HUP0203976A3 - Adenozine a3 receptors, process for their preparation and pharmaceutical compositions containing them - Google Patents

Adenozine a3 receptors, process for their preparation and pharmaceutical compositions containing them

Info

Publication number
HUP0203976A3
HUP0203976A3 HU0203976A HUP0203976A HUP0203976A3 HU P0203976 A3 HUP0203976 A3 HU P0203976A3 HU 0203976 A HU0203976 A HU 0203976A HU P0203976 A HUP0203976 A HU P0203976A HU P0203976 A3 HUP0203976 A3 HU P0203976A3
Authority
HU
Hungary
Prior art keywords
adenozine
receptors
preparation
pharmaceutical compositions
compositions containing
Prior art date
Application number
HU0203976A
Other languages
English (en)
Hungarian (hu)
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Priority to HU0203976A priority Critical patent/HUP0203976A3/hu
Publication of HU0203976D0 publication Critical patent/HU0203976D0/hu
Priority to BR0316355-5A priority patent/BR0316355A/pt
Priority to YUP-2005/0364A priority patent/RS51320B/sr
Priority to PT03773882T priority patent/PT1560828E/pt
Priority to EP03773882A priority patent/EP1560828B9/en
Priority to HK05109885.4A priority patent/HK1077819B/en
Priority to ES03773882T priority patent/ES2263039T3/es
Priority to PL376837A priority patent/PL376837A1/pl
Priority to MXPA05005198A priority patent/MXPA05005198A/es
Priority to AU2003282263A priority patent/AU2003282263B2/en
Priority to DK03773882T priority patent/DK1560828T3/da
Priority to EA200500830A priority patent/EA007595B1/ru
Priority to HR20050540A priority patent/HRP20050540A2/xx
Priority to CNB2003801062293A priority patent/CN1332960C/zh
Priority to AT03773882T priority patent/ATE325123T1/de
Priority to SI200330299T priority patent/SI1560828T1/sl
Priority to JP2004552920A priority patent/JP4533148B2/ja
Priority to KR1020057008683A priority patent/KR20050088291A/ko
Priority to CA2505910A priority patent/CA2505910C/en
Priority to UAA200505875A priority patent/UA78889C2/uk
Priority to PCT/HU2003/000095 priority patent/WO2004046146A1/en
Priority to MEP-190/08A priority patent/MEP19008A/xx
Priority to NZ540029A priority patent/NZ540029A/en
Priority to DE60305058T priority patent/DE60305058T2/de
Priority to TW092131901A priority patent/TWI248934B/zh
Priority to ARP030104200A priority patent/AR041968A1/es
Publication of HUP0203976A2 publication Critical patent/HUP0203976A2/hu
Publication of HUP0203976A3 publication Critical patent/HUP0203976A3/hu
Priority to IL168516A priority patent/IL168516A/en
Priority to TNP2005000133A priority patent/TNSN05133A1/en
Priority to ZA200503807A priority patent/ZA200503807B/en
Priority to US11/130,429 priority patent/US7419977B2/en
Priority to IS7874A priority patent/IS2456B/is
Priority to MA28334A priority patent/MA27501A1/fr
Priority to NO20052866A priority patent/NO20052866L/no
Priority to CO05057645A priority patent/CO5690577A2/es
Priority to CY20061101054T priority patent/CY1105180T1/el
Priority to US12/140,512 priority patent/US7709489B2/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/02—Nasal agents, e.g. decongestants
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/16—Central respiratory analeptics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
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    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
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    • A61P25/00—Drugs for disorders of the nervous system
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/06—Antiarrhythmics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Pulmonology (AREA)
  • Diabetes (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Psychiatry (AREA)
  • Immunology (AREA)
  • Urology & Nephrology (AREA)
  • Dermatology (AREA)
  • Hematology (AREA)
  • Pain & Pain Management (AREA)
  • Epidemiology (AREA)
  • Obesity (AREA)
  • Rheumatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Psychology (AREA)
  • Endocrinology (AREA)
  • Hospice & Palliative Care (AREA)
  • Emergency Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Otolaryngology (AREA)
  • Vascular Medicine (AREA)
HU0203976A 2002-11-15 2002-11-15 Adenozine a3 receptors, process for their preparation and pharmaceutical compositions containing them HUP0203976A3 (en)

Priority Applications (36)

