HK1252083A1 - Janus激酶(jak)抑制劑的給藥方案 - Google Patents

Janus激酶(jak)抑制劑的給藥方案

Info

Publication number
HK1252083A1
HK1252083A1 HK18110906.2A HK18110906A HK1252083A1 HK 1252083 A1 HK1252083 A1 HK 1252083A1 HK 18110906 A HK18110906 A HK 18110906A HK 1252083 A1 HK1252083 A1 HK 1252083A1
Authority
HK
Hong Kong
Prior art keywords
jak
inhibitors
dosing regimen
janus kinase
janus
Prior art date
Application number
HK18110906.2A
Other languages
English (en)
Inventor
A‧J‧岡薩雷斯
S‧B‧科斯格羅夫
P‧B‧馬爾帕斯
M‧R‧斯特格曼
W‧T‧科勒德
Original Assignee
碩騰服務有限責任公司
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=48901189&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1252083(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by 碩騰服務有限責任公司 filed Critical 碩騰服務有限責任公司
Publication of HK1252083A1 publication Critical patent/HK1252083A1/zh

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/04—Antipruritics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Organic Chemistry (AREA)
  • Immunology (AREA)
  • Dermatology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Plant Substances (AREA)
HK18110906.2A 2012-07-20 2018-08-23 Janus激酶(jak)抑制劑的給藥方案 HK1252083A1 (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261674289P 2012-07-20 2012-07-20
US201361815803P 2013-04-25 2013-04-25

Publications (1)

Publication Number Publication Date
HK1252083A1 true HK1252083A1 (zh) 2019-05-17

Family

ID=48901189

Family Applications (2)

Application Number Title Priority Date Filing Date
HK15109423.1A HK1209314A1 (zh) 2012-07-20 2015-09-24 激酶 抑制劑的給藥方案
HK18110906.2A HK1252083A1 (zh) 2012-07-20 2018-08-23 Janus激酶(jak)抑制劑的給藥方案

Family Applications Before (1)

Application Number Title Priority Date Filing Date
HK15109423.1A HK1209314A1 (zh) 2012-07-20 2015-09-24 激酶 抑制劑的給藥方案

Country Status (24)

Country Link
US (1) US9522151B2 (zh)
EP (1) EP2874630B1 (zh)
JP (2) JP6022063B2 (zh)
KR (2) KR20170034949A (zh)
CN (2) CN108354938A (zh)
AU (1) AU2013292547B2 (zh)
BR (1) BR112015000808A2 (zh)
CA (1) CA2878867C (zh)
CY (1) CY1121436T1 (zh)
DK (1) DK2874630T3 (zh)
ES (1) ES2707627T3 (zh)
HK (2) HK1209314A1 (zh)
HR (1) HRP20182088T1 (zh)
HU (1) HUE042771T2 (zh)
IN (1) IN2015DN00370A (zh)
LT (1) LT2874630T (zh)
MX (1) MX360857B (zh)
NZ (1) NZ703152A (zh)
PL (1) PL2874630T3 (zh)
PT (1) PT2874630T (zh)
RS (1) RS58242B1 (zh)
SI (1) SI2874630T1 (zh)
WO (1) WO2014015107A1 (zh)
ZA (1) ZA201500134B (zh)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HUE037192T2 (hu) 2013-02-22 2018-08-28 Pfizer Pirrolo [2,3-D]pirimidin származékok mint a Janus-kinázok (JAK) inhibitorai
WO2016024185A1 (en) 2014-08-12 2016-02-18 Pfizer Inc. Pyrrolo[2,3-d]pyrimidine derivatives useful for inhibiting janus kinase
SG11201802990RA (en) 2015-10-16 2018-05-30 Abbvie Inc PROCESSES FOR THE PREPARATION OF (3S,4R)-3-ETHYL-4-(3H-IMIDAZO[1,2-a]PYRROLO[2,3-e]-PYRAZIN-8-YL)-N-(2,2,2-TRIFLUOROETHYL)PYRROLIDINE-1-CARBOXAMIDE AND SOLID STATE FORMS THEREOF
US11780848B2 (en) 2015-10-16 2023-10-10 Abbvie Inc. Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-n-(2,2,2-trifluoroethyl)pyrrolidine-1- carboxamide and solid state forms thereof
US10550126B2 (en) 2015-10-16 2020-02-04 Abbvie Inc. Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-A]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof
US11365198B2 (en) 2015-10-16 2022-06-21 Abbvie Inc. Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof
US10973913B2 (en) 2016-02-16 2021-04-13 Washington University JAK inhibitors and uses thereof
CN107098908B (zh) * 2016-02-23 2021-01-08 欣凯医药科技(上海)有限公司 一种吡咯并嘧啶类化合物的制备方法和应用
KR20210120074A (ko) * 2019-01-30 2021-10-06 가르가멜 (주하이) 바이오테크 리미티드 Jak 억제제 및 그 제조 방법
US11992490B2 (en) 2019-10-16 2024-05-28 Incyte Corporation Use of JAK1 inhibitors for the treatment of cutaneous lupus erythematosus and Lichen planus (LP)
WO2022133420A1 (en) 2020-12-18 2022-06-23 Boehringer Ingelheim Animal Health USA Inc. Boron containing pyrazole compounds, compositions comprising them, methods and uses thereof

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RS50087B (sr) * 1998-06-19 2009-01-22 Pfizer Products Inc., Pirolo (2,3-d) pirimidin jedinjenja
ES2467109T3 (es) * 2008-08-20 2014-06-11 Zoetis Llc Compuestos de pirrolo[2,3-d]pirimidina

Also Published As

Publication number Publication date
HK1209314A1 (zh) 2016-04-01
AU2013292547B2 (en) 2017-05-04
JP2017019816A (ja) 2017-01-26
JP6022063B2 (ja) 2016-11-09
AU2013292547A1 (en) 2015-01-22
CA2878867C (en) 2018-01-09
US20150126535A1 (en) 2015-05-07
JP2015522620A (ja) 2015-08-06
CY1121436T1 (el) 2020-05-29
PT2874630T (pt) 2019-01-31
MX2015000871A (es) 2015-05-07
PL2874630T3 (pl) 2019-04-30
BR112015000808A2 (pt) 2017-06-27
IN2015DN00370A (zh) 2015-06-12
WO2014015107A1 (en) 2014-01-23
EP2874630B1 (en) 2018-12-05
US9522151B2 (en) 2016-12-20
SI2874630T1 (sl) 2019-04-30
CN104470525A (zh) 2015-03-25
CA2878867A1 (en) 2014-01-23
MX360857B (es) 2018-11-20
KR20170034949A (ko) 2017-03-29
NZ703152A (en) 2016-03-31
EP2874630A1 (en) 2015-05-27
CN108354938A (zh) 2018-08-03
RS58242B1 (sr) 2019-03-29
LT2874630T (lt) 2019-02-11
ES2707627T3 (es) 2019-04-04
HRP20182088T1 (hr) 2019-02-08
HUE042771T2 (hu) 2019-07-29
DK2874630T3 (en) 2019-01-28
KR20150028299A (ko) 2015-03-13
ZA201500134B (en) 2016-08-31

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