HU187572B - Process for preparing 1,5-diphenyl-pyrazolin-3-one derivatives - Google Patents

Process for preparing 1,5-diphenyl-pyrazolin-3-one derivatives Download PDF

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Publication number
HU187572B
HU187572B HU822675A HU267582A HU187572B HU 187572 B HU187572 B HU 187572B HU 822675 A HU822675 A HU 822675A HU 267582 A HU267582 A HU 267582A HU 187572 B HU187572 B HU 187572B
Authority
HU
Hungary
Prior art keywords
formula
compound
hydrogen
alkyl
alkoxy
Prior art date
Application number
HU822675A
Other languages
English (en)
Hungarian (hu)
Inventor
Henning Heinemann
Daniel Jasserand
Wolfgang Milkowski
Dimitri Yavordios
Horst Zeugner
Original Assignee
Kali-Chemie Pharma Gmbh,De
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kali-Chemie Pharma Gmbh,De filed Critical Kali-Chemie Pharma Gmbh,De
Publication of HU187572B publication Critical patent/HU187572B/hu

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/18One oxygen or sulfur atom
    • C07D231/20One oxygen atom attached in position 3 or 5
    • C07D231/22One oxygen atom attached in position 3 or 5 with aryl radicals attached to ring nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pulmonology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Immunology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Detergent Compositions (AREA)
  • Luminescent Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
HU822675A 1981-08-20 1982-08-18 Process for preparing 1,5-diphenyl-pyrazolin-3-one derivatives HU187572B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19813132915 DE3132915A1 (de) 1981-08-20 1981-08-20 1,5-diphenylpyrazolin-3-on-verbindungen sowie verfahren und zwischenprodukte zu ihrer herstellung und diese verbindungen enthaltende arzneimittel

Publications (1)

Publication Number Publication Date
HU187572B true HU187572B (en) 1986-01-28

Family

ID=6139713

Family Applications (1)

Application Number Title Priority Date Filing Date
HU822675A HU187572B (en) 1981-08-20 1982-08-18 Process for preparing 1,5-diphenyl-pyrazolin-3-one derivatives

Country Status (20)

Country Link
US (2) US4442102A (US20100223739A1-20100909-C00005.png)
EP (1) EP0072960B1 (US20100223739A1-20100909-C00005.png)
JP (1) JPS5839668A (US20100223739A1-20100909-C00005.png)
AT (1) ATE43841T1 (US20100223739A1-20100909-C00005.png)
AU (1) AU555215B2 (US20100223739A1-20100909-C00005.png)
CA (1) CA1208643A (US20100223739A1-20100909-C00005.png)
DD (1) DD202563A5 (US20100223739A1-20100909-C00005.png)
DE (2) DE3132915A1 (US20100223739A1-20100909-C00005.png)
DK (1) DK149947C (US20100223739A1-20100909-C00005.png)
ES (1) ES8306143A1 (US20100223739A1-20100909-C00005.png)
FI (1) FI73673C (US20100223739A1-20100909-C00005.png)
GR (2) GR76272B (US20100223739A1-20100909-C00005.png)
HU (1) HU187572B (US20100223739A1-20100909-C00005.png)
IE (1) IE55377B1 (US20100223739A1-20100909-C00005.png)
IL (1) IL66580A (US20100223739A1-20100909-C00005.png)
NO (1) NO158185C (US20100223739A1-20100909-C00005.png)
NZ (1) NZ201643A (US20100223739A1-20100909-C00005.png)
PH (1) PH19107A (US20100223739A1-20100909-C00005.png)
PT (1) PT75353B (US20100223739A1-20100909-C00005.png)
ZA (1) ZA825381B (US20100223739A1-20100909-C00005.png)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3442860A1 (de) * 1984-11-24 1986-05-28 Kali-Chemie Pharma Gmbh, 3000 Hannover 5-alkyl-1-phenyl-2-piperazinoalkylpyrazolin-3- on-verbindungen sowie verfahren und zwischenprodukte zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
NZ524193A (en) * 2000-08-14 2004-12-24 Ortho Mcneil Pharm Inc Substituted pyrazoles
CA2488202C (en) * 2002-06-12 2011-03-08 Chemocentryx, Inc. 1-aryl-4-substituted piperazine derivatives for use as ccr1 antagonists for the treatment of inflammation and immune disorders
US20050256130A1 (en) * 2002-06-12 2005-11-17 Chemocentryx, Inc. Substituted piperazines
US7842693B2 (en) * 2002-06-12 2010-11-30 Chemocentryx, Inc. Substituted piperazines
US7589199B2 (en) * 2002-06-12 2009-09-15 Chemocentryx, Inc. Substituted piperazines
EP1720545B1 (en) * 2004-03-03 2014-10-29 ChemoCentryx, Inc. Bicyclic and bridged nitrogen heterocycles
US7435831B2 (en) * 2004-03-03 2008-10-14 Chemocentryx, Inc. Bicyclic and bridged nitrogen heterocycles
WO2011051958A1 (en) * 2009-10-30 2011-05-05 E.I. Du Pont De Nemours And Company Fungicidal pyrazolones

