HK1206012A1 - Pyrazol-1-yl benzene sulfonamides as ccr9 antagonists ccr9 -1- - Google Patents

Pyrazol-1-yl benzene sulfonamides as ccr9 antagonists ccr9 -1-

Info

Publication number
HK1206012A1
HK1206012A1 HK15106465.6A HK15106465A HK1206012A1 HK 1206012 A1 HK1206012 A1 HK 1206012A1 HK 15106465 A HK15106465 A HK 15106465A HK 1206012 A1 HK1206012 A1 HK 1206012A1
Authority
HK
Hong Kong
Prior art keywords
ccr9
pyrazol
antagonists
benzene sulfonamides
sulfonamides
Prior art date
Application number
HK15106465.6A
Other languages
English (en)
Chinese (zh)
Inventor
Xi Chen
Junfa Fan
Pingchen Fan
Antoni Krasinski
Lianfa Li
Rebecca M Lui
Jeffrey P Mcmahon
Jay P Powers
Yibin Zeng
Penglie Zhang
Original Assignee
Chemocentryx Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chemocentryx Inc filed Critical Chemocentryx Inc
Publication of HK1206012A1 publication Critical patent/HK1206012A1/xx

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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/472—Non-condensed isoquinolines, e.g. papaverine
    • A61K31/4725—Non-condensed isoquinolines, e.g. papaverine containing further heterocyclic rings
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
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HK15106465.6A 2012-02-29 2015-07-07 Pyrazol-1-yl benzene sulfonamides as ccr9 antagonists ccr9 -1- HK1206012A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261604998P 2012-02-29 2012-02-29
PCT/US2013/028328 WO2013130811A1 (en) 2012-02-29 2013-02-28 Pyrazol-1-yl benzene sulfonamides as ccr9 antagonists

Publications (1)

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HK1206012A1 true HK1206012A1 (en) 2015-12-31

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Application Number Title Priority Date Filing Date
HK15106465.6A HK1206012A1 (en) 2012-02-29 2015-07-07 Pyrazol-1-yl benzene sulfonamides as ccr9 antagonists ccr9 -1-
HK15109875.4A HK1209119A1 (en) 2012-02-29 2015-10-09 Pyrazol-1-yl benzene sulfonamides as ccr9 antagonists ccr9 -1-
HK18105070.2A HK1245773A1 (zh) 2012-02-29 2018-04-19 作為ccr9拮抗劑的吡唑-1-基苯磺酰胺

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HK15109875.4A HK1209119A1 (en) 2012-02-29 2015-10-09 Pyrazol-1-yl benzene sulfonamides as ccr9 antagonists ccr9 -1-
HK18105070.2A HK1245773A1 (zh) 2012-02-29 2018-04-19 作為ccr9拮抗劑的吡唑-1-基苯磺酰胺

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US (5) US8916601B2 (ru)
EP (3) EP2820006B1 (ru)
JP (3) JP6249966B2 (ru)
KR (1) KR102083693B1 (ru)
CN (2) CN107266425B (ru)
AU (3) AU2013225938B2 (ru)
BR (1) BR112014021148B1 (ru)
CA (1) CA2865714C (ru)
DK (2) DK3263564T3 (ru)
ES (2) ES2645617T3 (ru)
HK (3) HK1206012A1 (ru)
MX (1) MX2014010340A (ru)
PL (2) PL2820006T3 (ru)
PT (1) PT3263564T (ru)
RU (1) RU2627268C2 (ru)
SG (2) SG11201405241VA (ru)
WO (1) WO2013130811A1 (ru)
ZA (1) ZA201406432B (ru)

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US9100454B2 (en) 2006-04-07 2015-08-04 Groupon, Inc. Method and system for enabling the creation and maintenance of proximity-related user groups
US10827315B2 (en) * 2006-04-07 2020-11-03 Groupon, Inc. Facilitating user interactions based on proximity
CN107266425B (zh) * 2012-02-29 2020-03-03 坎莫森特里克斯公司 作为ccr9拮抗剂的吡唑-1-基苯磺酰胺
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