HK1109151A1 - Aspartyl protease inhibitors - Google Patents

Aspartyl protease inhibitors

Info

Publication number
HK1109151A1
HK1109151A1 HK08103079.0A HK08103079A HK1109151A1 HK 1109151 A1 HK1109151 A1 HK 1109151A1 HK 08103079 A HK08103079 A HK 08103079A HK 1109151 A1 HK1109151 A1 HK 1109151A1
Authority
HK
Hong Kong
Prior art keywords
protease inhibitors
aspartyl protease
aspartyl
inhibitors
protease
Prior art date
Application number
HK08103079.0A
Other languages
English (en)
Inventor
Zhaoning Zhu
Brian Mckittrick
Andrew W Stamford
Ying Huang
Elizabeth M Smith
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corp filed Critical Schering Corp
Publication of HK1109151A1 publication Critical patent/HK1109151A1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Epidemiology (AREA)
  • Virology (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Molecular Biology (AREA)
  • AIDS & HIV (AREA)
  • Oncology (AREA)
  • Cardiology (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
HK08103079.0A 2005-06-14 2008-03-18 Aspartyl protease inhibitors HK1109151A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US69032605P 2005-06-14 2005-06-14
PCT/US2006/022698 WO2006138192A1 (en) 2005-06-14 2006-06-12 Aspartyl protease inhibitors

Publications (1)

Publication Number Publication Date
HK1109151A1 true HK1109151A1 (en) 2008-05-30

Family

ID=37074234

Family Applications (1)

Application Number Title Priority Date Filing Date
HK08103079.0A HK1109151A1 (en) 2005-06-14 2008-03-18 Aspartyl protease inhibitors

Country Status (18)

Country Link
US (1) US7759354B2 (ko)
EP (1) EP1896477B1 (ko)
JP (1) JP2008543840A (ko)
KR (1) KR20080031189A (ko)
CN (1) CN101198609A (ko)
AR (1) AR054620A1 (ko)
AT (1) ATE482214T1 (ko)
AU (1) AU2006259675A1 (ko)
CA (1) CA2610812A1 (ko)
DE (1) DE602006017073D1 (ko)
ES (1) ES2350854T3 (ko)
HK (1) HK1109151A1 (ko)
IL (1) IL187623A0 (ko)
MX (1) MX2007016175A (ko)
PE (1) PE20070018A1 (ko)
TW (1) TW200716644A (ko)
WO (1) WO2006138192A1 (ko)
ZA (1) ZA200710337B (ko)

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CN104270945B (zh) 2012-03-19 2017-03-29 巴克老龄化研究所 App特异性bace抑制剂(asbi)及其用途
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Also Published As

Publication number Publication date
EP1896477B1 (en) 2010-09-22
CN101198609A (zh) 2008-06-11
AR054620A1 (es) 2007-07-04
JP2008543840A (ja) 2008-12-04
DE602006017073D1 (en) 2010-11-04
PE20070018A1 (es) 2007-03-08
KR20080031189A (ko) 2008-04-08
ATE482214T1 (de) 2010-10-15
IL187623A0 (en) 2008-03-20
WO2006138192A1 (en) 2006-12-28
EP1896477A1 (en) 2008-03-12
ZA200710337B (en) 2008-12-31
MX2007016175A (es) 2008-03-07
US7759354B2 (en) 2010-07-20
ES2350854T3 (es) 2011-01-27
CA2610812A1 (en) 2006-12-28
TW200716644A (en) 2007-05-01
US20060281730A1 (en) 2006-12-14
AU2006259675A1 (en) 2006-12-28

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PC Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)

Effective date: 20140612