HU217439B - Tetrazolil-epesav-származékok, eljárás előállításukra és ezeket tartalmazó gyógyszerkészítmények - Google Patents

Tetrazolil-epesav-származékok, eljárás előállításukra és ezeket tartalmazó gyógyszerkészítmények Download PDF

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Publication number
HU217439B
HU217439B HU9401443A HU9401443A HU217439B HU 217439 B HU217439 B HU 217439B HU 9401443 A HU9401443 A HU 9401443A HU 9401443 A HU9401443 A HU 9401443A HU 217439 B HU217439 B HU 217439B
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HU
Hungary
Prior art keywords
formula
group
bile acid
hydrogen
compound
Prior art date
Application number
HU9401443A
Other languages
English (en)
Hungarian (hu)
Other versions
HUT67390A (en
HU9401443D0 (en
Inventor
Alfons Enhsen
Heiner Glombik
Werner Kramer
Günther Wess
Original Assignee
Hoechst Ag.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Ag. filed Critical Hoechst Ag.
Publication of HU9401443D0 publication Critical patent/HU9401443D0/hu
Publication of HUT67390A publication Critical patent/HUT67390A/hu
Publication of HU217439B publication Critical patent/HU217439B/hu

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J9/00Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane
    • C07J9/005Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane containing a carboxylic function directly attached or attached by a chain containing only carbon atoms to the cyclopenta[a]hydrophenanthrene skeleton
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J17/00Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0005Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0094Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 containing nitrile radicals, including thiocyanide radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J43/00Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Toxicology (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Obesity (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
HU9401443A 1993-05-08 1994-05-06 Tetrazolil-epesav-származékok, eljárás előállításukra és ezeket tartalmazó gyógyszerkészítmények HU217439B (hu)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4315368 1993-05-08

Publications (3)

Publication Number Publication Date
HU9401443D0 HU9401443D0 (en) 1994-08-29
HUT67390A HUT67390A (en) 1995-04-28
HU217439B true HU217439B (hu) 2000-01-28

Family

ID=6487579

Family Applications (1)

Application Number Title Priority Date Filing Date
HU9401443A HU217439B (hu) 1993-05-08 1994-05-06 Tetrazolil-epesav-származékok, eljárás előállításukra és ezeket tartalmazó gyógyszerkészítmények

Country Status (19)

Country Link
US (1) US5466815A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
EP (1) EP0624596B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
JP (1) JP3476157B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
KR (1) KR100333149B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
AT (1) ATE163938T1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
AU (1) AU666440B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CA (1) CA2123048C (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CY (1) CY2119B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CZ (1) CZ289515B6 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DE (1) DE59405410D1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DK (1) DK0624596T3 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
ES (1) ES2115096T3 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
FI (1) FI942075L (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
GR (1) GR3026496T3 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
HU (1) HU217439B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IL (1) IL109581A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NO (1) NO304795B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NZ (1) NZ260469A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
TW (1) TW289757B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)

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TW289020B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) * 1993-05-08 1996-10-21 Hoechst Sktiengesellschaft
US6323190B1 (en) 1998-07-31 2001-11-27 The Univeristy Of Georgia Research Foundation, Inc. Estrogen mimetics lacking reproductive tract effects
JP2002543216A (ja) 1999-04-30 2002-12-17 アーチ ディベロップメント コーポレイション ステロイド誘導体
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CN1498222A (zh) * 2001-02-08 2004-05-19 芝加哥大学 类固醇衍生物
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Publication number Priority date Publication date Assignee Title
DE3930696A1 (de) * 1989-09-14 1991-03-28 Hoechst Ag Gallensaeurederivate, verfahren zu ihrer herstellung, verwendung als arzneimittel
IL100240A (en) * 1990-12-06 1995-10-31 Hoechst Ag Bile acid derivatives process for their preparation and use of these compounds as pharmaceuticals

Also Published As

Publication number Publication date
NO941677D0 (no) 1994-05-06
GR3026496T3 (en) 1998-07-31
EP0624596B1 (de) 1998-03-11
DE59405410D1 (de) 1998-04-16
FI942075A7 (fi) 1994-11-09
IL109581A0 (en) 1994-08-26
AU6194794A (en) 1994-11-10
IL109581A (en) 1998-03-10
US5466815A (en) 1995-11-14
EP0624596A3 (de) 1995-06-07
KR100333149B1 (ko) 2002-09-19
ATE163938T1 (de) 1998-03-15
CZ113594A3 (en) 1994-12-15
CZ289515B6 (cs) 2002-02-13
EP0624596A2 (de) 1994-11-17
JP3476157B2 (ja) 2003-12-10
FI942075L (fi) 1994-11-09
FI942075A0 (fi) 1994-05-05
ES2115096T3 (es) 1998-06-16
JPH06329695A (ja) 1994-11-29
TW289757B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1996-11-01
CY2119B1 (en) 2002-04-26
CA2123048A1 (en) 1994-11-09
AU666440B2 (en) 1996-02-08
NZ260469A (en) 1995-03-28
NO304795B1 (no) 1999-02-15
HUT67390A (en) 1995-04-28
HU9401443D0 (en) 1994-08-29
NO941677L (no) 1994-11-09
CA2123048C (en) 2005-11-29
DK0624596T3 (da) 1998-10-07

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