HK47487A - 3-phenoxy-1-azetidinecarboxamides and their use and preparation - Google Patents

3-phenoxy-1-azetidinecarboxamides and their use and preparation

Info

Publication number
HK47487A
HK47487A HK474/87A HK47487A HK47487A HK 47487 A HK47487 A HK 47487A HK 474/87 A HK474/87 A HK 474/87A HK 47487 A HK47487 A HK 47487A HK 47487 A HK47487 A HK 47487A
Authority
HK
Hong Kong
Prior art keywords
phenoxy
trifluoromethyl
azetidine
formula
azetidinecarboxamide
Prior art date
Application number
HK474/87A
Other languages
German (de)
English (en)
French (fr)
Inventor
Lina Chen Teng
Original Assignee
A. H. Robins Company, Incorporated
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by A. H. Robins Company, Incorporated filed Critical A. H. Robins Company, Incorporated
Publication of HK47487A publication Critical patent/HK47487A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/04—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
HK474/87A 1982-08-19 1987-06-18 3-phenoxy-1-azetidinecarboxamides and their use and preparation HK47487A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US40947682A 1982-08-19 1982-08-19

Publications (1)

Publication Number Publication Date
HK47487A true HK47487A (en) 1987-06-26

Family

ID=23620657

Family Applications (1)

Application Number Title Priority Date Filing Date
HK474/87A HK47487A (en) 1982-08-19 1987-06-18 3-phenoxy-1-azetidinecarboxamides and their use and preparation

Country Status (25)

Country Link
EP (1) EP0102194B1 (cs)
JP (1) JPH0643388B2 (cs)
KR (1) KR900001210B1 (cs)
AU (1) AU553528B2 (cs)
CA (1) CA1173841A (cs)
CS (1) CS236796B2 (cs)
DE (1) DE3367089D1 (cs)
DK (1) DK165741C (cs)
EG (1) EG16472A (cs)
ES (1) ES523193A0 (cs)
FI (1) FI77225C (cs)
GR (1) GR79634B (cs)
HK (1) HK47487A (cs)
HU (1) HU190608B (cs)
IE (1) IE55769B1 (cs)
IL (1) IL68699A (cs)
IN (1) IN157045B (cs)
MX (1) MX9203639A (cs)
NO (1) NO157976C (cs)
NZ (1) NZ205317A (cs)
PH (1) PH19595A (cs)
PL (1) PL140765B1 (cs)
PT (1) PT77217B (cs)
YU (1) YU44854B (cs)
ZA (1) ZA834371B (cs)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4594189A (en) * 1983-07-06 1986-06-10 A. H. Robins Company, Inc. Process for preparing 3-phenoxy-1-azetidines and carboxamide derivatives
US5151418A (en) * 1985-02-28 1992-09-29 A. H. Robins Company, Incorporated Method of treating muscular tension, muscle spasticity and anxiety with 3-aryloxy and 3-arylthioazetidinecarboxamides
US4956359A (en) * 1985-02-28 1990-09-11 A. H. Robins Company, Inc. 3-aryloxy and 3-arylthioazetidinecarboxamides as anticonvulsants and antiepileptics
FI87559C (fi) * 1985-02-28 1993-01-25 Robins Co Inc A H Foerfarande foer framstaellning av aktiva 3-fenyloxiazetidinkarboxamider
ZA861210B (en) * 1985-02-28 1987-10-28 Robins Co Inc A H 3-aryloxyazetidinecarboxamides as anticonvulsants and antiepileptics
US5183902A (en) * 1985-02-28 1993-02-02 A. H. Robins Company, Incorporated Method of treating muscular tension, muscle spasticity and anxiety with 3-aryloxy and 3-arylthioazetidinecarboxamides
US5068231A (en) * 1985-02-28 1991-11-26 A. H. Robins Company Incorporated Method of treating muscular tension, muscle spasticity and anxiety with 3-aryloxy and 3-arylthioazetidinecarboxamides
IN162808B (cs) * 1985-02-28 1988-07-09 Robins Co Inc A H
US5183903A (en) * 1991-11-26 1993-02-02 A. H. Robins Company, Incorporated Urea fusion process for the synthesis of 3-phenoxy-1-azetidinecarboxamides
WO1999037612A1 (en) * 1998-01-23 1999-07-29 Vernalis Research Limited Azetidinecarboxamide derivatives for treating cns disorders
ES2181387T3 (es) * 1998-01-23 2003-02-16 Vernalis Res Ltd Derivados de azetidinocarboxamida para el tratamiento de trastornos del sistema nervioso central.
GB9917386D0 (en) * 1999-07-23 1999-09-22 Cerebrus Ltd Chemical compounds-II
CN113754541B (zh) * 2020-06-02 2025-01-03 深圳湾实验室 靶向eb病毒核抗原蛋白的小分子抑制剂、制备方法及其应用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB872447A (en) * 1958-12-23 1961-07-12 Lepetit Spa 1-carbamyl-3-substituted azetidines
US4226861A (en) * 1978-04-18 1980-10-07 A. H. Robins Company, Inc. N-Lower-alkyl 3-phenoxy-1-azetidinecarboxamides

Also Published As

Publication number Publication date
DK376183D0 (da) 1983-08-17
AU553528B2 (en) 1986-07-17
IE55769B1 (en) 1991-01-16
JPH0643388B2 (ja) 1994-06-08
KR900001210B1 (ko) 1990-02-28
ES8500225A1 (es) 1984-10-01
YU158683A (en) 1985-12-31
FI77225C (fi) 1989-02-10
CS236796B2 (en) 1985-05-15
PL243255A1 (en) 1984-08-27
PT77217B (en) 1986-02-04
IL68699A0 (en) 1983-09-30
HU190608B (en) 1986-09-29
PT77217A (en) 1983-09-01
NO157976B (no) 1988-03-14
KR840005715A (ko) 1984-11-15
IE831651L (en) 1984-02-19
DK165741C (da) 1993-06-07
GR79634B (cs) 1984-10-31
IN157045B (cs) 1986-01-04
AU1459783A (en) 1984-02-23
NO832971L (no) 1984-02-20
EP0102194B1 (en) 1986-10-22
CA1173841A (en) 1984-09-04
IL68699A (en) 1986-08-31
NZ205317A (en) 1985-08-30
NO157976C (no) 1988-06-22
MX9203639A (es) 1992-07-01
DK165741B (da) 1993-01-11
DE3367089D1 (en) 1986-11-27
FI77225B (fi) 1988-10-31
PL140765B1 (en) 1987-05-30
PH19595A (en) 1986-05-26
JPS5980657A (ja) 1984-05-10
YU44854B (en) 1991-04-30
ES523193A0 (es) 1984-10-01
FI832956A0 (fi) 1983-08-18
FI832956L (fi) 1984-02-20
EG16472A (en) 1987-03-30
EP0102194A1 (en) 1984-03-07
ZA834371B (en) 1984-03-28
DK376183A (da) 1984-02-20

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Legal Events

Date Code Title Description
PC Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)