HN2001000261A - NEW DERIVATIVES OF PIRAZOLPIRIDINA REPLACED WITH PIRIDINE. - Google Patents

NEW DERIVATIVES OF PIRAZOLPIRIDINA REPLACED WITH PIRIDINE.

Info

Publication number
HN2001000261A
HN2001000261A HN2001000261A HN2001000261A HN2001000261A HN 2001000261 A HN2001000261 A HN 2001000261A HN 2001000261 A HN2001000261 A HN 2001000261A HN 2001000261 A HN2001000261 A HN 2001000261A HN 2001000261 A HN2001000261 A HN 2001000261A
Authority
HN
Honduras
Prior art keywords
pirazolpiridina
piridine
replaced
new derivatives
circulatories
Prior art date
Application number
HN2001000261A
Other languages
Spanish (es)
Inventor
Johannes Peter Stasch
Achim Feurer
Stefan Weigand
Elke Sthal
Flubacher Dietmar
Cristina Alonso Alija
Frank Wunder
Dieter Lang
Klaus Dembowsky
Alexander Straub
Elisabeth Perzborn
Original Assignee
Basf Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Ag filed Critical Basf Ag
Publication of HN2001000261A publication Critical patent/HN2001000261A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

LA PRESENTE INVENCION SE REFIERE A NUEVOS COMPUESTOS QQUIMICOS, LOS CUALES ESTIMULAN LA GUANILATO CICLASA SOLUBLE, A SU PREPARACION Y A SU UTILIZACION COMO MEDICAMENTOS, EN ESPECIAL COMO MEDICAMENTOS PARA EL TRATAMIENTO DE ENFERMEDADES CORONARIO - CIRCULATORIAS.THE PRESENT INVENTION REFERS TO NEW CHEMICAL COMPOUNDS, WHICH STIMULATE THE SOLUBLE CYCLING GUANILATE, ITS PREPARATION AND ITS USE AS MEDICINES, IN SPECIAL AS MEDICATIONS FOR THE TREATMENT OF CORONARY DISEASES - CIRCULATORIES.

HN2001000261A 2000-11-22 2001-11-21 NEW DERIVATIVES OF PIRAZOLPIRIDINA REPLACED WITH PIRIDINE. HN2001000261A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10057753 2000-11-22
DE10131987A DE10131987A1 (en) 2000-11-22 2001-07-02 New pyridinyl-substituted pyrazolo (3,4-b) pyridine derivatives, are soluble guanylate cyclase stimulants useful e.g. for treating cardiovascular or central nervous system diseases, sexual dysfunction or inflammation

Publications (1)

Publication Number Publication Date
HN2001000261A true HN2001000261A (en) 2002-01-30

Family

ID=7664122

Family Applications (1)

Application Number Title Priority Date Filing Date
HN2001000261A HN2001000261A (en) 2000-11-22 2001-11-21 NEW DERIVATIVES OF PIRAZOLPIRIDINA REPLACED WITH PIRIDINE.

Country Status (12)

Country Link
KR (1) KR20030065519A (en)
DE (2) DE10131987A1 (en)
DO (1) DOP2001000291A (en)
EC (1) ECSP034616A (en)
GT (1) GT200100235A (en)
HN (1) HN2001000261A (en)
MY (1) MY127212A (en)
PE (1) PE20020581A1 (en)
RU (1) RU2003118584A (en)
SV (1) SV2003000743A (en)
UA (1) UA74404C2 (en)
ZA (1) ZA200303887B (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102485724B (en) * 2010-12-06 2015-08-12 中国人民解放军军事医学科学院毒物药物研究所 Substituted thiophene base pyrazolo-pyridines and medicinal use thereof
CA3040720C (en) 2011-11-25 2021-06-15 Adverio Pharma Gmbh Method for producing substituted 5-fluoro-1h-pyrazolopyridines
EP3525779B1 (en) * 2016-10-11 2024-06-05 Bayer Pharma Aktiengesellschaft Combination containing the sgc stimulator vericuguat and the mineralcorticoid receptor antagonist finerenone

Also Published As

Publication number Publication date
DOP2001000291A (en) 2002-12-15
UA74404C2 (en) 2005-12-15
MY127212A (en) 2006-11-30
DE50106655D1 (en) 2005-08-04
ZA200303887B (en) 2004-06-21
RU2003118584A (en) 2004-12-20
SV2003000743A (en) 2003-01-13
ECSP034616A (en) 2003-06-25
GT200100235A (en) 2002-06-25
PE20020581A1 (en) 2002-07-13
DE10131987A1 (en) 2002-05-23
KR20030065519A (en) 2003-08-06

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