HK1176548A1 - Pharmaceutical for oral delivery comprising mgbg and methods of treating disease mgbg - Google Patents

Pharmaceutical for oral delivery comprising mgbg and methods of treating disease mgbg

Info

Publication number
HK1176548A1
HK1176548A1 HK13103363.8A HK13103363A HK1176548A1 HK 1176548 A1 HK1176548 A1 HK 1176548A1 HK 13103363 A HK13103363 A HK 13103363A HK 1176548 A1 HK1176548 A1 HK 1176548A1
Authority
HK
Hong Kong
Prior art keywords
mgbg
pharmaceutical
methods
oral delivery
treating disease
Prior art date
Application number
HK13103363.8A
Other languages
English (en)
Chinese (zh)
Inventor
.麥基爾恩
.布利策
Original Assignee
帕薩羅杰卡有限公司
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 帕薩羅杰卡有限公司 filed Critical 帕薩羅杰卡有限公司
Publication of HK1176548A1 publication Critical patent/HK1176548A1/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/155Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0002Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2031Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4858Organic compounds
    • AHUMAN NECESSITIES
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    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
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    • A61K9/4866Organic macromolecular compounds
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    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
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    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
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    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
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    • A61P9/12Antihypertensives

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Virology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Immunology (AREA)
  • Molecular Biology (AREA)
  • Oncology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Communicable Diseases (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Biophysics (AREA)
  • Dermatology (AREA)
  • Obesity (AREA)
  • Psychiatry (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Biotechnology (AREA)
  • Urology & Nephrology (AREA)
  • Hematology (AREA)
  • Pulmonology (AREA)
  • Endocrinology (AREA)
HK13103363.8A 2009-07-16 2013-03-18 Pharmaceutical for oral delivery comprising mgbg and methods of treating disease mgbg HK1176548A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US22606009P 2009-07-16 2009-07-16
US29009509P 2009-12-24 2009-12-24
PCT/US2010/042253 WO2011009039A2 (en) 2009-07-16 2010-07-16 Pharmaceutical for oral delivery comprising mgbg and methods of treating disease

Publications (1)

Publication Number Publication Date
HK1176548A1 true HK1176548A1 (en) 2013-08-02

Family

ID=43450234

Family Applications (1)

Application Number Title Priority Date Filing Date
HK13103363.8A HK1176548A1 (en) 2009-07-16 2013-03-18 Pharmaceutical for oral delivery comprising mgbg and methods of treating disease mgbg

Country Status (12)

Country Link
US (4) US8258186B2 (ja)
EP (2) EP3473247A1 (ja)
JP (4) JP6112449B2 (ja)
CN (2) CN104997762B (ja)
AU (2) AU2010273277B2 (ja)
BR (1) BR112012000862A8 (ja)
CA (1) CA2768018C (ja)
DK (1) DK2453886T3 (ja)
ES (1) ES2715173T3 (ja)
HK (1) HK1176548A1 (ja)
NZ (3) NZ628513A (ja)
WO (1) WO2011009039A2 (ja)

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WO2011009039A2 (en) 2011-01-20
AU2010273277A1 (en) 2012-02-02
JP2012533565A (ja) 2012-12-27
US8258186B2 (en) 2012-09-04
EP2453886A4 (en) 2012-12-05
CN104997762A (zh) 2015-10-28
BR112012000862A8 (pt) 2018-01-09
DK2453886T3 (en) 2019-03-25
EP3473247A1 (en) 2019-04-24
EP2453886B1 (en) 2018-12-12
JP2016065045A (ja) 2016-04-28
CN104997762B (zh) 2019-03-08
AU2016266049A1 (en) 2016-12-22
JP2020063258A (ja) 2020-04-23
CN102686222A (zh) 2012-09-19
US20140051765A1 (en) 2014-02-20
NZ715686A (en) 2017-08-25
US8609734B2 (en) 2013-12-17
CA2768018C (en) 2019-08-27
WO2011009039A3 (en) 2011-06-16
US20170290788A1 (en) 2017-10-12
NZ628513A (en) 2016-01-29
ES2715173T3 (es) 2019-06-03
CA2768018A1 (en) 2011-01-20
US20110112199A1 (en) 2011-05-12
NZ597488A (en) 2014-10-31
CN102686222B (zh) 2015-06-24
US9616035B2 (en) 2017-04-11
US20120289604A1 (en) 2012-11-15
BR112012000862A2 (pt) 2017-10-31
JP6883930B2 (ja) 2021-06-09
AU2016266049B2 (en) 2018-10-18
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JP2018127460A (ja) 2018-08-16

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