HK1185878A1 - 用於治療或預防由血清素、去甲腎上腺素或多巴胺的神經傳遞的減少而引起的疾病的雜環化合物 - Google Patents
用於治療或預防由血清素、去甲腎上腺素或多巴胺的神經傳遞的減少而引起的疾病的雜環化合物Info
- Publication number
- HK1185878A1 HK1185878A1 HK13113304.9A HK13113304A HK1185878A1 HK 1185878 A1 HK1185878 A1 HK 1185878A1 HK 13113304 A HK13113304 A HK 13113304A HK 1185878 A1 HK1185878 A1 HK 1185878A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- norephnephrine
- serotonin
- dopamine
- treating
- heterocyclic compounds
- Prior art date
Links
- VYFYYTLLBUKUHU-UHFFFAOYSA-N dopamine Chemical compound NCCC1=CC=C(O)C(O)=C1 VYFYYTLLBUKUHU-UHFFFAOYSA-N 0.000 title 2
- QZAYGJVTTNCVMB-UHFFFAOYSA-N serotonin Chemical compound C1=C(O)C=C2C(CCN)=CNC2=C1 QZAYGJVTTNCVMB-UHFFFAOYSA-N 0.000 title 2
- 229960003638 dopamine Drugs 0.000 title 1
- 150000002391 heterocyclic compounds Chemical class 0.000 title 1
- 229940076279 serotonin Drugs 0.000 title 1
- 230000005062 synaptic transmission Effects 0.000 title 1
Classifications
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PCT/JP2011/071174 WO2012036253A1 (en) | 2010-09-13 | 2011-09-12 | Heterocyclic compounds for treating or preventing disorders caused by reduced neurotransmission of serotonin, norephnephrine or dopamine. |
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JP6415982B2 (ja) * | 2012-03-12 | 2018-10-31 | 大塚製薬株式会社 | 複素環化合物 |
MX2014013489A (es) | 2012-05-09 | 2015-02-12 | Bayer Cropscience Ag | 5-halogenopirazolindanil carboxamidas. |
US20160287589A1 (en) | 2013-02-20 | 2016-10-06 | Bayer Pharma Aktiengesellschaft | Substituted-imidazopyridazines |
WO2019076358A1 (en) | 2017-10-19 | 2019-04-25 | Js Innopharm (Shanghai) Ltd | HETEROCYCLIC COMPOUNDS, COMPOSITIONS COMPRISING THE HETEROCYCLIC COMPOUND, AND METHODS OF USE THEREOF |
WO2023286768A1 (en) * | 2021-07-13 | 2023-01-19 | Otsuka Pharmaceutical Co., Ltd. | Hydrogenated quinoxalines |
CN116554127A (zh) * | 2022-01-28 | 2023-08-08 | 成都麻沸散医药科技有限公司 | 哌嗪取代苯酚类衍生物及其用途 |
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SU390391A1 (ru) | 1971-04-12 | 1973-07-11 | УСТРОЙСТВО дл ИЗМЕРЕНИЯ ДАВЛЕНИЯ | |
SU390091A1 (ru) * | 1971-07-12 | 1973-07-11 | С. И. Бурмистров, Н. В. Макаревич , Л. Я. Кравченко Днепропетровский химико технологический институт Дзержинского | Способ получения 1-аренсульфонил-4- -арилдекагидрохиноксалинов |
DE4210941A1 (de) | 1992-04-02 | 1993-10-07 | Bayer Ag | Neue 9-Fluor-7.oxo-7H-pyrido[1,2,3-d,e][1,4]benzoxacin-6-carbonsäuren und -ester |
DE4337609A1 (de) * | 1993-11-04 | 1995-05-11 | Boehringer Ingelheim Kg | Neue Pyrazincarboxamidderivate, ihre Herstellung und ihre Verwendung in Arzneimitteln |
AU1303897A (en) | 1996-01-05 | 1997-08-01 | Ciba-Geigy Ag | Herbicidal 1,2,4,6-thiatriazines |
DE69919436T2 (de) * | 1998-04-16 | 2005-09-15 | Pfizer Products Inc., Groton | N-Acyl und N-Aroyl Aralkylamide |
IT1312310B1 (it) * | 1999-05-07 | 2002-04-15 | Recordati Ind Chimica E Farma | Uso di antagonisti selettivi del recettore adrenergico a 1b per ilmiglioramento della disfunzione sessuale |
PE20040804A1 (es) * | 2002-12-19 | 2004-12-31 | Boehringer Ingelheim Pharma | DERIVADOS DE CARBOXAMIDAS COMO INHIBIDORES DEL FACTOR Xa |
JP5512268B2 (ja) * | 2006-08-07 | 2014-06-04 | アルバニー モルキュラー リサーチ,インコーポレイテッド | 5ht3モジュレーターとしての2−アミノベンゾオキサゾールカルボキサミド |
EP2057141B1 (en) * | 2006-08-23 | 2011-10-26 | Pfizer Products Inc. | Pyrimidone compounds as gsk-3 inhibitors |
UA108596C2 (xx) * | 2007-11-09 | 2015-05-25 | Інгібітори пептиддеформілази | |
TWM369750U (en) | 2009-06-03 | 2009-12-01 | Yu-Hao Shen | Self-rotation mop structure |
WO2010141540A1 (en) * | 2009-06-03 | 2010-12-09 | Glaxosmithkline Llc | Bis-pyridylpyridones as melanin-concentrating hormone receptor 1 antagonists |
WO2011068171A1 (ja) * | 2009-12-03 | 2011-06-09 | 第一三共株式会社 | 二環性含窒素飽和へテロ環誘導体 |
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