HK1198587A1 - 異噻唑並吡啶- -甲酰胺和它們作為藥物的用途 - Google Patents
異噻唑並吡啶- -甲酰胺和它們作為藥物的用途Info
- Publication number
- HK1198587A1 HK1198587A1 HK14112083A HK14112083A HK1198587A1 HK 1198587 A1 HK1198587 A1 HK 1198587A1 HK 14112083 A HK14112083 A HK 14112083A HK 14112083 A HK14112083 A HK 14112083A HK 1198587 A1 HK1198587 A1 HK 1198587A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- isothiazolopyridine
- carboxamides
- pharmaceuticals
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H13/00—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids
- C07H13/02—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids by carboxylic acids
- C07H13/04—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids by carboxylic acids having the esterifying carboxyl radicals attached to acyclic carbon atoms
- C07H13/06—Fatty acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H13/00—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids
- C07H13/12—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids by acids having the group -X-C(=X)-X-, or halides thereof, in which each X means nitrogen, oxygen, sulfur, selenium or tellurium, e.g. carbonic acid, carbamic acid
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Physical Education & Sports Medicine (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Psychology (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Gastroenterology & Hepatology (AREA)
- Hospice & Palliative Care (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Immunology (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyridine Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Saccharide Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP11306711 | 2011-12-20 | ||
PCT/EP2012/075932 WO2013092574A1 (en) | 2011-12-20 | 2012-12-18 | Isothiazolopyridine-2-carboxamides and their use as pharmaceuticals |
Publications (1)
Publication Number | Publication Date |
---|---|
HK1198587A1 true HK1198587A1 (zh) | 2015-04-30 |
Family
ID=47429823
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HK14112083A HK1198587A1 (zh) | 2011-12-20 | 2014-12-01 | 異噻唑並吡啶- -甲酰胺和它們作為藥物的用途 |
Country Status (24)
Country | Link |
---|---|
US (1) | US9260454B2 (zh) |
EP (1) | EP2794618B1 (zh) |
JP (1) | JP6099669B2 (zh) |
KR (1) | KR20140103150A (zh) |
CN (1) | CN104136443B (zh) |
AR (1) | AR089329A1 (zh) |
AU (1) | AU2012357864B2 (zh) |
BR (1) | BR112014015033A2 (zh) |
CA (1) | CA2856964A1 (zh) |
CY (1) | CY1118854T1 (zh) |
DK (1) | DK2794618T3 (zh) |
ES (1) | ES2613826T3 (zh) |
HK (1) | HK1198587A1 (zh) |
HR (1) | HRP20170159T1 (zh) |
HU (1) | HUE033049T2 (zh) |
IL (1) | IL232809A (zh) |
LT (1) | LT2794618T (zh) |
MX (1) | MX2014007465A (zh) |
PL (1) | PL2794618T3 (zh) |
PT (1) | PT2794618T (zh) |
RU (1) | RU2014129903A (zh) |
SG (1) | SG11201402623RA (zh) |
SI (1) | SI2794618T1 (zh) |
WO (1) | WO2013092574A1 (zh) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP6814730B2 (ja) * | 2014-09-05 | 2021-01-20 | ジェネンテック, インコーポレイテッド | 治療用化合物およびその使用 |
WO2017030892A1 (en) * | 2015-08-14 | 2017-02-23 | Reaction Biology Corp. | Histone deacetylase inhibitors and methods for use thereof |
Family Cites Families (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3892745A (en) * | 1972-11-20 | 1975-07-01 | Sankyo Co | Isoxazolone derivatives and process for preparing the same |
US3965107A (en) | 1974-07-08 | 1976-06-22 | Rohm And Haas Company | Isothiazolopyridinones |
LU84091A1 (fr) * | 1982-04-16 | 1984-03-02 | Oreal | Derives n-carbamoyl d'isothiazolo-(5,4b)pyridine one-3,leur procede de preparation et leurs utilisations comme agents bactericides et fongicides |
US4968713A (en) | 1989-07-31 | 1990-11-06 | Merck & Co., Inc. | Certain imidazole compounds as transglutaminase inhibitors |
DE10054687A1 (de) | 2000-11-03 | 2002-05-16 | N Zyme Biotec Gmbh | Inhibitoren von Transglutaminasen |
EP1613608A1 (en) * | 2003-04-01 | 2006-01-11 | Eli Lilly And Company | Phospholipase inhibitors |
EP1615900A1 (en) * | 2003-04-01 | 2006-01-18 | Eli Lilly And Company | Benzisothiazol-3-one-carboxylic acid amides as phospholipase inhibitors |
GB0314262D0 (en) | 2003-06-19 | 2003-07-23 | Univ Nottingham Trent | Novel compounds and methods of using the same |
JP2007529468A (ja) * | 2004-03-16 | 2007-10-25 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | ベンズイソオキサゾール |
DE102006014688A1 (de) | 2006-03-28 | 2007-10-04 | Sanofi-Aventis | Azolopyridin-3-on-derivate als Inhibitoren von Lipasen und Phospholipasen |
DE102006052755A1 (de) | 2006-11-08 | 2008-05-15 | N-Zyme Biotec Gmbh | Michaelsysteme als Transglutaminaseinhibitoren |
