HRP20030923A2 - Novel piperidinecarboxamide derivatives, method for prreparing same and pharmaceutical compositions containing same - Google Patents

Novel piperidinecarboxamide derivatives, method for prreparing same and pharmaceutical compositions containing same Download PDF

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Publication number
HRP20030923A2
HRP20030923A2 HR20030923A HRP20030923A HRP20030923A2 HR P20030923 A2 HRP20030923 A2 HR P20030923A2 HR 20030923 A HR20030923 A HR 20030923A HR P20030923 A HRP20030923 A HR P20030923A HR P20030923 A2 HRP20030923 A2 HR P20030923A2
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HR
Croatia
Prior art keywords
formula
compound
dichlorophenyl
morpholin
piperidin
Prior art date
Application number
HR20030923A
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English (en)
Croatian (hr)
Inventor
Xavier Emondsalt
Vincenzo Proietto
Original Assignee
Sanofi Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by Sanofi Synthelabo filed Critical Sanofi Synthelabo
Publication of HRP20030923A2 publication Critical patent/HRP20030923A2/hr

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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/06Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • AHUMAN NECESSITIES
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HR20030923A 2001-05-21 2003-11-12 Novel piperidinecarboxamide derivatives, method for prreparing same and pharmaceutical compositions containing same HRP20030923A2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0106691A FR2824828B1 (fr) 2001-05-21 2001-05-21 Nouveaux derives de piperidinecarboxamide, un procede pour leur preparation et les compositions pharmaceutiques les contenant
PCT/FR2002/001663 WO2002094821A1 (fr) 2001-05-21 2002-05-17 Nouveaux derives de piperidinecarboxamide, un procede pour leur preparation et les compositions pharmaceutiques les contenant

Publications (1)

Publication Number Publication Date
HRP20030923A2 true HRP20030923A2 (en) 2004-02-29

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Application Number Title Priority Date Filing Date
HR20030923A HRP20030923A2 (en) 2001-05-21 2003-11-12 Novel piperidinecarboxamide derivatives, method for prreparing same and pharmaceutical compositions containing same

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US (2) US20040180890A1 (bg)
EP (1) EP1395582B1 (bg)
JP (1) JP2004529968A (bg)
KR (1) KR20030097886A (bg)
CN (1) CN1249059C (bg)
AR (1) AR035247A1 (bg)
AT (1) ATE294798T1 (bg)
AU (1) AU2002313065B2 (bg)
BG (1) BG108341A (bg)
BR (1) BR0209877A (bg)
CA (1) CA2445631A1 (bg)
CZ (1) CZ20033132A3 (bg)
DE (1) DE60204015T2 (bg)
DK (1) DK1395582T3 (bg)
EA (1) EA006236B1 (bg)
EE (1) EE200300553A (bg)
ES (1) ES2242032T3 (bg)
FR (1) FR2824828B1 (bg)
HK (1) HK1060129A1 (bg)
HR (1) HRP20030923A2 (bg)
HU (1) HUP0401563A2 (bg)
IL (1) IL158660A0 (bg)
IS (1) IS7008A (bg)
MA (1) MA27022A1 (bg)
MX (1) MXPA03010133A (bg)
NO (1) NO20035163D0 (bg)
NZ (1) NZ529206A (bg)
PL (1) PL367341A1 (bg)
PT (1) PT1395582E (bg)
SK (1) SK14192003A3 (bg)
TN (1) TNSN03118A1 (bg)
TW (1) TWI258480B (bg)
UA (1) UA75400C2 (bg)
WO (1) WO2002094821A1 (bg)
YU (1) YU86603A (bg)
ZA (1) ZA200308344B (bg)

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WO2004055011A1 (en) * 2002-12-13 2004-07-01 Smithkline Beecham Corporation Heterocyclic compounds as ccr5 antagonists
FR2873373B1 (fr) * 2004-07-23 2006-09-08 Sanofi Synthelabo Derives de 4-arylmorpholin-3-one, leur preparation et leur application en therapeutique
US20070219214A1 (en) * 2006-02-01 2007-09-20 Solvay Pharmaceuticals Gmbh Dual NK2/NK3-antagonists, pharmaceutical compositions comprising them, and processes for their preparation
JP2009525308A (ja) * 2006-02-01 2009-07-09 ゾルファイ ファーマスーティカルズ ゲゼルシャフト ミット ベシュレンクテル ハフツング 新規のnk2/nk3−デュアルアンタゴニスト、それらを含有する医薬組成物並びにそれらの製造方法
FR2912058A1 (fr) * 2007-02-07 2008-08-08 Sanofi Aventis Sa Utilisation d'un compose antagoniste des recepteurs nk2 de la neurokinine a pour la preparation de medicaments utiles pour la prevention et le traitement des dysfonctions sexuelles
EP2244716B1 (en) * 2008-01-11 2019-09-25 United Paragon Associates Inc. Fertilized egg isolate and use thereof
US20110152233A1 (en) 2009-12-18 2011-06-23 Henner Knust Pyrrolidine compounds
KR101756495B1 (ko) * 2010-03-11 2017-07-10 다이닛본 스미토모 세이야꾸 가부시끼가이샤 N-아실 시클릭 아민 유도체 또는 이의 의약상 허용되는 염
US10314835B2 (en) 2014-06-25 2019-06-11 Emory University Methods of managing conditioned fear with neurokinin receptor antagonists
JPWO2020101017A1 (ja) * 2018-11-15 2021-09-30 国立大学法人九州大学 Il−31介在性疾患の予防又は治療剤及び医薬組成物

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US5689663A (en) * 1992-06-19 1997-11-18 Microsoft Corporation Remote controller user interface and methods relating thereto
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CN1518549A (zh) 2004-08-04
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ZA200308344B (en) 2004-10-27
UA75400C2 (en) 2006-04-17
CZ20033132A3 (cs) 2004-02-18
EA200301087A1 (ru) 2004-04-29
FR2824828B1 (fr) 2005-05-20
TWI258480B (en) 2006-07-21
ES2242032T3 (es) 2005-11-01
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AR035247A1 (es) 2004-05-05
US20040180890A1 (en) 2004-09-16
EP1395582A1 (fr) 2004-03-10
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YU86603A (sh) 2006-05-25
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BG108341A (bg) 2004-12-30
FR2824828A1 (fr) 2002-11-22
TNSN03118A1 (fr) 2005-12-23
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BR0209877A (pt) 2004-06-08
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IL158660A0 (en) 2004-05-12
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CA2445631A1 (fr) 2002-11-28
JP2004529968A (ja) 2004-09-30
MA27022A1 (fr) 2004-12-20
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US20080261976A1 (en) 2008-10-23
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