HK1245773A1 - 作為ccr9拮抗劑的吡唑-1-基苯磺酰胺 - Google Patents

作為ccr9拮抗劑的吡唑-1-基苯磺酰胺

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Publication number
HK1245773A1
HK1245773A1 HK18105070.2A HK18105070A HK1245773A1 HK 1245773 A1 HK1245773 A1 HK 1245773A1 HK 18105070 A HK18105070 A HK 18105070A HK 1245773 A1 HK1245773 A1 HK 1245773A1
Authority
HK
Hong Kong
Prior art keywords
pyrazol
benzene sulfonamides
ccr9 antagonists
ccr9
antagonists
Prior art date
Application number
HK18105070.2A
Other languages
English (en)
Inventor
Xi Chen
Junfa Fan
Pingchen Fan
Antoni Krasinski
Lianfa Li
Rebecca M Lui
Jeffrey P Mcmahon
Jay P Powers
Yibin Zeng
Penglie Zhang
Original Assignee
Chemocentryx Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chemocentryx Inc filed Critical Chemocentryx Inc
Publication of HK1245773A1 publication Critical patent/HK1245773A1/zh

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
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    • A61K31/47—Quinolines; Isoquinolines
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    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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  • Health & Medical Sciences (AREA)
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  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
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  • Physical Education & Sports Medicine (AREA)
  • Diabetes (AREA)
  • Dermatology (AREA)
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HK18105070.2A 2012-02-29 2018-04-19 作為ccr9拮抗劑的吡唑-1-基苯磺酰胺 HK1245773A1 (zh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201261604998P 2012-02-29 2012-02-29

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HK1245773A1 true HK1245773A1 (zh) 2018-08-31

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HK15106465.6A HK1206012A1 (zh) 2012-02-29 2015-07-07 作為 拮抗劑的吡唑- -基苯磺酰胺類
HK15109875.4A HK1209119A1 (zh) 2012-02-29 2015-10-09 作為 拮抗劑的吡唑- -基苯磺酰胺
HK18105070.2A HK1245773A1 (zh) 2012-02-29 2018-04-19 作為ccr9拮抗劑的吡唑-1-基苯磺酰胺

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HK15106465.6A HK1206012A1 (zh) 2012-02-29 2015-07-07 作為 拮抗劑的吡唑- -基苯磺酰胺類
HK15109875.4A HK1209119A1 (zh) 2012-02-29 2015-10-09 作為 拮抗劑的吡唑- -基苯磺酰胺

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US (5) US8916601B2 (zh)
EP (3) EP3738958A1 (zh)
JP (3) JP6249966B2 (zh)
KR (1) KR102083693B1 (zh)
CN (2) CN104520288B (zh)
AU (3) AU2013225938B2 (zh)
BR (1) BR112014021148B1 (zh)
CA (1) CA2865714C (zh)
DK (2) DK3263564T3 (zh)
ES (2) ES2816060T3 (zh)
HK (3) HK1206012A1 (zh)
MX (1) MX2014010340A (zh)
PL (2) PL3263564T3 (zh)
PT (1) PT3263564T (zh)
RU (1) RU2627268C2 (zh)
SG (2) SG11201405241VA (zh)
WO (1) WO2013130811A1 (zh)
ZA (1) ZA201406432B (zh)

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US9100454B2 (en) 2006-04-07 2015-08-04 Groupon, Inc. Method and system for enabling the creation and maintenance of proximity-related user groups
US10827315B2 (en) * 2006-04-07 2020-11-03 Groupon, Inc. Facilitating user interactions based on proximity
DK3263564T3 (da) 2012-02-29 2020-09-07 Chemocentryx Inc Aza-aryl-1h-pyrazol-1-yl-benzen-sulfonamider som ccr(9)- antagonister
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