Application Number Priority Date Filing Date Title
HU0203976A HUP0203976A3 (en) 2002-11-15 2002-11-15 Adenozine a3 receptors, process for their preparation and pharmaceutical compositions containing them
DE60305058T DE60305058T2 (de) 2002-11-15 2003-11-11 Imidazoquinoline derivate als adenosine a3 rezeptor liganden
CA2505910A CA2505910C (en) 2002-11-15 2003-11-11 Imidazoquinoline derivatives as adenosine a3 receptor ligands
UAA200505875A UA78889C2 (en) 2002-11-15 2003-11-11 Imidazoquinoline derivatives as an adenosine a3 receptor ligands
PT03773882T PT1560828E (pt) 2002-11-15 2003-11-11 Derivados de imidazoquinolina como ligandos receptores a3 da adenosina
EP03773882A EP1560828B9 (en) 2002-11-15 2003-11-11 Imidazoquinoline derivatives as adenosine a3 receptor ligands
HK05109885.4A HK1077819B (en) 2002-11-15 2003-11-11 Imidazoquinoline derivatives as adenosine a3 receptor ligands
MEP-190/08A MEP19008A (en) 2002-11-15 2003-11-11 Imidazoquinoline derivatives as adenosine a3 receptor ligands
PL376837A PL376837A1 (pl) 2002-11-15 2003-11-11 Pochodne imidazochinoliny jako ligandy receptora adenozyny A3
MXPA05005198A MXPA05005198A (es) 2002-11-15 2003-11-11 Derivados de imidazoquinolina, como ligandos del receptor a3 de adenosina.
AU2003282263A AU2003282263B2 (en) 2002-11-15 2003-11-11 Imidazoquinoline derivatives as adenosine A3 receptor ligands
DK03773882T DK1560828T3 (da) 2002-11-15 2003-11-11 Imidazoquinolinderivater som adenosin-A3-receptorligander
EA200500830A EA007595B1 (ru) 2002-11-15 2003-11-11 Производные имидазохинолина в качестве лигандов аденозиновых арецепторов
HR20050540A HRP20050540A2 (en) 2002-11-15 2003-11-11 Imidazoquinoline derivatives as adenosine a3 receptor ligands
CNB2003801062293A CN1332960C (zh) 2002-11-15 2003-11-11 作为腺苷a3受体配体的咪唑并喹啉衍生物
AT03773882T ATE325123T1 (de) 2002-11-15 2003-11-11 Imidazoquinoline derivate als adenosine a3 rezeptor liganden
SI200330299T SI1560828T1 (sl) 2002-11-15 2003-11-11 Imidazokinolinski derivati kot adenozin A3 receptorski ligandi
JP2004552920A JP4533148B2 (ja) 2002-11-15 2003-11-11 アデノシンａ３受容体リガンドとしてのイミダゾキノリン誘導体
KR1020057008683A KR20050088291A (ko) 2002-11-15 2003-11-11 아데노신 ａ３ 수용체 리간드로서의 이미다조퀴놀린 유도체
BR0316355-5A BR0316355A (pt) 2002-11-15 2003-11-11 Derivados de imidazoquinolina como ligantes de receptores de adenosina a3
PCT/HU2003/000095 WO2004046146A1 (en) 2002-11-15 2003-11-11 Imidazoquinoline derivatives as adenosine a3 receptor ligands
YUP-2005/0364A RS51320B (sr) 2002-11-15 2003-11-11 Derivati imidazohinolina kao veznici a3 receptora adenozina
ES03773882T ES2263039T3 (es) 2002-11-15 2003-11-11 Derivados de imidazoquinolina como ligandos del receptor a3 de adenosina.
NZ540029A NZ540029A (en) 2002-11-15 2003-11-11 Imidazoquinoline derivatives as adenosine A3 receptor ligands
TW092131901A TWI248934B (en) 2002-11-15 2003-11-14 Compounds of adenosine A3 receptor ligands and the process for manufacturing the same
ARP030104200A AR041968A1 (es) 2002-11-15 2003-11-14 Compuestos derivados de imidazol como ligandos del receptor de adenosina
IL168516A IL168516A (en) 2002-11-15 2005-05-10 Imidazoquinoline derivatives as adenosine a3 receptor ligands
TNP2005000133A TNSN05133A1 (en) 2002-11-15 2005-05-10 Imidazoquinoline derivatives as adenosine a3 receptor ligands
ZA200503807A ZA200503807B (en) 2002-11-15 2005-05-11 Imidazoquinoline derivatives as adenosine A3 receptor ligands
US11/130,429 US7419977B2 (en) 2002-11-15 2005-05-16 Imidazoquinoline derivatives as adenosine A3 receptor ligands
IS7874A IS2456B (is) 2002-11-15 2005-05-31 Ímídasókínólínafleiður sem adenósín A3 viðtakabindlar
MA28334A MA27501A1 (fr) 2002-11-15 2005-06-13 Derives d'imidazoquinoline en tant que ligands recepteurs de l'adenosine a3
NO20052866A NO20052866L (no) 2002-11-15 2005-06-13 Imidazokinolinderivater som adenosin A3 reseptorligander
CO05057645A CO5690577A2 (es) 2002-11-15 2005-06-14 Derivados de imidazoquinolina como ligandos receptores de adenosina a3
CY20061101054T CY1105180T1 (el) 2002-11-15 2006-07-28 Παραγωγα ιμιδαζοκινολινης ως α3 συνδετες υποδοχεων αδενοσινης
US12/140,512 US7709489B2 (en) 2002-11-15 2008-06-17 Imidazoquinoline derivatives as adenosine A3 receptor ligands

