not_active Expired - Lifetime
-
1996
- 1996-11-18 KR KR1019980703816A patent/KR100483442B1/ko not_active IP Right Cessation
- 1996-11-19 WO PCT/US1996/018529 patent/WO1997019062A1/en active IP Right Grant
- 1996-11-19 DE DE69633679T patent/DE69633679T2/de not_active Expired - Fee Related
- 1996-11-19 CA CA002238310A patent/CA2238310A1/en not_active Abandoned
- 1996-11-19 IL IL12459396A patent/IL124593A/en not_active IP Right Cessation
- 1996-11-19 EP EP96941395A patent/EP0862555B1/en not_active Expired - Lifetime
- 1996-11-19 IL IL14374896A patent/IL143748A0/xx unknown
- 1996-11-19 AT AT96941395T patent/ATE280160T1/de not_active IP Right Cessation
- 1996-11-19 NZ NZ323574A patent/NZ323574A/en unknown
- 1996-11-19 PL PL96326925A patent/PL326925A1/xx unknown
- 1996-11-19 BR BR9611615A patent/BR9611615A/pt not_active Application Discontinuation
- 1996-11-19 IL IL14374796A patent/IL143747A0/xx unknown
- 1996-11-19 JP JP51984097A patent/JP4125785B2/ja not_active Expired - Fee Related
- 1996-11-19 HU HU9901993A patent/HUP9901993A3/hu unknown
- 1996-11-19 CN CN96199731A patent/CN1207727A/zh active Pending
- 1996-11-19 AU AU10551/97A patent/AU715624B2/en not_active Ceased
-
1997
- 1997-03-19 US US08/820,792 patent/US5917048A/en not_active Expired - Fee Related
-
1998
- 1998-05-22 MX MX9809697A patent/MX230771B/es unknown
- 1998-05-22 MX MX9804103A patent/MX206851B/es unknown
- 1998-12-17 US US09/215,509 patent/US6051713A/en not_active Expired - Fee Related
-
2000
- 2000-04-17 US US09/550,744 patent/US6245786B1/en not_active Expired - Fee Related
-
2001
- 2001-04-09 US US09/829,310 patent/US6320047B1/en not_active Expired - Fee Related
- 2001-10-16 US US09/982,362 patent/US6437129B1/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
US6051713A (en) | 2000-04-18 |
KR100483442B1 (ko) | 2006-04-21 |
MX206851B (es) | 2002-02-25 |
US5663357A (en) | 1997-09-02 |
HUP9901993A2 (hu) | 1999-10-28 |
ATE280160T1 (de) | 2004-11-15 |
CN1207727A (zh) | 1999-02-10 |
EP0862555A1 (en) | 1998-09-09 |
KR19990071542A (ko) | 1999-09-27 |
PL326925A1 (en) | 1998-11-09 |
IL124593A0 (en) | 1998-12-06 |
IL143747A0 (en) | 2002-04-21 |
US6320047B1 (en) | 2001-11-20 |
JP4125785B2 (ja) | 2008-07-30 |
DE69633679D1 (de) | 2004-11-25 |
DE69633679T2 (de) | 2006-02-09 |
AU715624B2 (en) | 2000-02-03 |
EP0862555B1 (en) | 2004-10-20 |
US20020091262A1 (en) | 2002-07-11 |
US5917048A (en) | 1999-06-29 |
US6245786B1 (en) | 2001-06-12 |
WO1997019062A1 (en) | 1997-05-29 |
US6437129B1 (en) | 2002-08-20 |
IL143748A0 (en) | 2002-04-21 |
CA2238310A1 (en) | 1997-05-29 |
JP2000500498A (ja) | 2000-01-18 |
MX9804103A (es) | 1998-09-30 |
BR9611615A (pt) | 1999-05-25 |
MX230771B (es) | 2005-09-21 |
IL124593A (en) | 2002-09-12 |
NZ323574A (en) | 1999-10-28 |
AU1055197A (en) | 1997-06-11 |
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