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE74912C (US20100223739A1-20100909-C00005.png) *
DE66610C (de) * FARBWERKE VORM. MEISTER LUCIUS & BRÜNING in Höchst a. M Verfahren zur Darstellung von Oxaethylmethylphenylpyrazolon
GB666578A (en) * 1948-01-10 1952-02-13 Luxema Process for the preparation of derivatives of 1, 2, 3 substituted pyrazolones and derivatives obtained by this process
US3169966A (en) * 1961-01-24 1965-02-16 Ciba Geigy Corp Aminopyrazoles
DE2824764A1 (de) * 1978-06-06 1979-12-20 Hoechst Ag Neue pyridylpiperazinderivate und verfahren zu ihrer herstellung
DE2828529A1 (de) * 1978-06-29 1980-01-17 Kali Chemie Pharma Gmbh Neue 5-phenylpyrazol-derivate, verfahren zu deren herstellung und arzneimittel

Also Published As

Publication number Publication date
FI73673C (fi) 1987-11-09
DK372382A (da) 1983-02-21
ATE43841T1 (de) 1989-06-15
IL66580A0 (en) 1982-12-31
IE55377B1 (en) 1990-08-29
NZ201643A (en) 1985-04-30
NO822827L (no) 1983-02-21
PT75353A (en) 1982-08-01
NO158185C (no) 1988-07-27
ES515107A0 (es) 1983-05-01
NO158185B (no) 1988-04-18
FI73673B (fi) 1987-07-31
GR76272B (US20100223739A1-20100909-C00005.png) 1984-08-04
CA1208643A (en) 1986-07-29
IE822002L (en) 1983-02-20
DD202563A5 (de) 1983-09-21
EP0072960A2 (de) 1983-03-02
EP0072960B1 (de) 1989-06-07
AU8742482A (en) 1983-02-24
FI822883L (fi) 1983-02-21
DK149947B (da) 1986-11-03
IL66580A (en) 1985-10-31
US4442102A (en) 1984-04-10
US4515944A (en) 1985-05-07
DE3132915A1 (de) 1983-03-03
PH19107A (en) 1986-01-02
DE3279756D1 (en) 1989-07-13
EP0072960A3 (en) 1984-03-07
DK149947C (da) 1987-06-15
JPH0375542B2 (US20100223739A1-20100909-C00005.png) 1991-12-02
GR78228B (US20100223739A1-20100909-C00005.png) 1984-09-26
ZA825381B (en) 1983-05-25
FI822883A0 (fi) 1982-08-19
ES8306143A1 (es) 1983-05-01
AU555215B2 (en) 1986-09-18
JPS5839668A (ja) 1983-03-08
PT75353B (en) 1984-08-01

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Legal Events

Date Code Title Description
HU90 Patent valid on 900628
HMM4 Cancellation of final prot. due to non-payment of fee