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU0203976A HUP0203976A3 (en) 2002-11-15 2002-11-15 Adenozine a3 receptors, process for their preparation and pharmaceutical compositions containing them

Publications (3)

Publication Number Publication Date
HU0203976D0 HU0203976D0 (en) 2003-01-28
HUP0203976A2 HUP0203976A2 (hu) 2004-07-28
HUP0203976A3 true HUP0203976A3 (en) 2004-08-30

Family

ID=90001561

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0203976A HUP0203976A3 (en) 2002-11-15 2002-11-15 Adenozine a3 receptors, process for their preparation and pharmaceutical compositions containing them

Country Status (34)

Country Link
US (2) US7419977B2 (https=)
EP (1) EP1560828B9 (https=)
JP (1) JP4533148B2 (https=)
KR (1) KR20050088291A (https=)
CN (1) CN1332960C (https=)
AR (1) AR041968A1 (https=)
AT (1) ATE325123T1 (https=)
AU (1) AU2003282263B2 (https=)
BR (1) BR0316355A (https=)
CA (1) CA2505910C (https=)
CO (1) CO5690577A2 (https=)
CY (1) CY1105180T1 (https=)
DE (1) DE60305058T2 (https=)
DK (1) DK1560828T3 (https=)
EA (1) EA007595B1 (https=)
ES (1) ES2263039T3 (https=)
HR (1) HRP20050540A2 (https=)
HU (1) HUP0203976A3 (https=)
IL (1) IL168516A (https=)
IS (1) IS2456B (https=)
MA (1) MA27501A1 (https=)
ME (1) MEP19008A (https=)
MX (1) MXPA05005198A (https=)
NO (1) NO20052866L (https=)
NZ (1) NZ540029A (https=)
PL (1) PL376837A1 (https=)
PT (1) PT1560828E (https=)
RS (1) RS51320B (https=)
SI (1) SI1560828T1 (https=)
TN (1) TNSN05133A1 (https=)
TW (1) TWI248934B (https=)
UA (1) UA78889C2 (https=)
WO (1) WO2004046146A1 (https=)
ZA (1) ZA200503807B (https=)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HUP0105406A3 (en) * 2001-12-21 2003-12-29 Sanofi Aventis Imidazo[1,2-a]quinolin derivatives, process for their preparation, pharmaceutical compositions thereof and intermediates
HUP0203976A3 (en) * 2002-11-15 2004-08-30 Sanofi Aventis Adenozine a3 receptors, process for their preparation and pharmaceutical compositions containing them
HUP0400812A2 (en) * 2004-04-19 2006-02-28 Sanofi Aventis Crystalline forms of 2-amino-3-cyano-quinoline derivatives, process for their preparation and pharmaceutical compositions containing them
GT200600381A (es) 2005-08-25 2007-03-28 Compuestos organicos
US20090088403A1 (en) * 2007-05-07 2009-04-02 Randy Blakely A3 adenosine receptors as targets for the modulation of central serotonergic signaling
HUP0700395A2 (en) * 2007-06-07 2009-03-02 Sanofi Aventis Substituted [1,2,4] triazolo [1,5-a] quinolines, process for their preparation, pharmaceutical compositions thereof, and intermediates
WO2011010306A1 (en) 2009-07-21 2011-01-27 Ramot At Tel-Aviv University Ltd. A3 adenosine receptor ligands for modulation of pigmentation
DK2950649T3 (da) 2013-02-01 2020-05-04 Wellstat Therapeutics Corp Aminforbindelser med antiinflammations-, antisvampe-, antiparasit- og anticanceraktivitet
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