HUP0400474A2 - Klórozott pirimidinek előállítása - Google Patents

Klórozott pirimidinek előállítása

Info

Publication number
HUP0400474A2
HUP0400474A2 HU0400474A HUP0400474A HUP0400474A2 HU P0400474 A2 HUP0400474 A2 HU P0400474A2 HU 0400474 A HU0400474 A HU 0400474A HU P0400474 A HUP0400474 A HU P0400474A HU P0400474 A2 HUP0400474 A2 HU P0400474A2
Authority
HU
Hungary
Prior art keywords
synthesis
chlorinated pyrimidines
formula
pyrimidines
chlorinated
Prior art date
Application number
HU0400474A
Other languages
English (en)
Inventor
Timothy John Doyles
Michael Charles Henry Standen
Peter Karl Wehrenberg
Original Assignee
Syngenta Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Limited filed Critical Syngenta Limited
Publication of HUP0400474A2 publication Critical patent/HUP0400474A2/hu
Publication of HUP0400474A3 publication Critical patent/HUP0400474A3/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/30—Halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/52—Two oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

A találmány tárgya eljárás 4,6-diklór-pirimidin előállítására olymódon, hogy egy (I) általános képletű vegyületet - a képletben X1 és Yegymástól függetlenül hidroxilcsoportot, 1-4 szénatomosalkoxicsoportot vagy halogénatomot jelent - legalább egy kvaternerammóniumsó vagy kvaterner foszfóniumsó jelenlétében foszgénnel hoznakérintkezésbe. Ó
HU0400474A 2000-06-26 2001-06-13 Synthesis of chlorinated pyrimidines HUP0400474A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US21412100P 2000-06-26 2000-06-26
PCT/GB2001/002592 WO2002000628A2 (en) 2000-06-26 2001-06-13 Synthesis of chlorinated pyrimidines

Publications (2)

Publication Number Publication Date
HUP0400474A2 true HUP0400474A2 (hu) 2004-08-30
HUP0400474A3 HUP0400474A3 (en) 2006-01-30

Family

ID=22797855

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0400474A HUP0400474A3 (en) 2000-06-26 2001-06-13 Synthesis of chlorinated pyrimidines

Country Status (11)

Country Link
US (1) US20020042514A1 (hu)
EP (1) EP1296957A2 (hu)
JP (1) JP2004501900A (hu)
KR (1) KR20030011893A (hu)
CN (1) CN1697829A (hu)
AR (1) AR030296A1 (hu)
AU (1) AU2001264095A1 (hu)
BR (1) BR0111960A (hu)
HU (1) HUP0400474A3 (hu)
IL (1) IL153099A0 (hu)
WO (1) WO2002000628A2 (hu)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10226220A1 (de) * 2002-06-13 2003-12-24 Bayer Cropscience Ag Verfahren zur Herstellung von 4,6-Dichlor-5-fluorpyrimidin
IL180134A0 (en) * 2006-12-17 2007-07-04 David Ovadia Process for the preparation of substituted cyanophenoxy-pyrimidinyloxy -phenyl acrylate derivatives
IL181125A0 (en) * 2007-02-01 2007-07-04 Maktheshim Chemical Works Ltd Polymorphs of 3-(e)-2-{2-[6-(2-
CN103073505B (zh) * 2013-01-28 2015-11-18 泰州百力化学股份有限公司 4-氯-6-甲氧基嘧啶合成4，6-二氯嘧啶的方法
CN103242236B (zh) * 2013-04-26 2014-11-19 扬州大学 以丙烯腈为氮源合成取代苯并咪唑的制备方法
WO2019016111A1 (en) * 2017-07-18 2019-01-24 Lonza Ltd PROCESS FOR THE PREPARATION OF CHLORINATED S-PROPYLTHIOBARBITURIC ACID
WO2020126716A1 (en) * 2018-12-20 2020-06-25 Basf Se Manufacturing method for an aromatic isocyanate compound

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3220105A1 (de) * 1982-05-28 1983-12-01 Bayer Ag, 5090 Leverkusen Verfahren zur herstellung in (alpha)-stellung chlorierten stickstoff-heterocyclen
GB9408270D0 (en) * 1994-04-26 1994-06-15 Zeneca Ltd Chemical process
US6160117A (en) * 1997-11-06 2000-12-12 Zeneca Limited Chemical process
AU2801500A (en) * 1999-02-05 2000-08-25 Syngenta Participations Ag Method of producing substituted pyrimidine derivatives
DE19935322A1 (de) * 1999-07-28 2001-02-01 Bayer Ag Verfahren zur Herstellung von 4,6-Dichlorpyrimidin mit Phosgen

Also Published As

Publication number Publication date
KR20030011893A (ko) 2003-02-11
WO2002000628A2 (en) 2002-01-03
WO2002000628A3 (en) 2002-04-11
JP2004501900A (ja) 2004-01-22
AR030296A1 (es) 2003-08-20
EP1296957A2 (en) 2003-04-02
IL153099A0 (en) 2003-06-24
AU2001264095A1 (en) 2002-01-08
CN1697829A (zh) 2005-11-16
US20020042514A1 (en) 2002-04-11
HUP0400474A3 (en) 2006-01-30
BR0111960A (pt) 2003-07-29

Similar Documents

Publication Publication Date Title
NO2022001I1 (no) Pazopanib
DE60009511D1 (de) Nematizide trifluorbutene
GB0124627D0 (en) Novel compounds
EP1432714A4 (en) CHEMICAL COMPOUNDS
NO20053115D0 (no) Fremgangsmate for fremstilling av 2'-forgrenede nukleosider.
MXPA03006001A (es) Derivados de fosfonato de nucleosido aciclico novedoso, sales de estos y proceso para la preparacion de los mismos.
MXPA03008754A (es) Derivados de piridina fundidos para utilizarse como agonistas receptores vaniloide para tratar dolor.
WO2004028454A3 (en) 1, 3, 5-triazines for treatment of viral diseases
MY130718A (en) Antitumor compounds and methods
MXPA02010088A (es) Derivados de ecteinascidina antitumorales.
WO2003051886A8 (en) Pyrazolopyridazine derivatives
ATE347555T1 (de) 6-aminomorphinanderivate, herstellungsverfahren dafür und deren verwendung
HUP0400474A2 (hu) Klórozott pirimidinek előállítása
MXPA04006041A (es) Antivirales de piridoquinoxalina.
DK1383742T3 (da) Syntese og fremgangsmåder til anvendelse af tetrahydroindolonanaloge og derivater
MXPA04003755A (es) Endoprotesis vasculares.
ATE298742T1 (de) Zykloalkenylsulfonamidderivate
DE60210970D1 (de) Mutante formen von etxb und ctxb und ihre verwendung als träger
EP1613606A4 (en) PROCESS FOR PREPARING 2,3,5,6-SUBSTITUTED 3H-PYRIMIDIN-4-ONES
NO934040D0 (no) Finfordelt silisium innbefattende et overflatebundet halogen, fremgangsmaate for fremstilling og anvendelse derav
CY1110212T1 (el) Χαμηλης υγροσκοπικοτητας αριπιπραζολη ως φαρμακευτικη ουσια και μεθοδοι για την παρασκευη της
DK0833847T3 (da) Krystaller af fregmenter af CD40-ligand og deres anvendelse
HUP0301608A2 (hu) Klórozott pirimidinek szintézise
HUP0101446A2 (hu) Új triszulfidok
GR20010100524A (el) Αναρτηση διακοσμητικων παραστασεων

Legal Events

Date Code Title Description
FD9A Lapse of provisional protection due to non-payment of fees