HK1206012A1 - Pyrazol-1-yl benzene sulfonamides as ccr9 antagonists ccr9 -1- - Google Patents
Pyrazol-1-yl benzene sulfonamides as ccr9 antagonists ccr9 -1-Info
- Publication number
- HK1206012A1 HK1206012A1 HK15106465.6A HK15106465A HK1206012A1 HK 1206012 A1 HK1206012 A1 HK 1206012A1 HK 15106465 A HK15106465 A HK 15106465A HK 1206012 A1 HK1206012 A1 HK 1206012A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- ccr9
- pyrazol
- antagonists
- benzene sulfonamides
- sulfonamides
- Prior art date
Links
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
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- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/472—Non-condensed isoquinolines, e.g. papaverine
- A61K31/4725—Non-condensed isoquinolines, e.g. papaverine containing further heterocyclic rings
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- A61K31/50—Pyridazines; Hydrogenated pyridazines
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- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
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- C07D231/42—Benzene-sulfonamido pyrazoles
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- C—CHEMISTRY; METALLURGY
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- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
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- Dermatology (AREA)
- Diabetes (AREA)
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- Communicable Diseases (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Endocrinology (AREA)
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- Neurology (AREA)
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- AIDS & HIV (AREA)
- Hospice & Palliative Care (AREA)
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Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201261604998P | 2012-02-29 | 2012-02-29 | |
PCT/US2013/028328 WO2013130811A1 (en) | 2012-02-29 | 2013-02-28 | Pyrazol-1-yl benzene sulfonamides as ccr9 antagonists |
Publications (1)
Publication Number | Publication Date |
---|---|
HK1206012A1 true HK1206012A1 (en) | 2015-12-31 |
Family
ID=47844528
Family Applications (3)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HK15106465.6A HK1206012A1 (en) | 2012-02-29 | 2015-07-07 | Pyrazol-1-yl benzene sulfonamides as ccr9 antagonists ccr9 -1- |
HK15109875.4A HK1209119A1 (en) | 2012-02-29 | 2015-10-09 | Pyrazol-1-yl benzene sulfonamides as ccr9 antagonists ccr9 -1- |
HK18105070.2A HK1245773A1 (zh) | 2012-02-29 | 2018-04-19 | 作為ccr9拮抗劑的吡唑-1-基苯磺酰胺 |
Family Applications After (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HK15109875.4A HK1209119A1 (en) | 2012-02-29 | 2015-10-09 | Pyrazol-1-yl benzene sulfonamides as ccr9 antagonists ccr9 -1- |
HK18105070.2A HK1245773A1 (zh) | 2012-02-29 | 2018-04-19 | 作為ccr9拮抗劑的吡唑-1-基苯磺酰胺 |
Country Status (18)
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US (5) | US8916601B2 (xx) |
EP (3) | EP2820006B1 (xx) |
JP (3) | JP6249966B2 (xx) |
KR (1) | KR102083693B1 (xx) |
CN (2) | CN107266425B (xx) |
AU (3) | AU2013225938B2 (xx) |
BR (1) | BR112014021148B1 (xx) |
CA (1) | CA2865714C (xx) |
DK (2) | DK2820006T3 (xx) |
ES (2) | ES2816060T3 (xx) |
HK (3) | HK1206012A1 (xx) |
MX (1) | MX2014010340A (xx) |
PL (2) | PL3263564T3 (xx) |
PT (1) | PT3263564T (xx) |
RU (1) | RU2627268C2 (xx) |
SG (2) | SG10201700493XA (xx) |
WO (1) | WO2013130811A1 (xx) |
ZA (1) | ZA201406432B (xx) |
Families Citing this family (19)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US10827315B2 (en) * | 2006-04-07 | 2020-11-03 | Groupon, Inc. | Facilitating user interactions based on proximity |
US9100454B2 (en) | 2006-04-07 | 2015-08-04 | Groupon, Inc. | Method and system for enabling the creation and maintenance of proximity-related user groups |
SG10201700493XA (en) | 2012-02-29 | 2017-03-30 | Chemocentryx Inc | Pyrazol-1-yl benzene sulfonamides as ccr9 antagonists |
WO2014088113A1 (en) | 2012-12-04 | 2014-06-12 | Millennium Pharmaceuticals, Inc. | Prophylactic or therapeutic method for sjogren's syndrome using specific ccr9 receptor inhibitors/antagonists |
GB201308978D0 (en) | 2013-05-17 | 2013-07-03 | Imp Innovations Ltd | Method for producing polymers and block copolymers |
JP6563947B2 (ja) * | 2013-12-02 | 2019-08-21 | ケモセントリックス,インコーポレイティド | Ccr6化合物 |
WO2015097121A1 (en) * | 2013-12-23 | 2015-07-02 | Norgine B.V. | Compounds useful as ccr9 modulators |
NZ729878A (en) | 2014-10-06 | 2024-03-22 | Chemocentryx Inc | Combination therapy of inhibitors of c-c chemokine receptor type 9 (ccr9) and anti-alpha4beta7 integrin blocking antibodies |
GB201515350D0 (en) | 2015-08-28 | 2015-10-14 | Econic Technologies Ltd | Method for preparing polyols |
RU2743747C2 (ru) * | 2016-01-20 | 2021-02-25 | Кемосентрикс, Инк. | 2-оксиндольные соединения |
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