WO2011060321A1 (en) | 2009-11-16 | 2011-05-19 | Chdi, Inc. | Transglutaminase tg2 inhibitors, pharmaceutical compositions, and methods of use thereof |
WO2011157827A1 (de) * | 2010-06-18 | 2011-12-22 | Sanofi | Azolopyridin-3-on-derivate als inhibitoren von lipasen und phospholipasen |
-
2012
- 2012-12-18 PT PT128060431T patent/PT2794618T/pt unknown
- 2012-12-18 EP EP12806043.1A patent/EP2794618B1/en active Active
- 2012-12-18 RU RU2014129903A patent/RU2014129903A/ru not_active Application Discontinuation
- 2012-12-18 HU HUE12806043A patent/HUE033049T2/hu unknown
- 2012-12-18 BR BR112014015033A patent/BR112014015033A2/pt not_active IP Right Cessation
- 2012-12-18 LT LTEP12806043.1T patent/LT2794618T/lt unknown
- 2012-12-18 MX MX2014007465A patent/MX2014007465A/es unknown
- 2012-12-18 JP JP2014547921A patent/JP6099669B2/ja not_active Expired - Fee Related
- 2012-12-18 ES ES12806043.1T patent/ES2613826T3/es active Active
- 2012-12-18 DK DK12806043.1T patent/DK2794618T3/en active
- 2012-12-18 SI SI201230855A patent/SI2794618T1/sl unknown
- 2012-12-18 PL PL12806043T patent/PL2794618T3/pl unknown
- 2012-12-18 WO PCT/EP2012/075932 patent/WO2013092574A1/en active Application Filing
- 2012-12-18 CA CA2856964A patent/CA2856964A1/en not_active Abandoned
- 2012-12-18 SG SG11201402623RA patent/SG11201402623RA/en unknown
- 2012-12-18 KR KR1020147019341A patent/KR20140103150A/ko not_active Application Discontinuation
- 2012-12-18 CN CN201280070206.0A patent/CN104136443B/zh not_active Expired - Fee Related
- 2012-12-18 AU AU2012357864A patent/AU2012357864B2/en not_active Ceased
- 2012-12-19 AR ARP120104822A patent/AR089329A1/es unknown
-
2014
- 2014-05-26 IL IL232809A patent/IL232809A/en not_active IP Right Cessation
- 2014-06-18 US US14/307,961 patent/US9260454B2/en active Active
- 2014-12-01 HK HK14112083A patent/HK1198587A1/zh not_active IP Right Cessation
-
2017
- 2017-02-01 HR HRP20170159TT patent/HRP20170159T1/hr unknown
- 2017-02-15 CY CY20171100208T patent/CY1118854T1/el unknown
Also Published As
Publication number | Publication date |
---|---|
CN104136443B (zh) | 2017-01-18 |
IL232809A0 (en) | 2014-08-03 |
US9260454B2 (en) | 2016-02-16 |
AU2012357864A1 (en) | 2014-07-03 |
CN104136443A (zh) | 2014-11-05 |
CA2856964A1 (en) | 2013-06-27 |
DK2794618T3 (en) | 2017-02-20 |
BR112014015033A2 (pt) | 2017-06-13 |
AR089329A1 (es) | 2014-08-13 |
PT2794618T (pt) | 2017-01-17 |
CY1118854T1 (el) | 2018-01-10 |
IL232809A (en) | 2017-05-29 |
SG11201402623RA (en) | 2014-09-26 |
LT2794618T (lt) | 2017-02-27 |
JP6099669B2 (ja) | 2017-03-22 |
JP2015500855A (ja) | 2015-01-08 |
EP2794618B1 (en) | 2016-11-16 |
EP2794618A1 (en) | 2014-10-29 |
US20140296169A1 (en) | 2014-10-02 |
HUE033049T2 (hu) | 2017-11-28 |
KR20140103150A (ko) | 2014-08-25 |
MX2014007465A (es) | 2014-07-30 |
AU2012357864B2 (en) | 2017-03-02 |
PL2794618T3 (pl) | 2017-05-31 |
WO2013092574A1 (en) | 2013-06-27 |
RU2014129903A (ru) | 2016-02-10 |
SI2794618T1 (sl) | 2017-03-31 |
HRP20170159T1 (hr) | 2017-03-24 |
ES2613826T3 (es) | 2017-05-26 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
HUS2100012I1 (hu) | 4-Imidazopiridazin-1-il-benzamidok és 4-imidazotriazin-1-il-benzamidok mint BTK-gátlók | |
IL233051B (en) | Anti-phf-tau antibodies and uses thereof | |
HK1198433A1 (zh) | -酰基二肽衍生物及其應用 | |
GB201111705D0 (en) | Compounds and their use | |
IL229844B (en) | Anti-psgl-1 antibodies and their use | |
HK1191034A1 (zh) | -羧烷基耳他汀類及其應用 | |
GB201110783D0 (en) | Methods and uses | |
IL231082A0 (en) | Pyrimido-pyridazinone compounds and their use | |
EP2688588A4 (en) | FAST AND LONG-TERM IMMUNOLOGICAL THERAPEUTIC | |
GB201111630D0 (en) | Novel compounds and their use | |
GB201116774D0 (en) | Uses and methods | |
EP2697386A4 (en) | DESIGN AND USE OF PEPDUCINE | |
EP2716359A4 (en) | COMPLEX AND USES THEREOF | |
GB201111775D0 (en) | Compounds and uses thereof | |
GB201114448D0 (en) | Compounds and their use | |
EP2668044A4 (en) | COMPOSITIONS AND THEIR USE | |
GB201106357D0 (en) | Composition and uses thereof | |
EP2693879A4 (en) | MIGRASTATINES AND THEIR USES | |
HK1198587A1 (zh) | 異噻唑並吡啶- -甲酰胺和它們作為藥物的用途 | |
GB201108490D0 (en) | Methods and uses | |
PT2734522T (pt) | 4-imidazopiridazina-1-il-benzamidas e 4-imidazotriazin-1- il-benzamidas como inibidores de btk | |
GB201104444D0 (en) | Compounds and their use | |
GB201121551D0 (en) | Compounds and uses thereof |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
PC | Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee) |
Effective date: 20201220 |