HK1060129A1 - Novel piperidinecarboxamide derivatives, method f or preparing same and pharmaceutical compositions containing same. - Google Patents

Novel piperidinecarboxamide derivatives, method f or preparing same and pharmaceutical compositions containing same.

Info

Publication number
HK1060129A1
HK1060129A1 HK04103130A HK04103130A HK1060129A1 HK 1060129 A1 HK1060129 A1 HK 1060129A1 HK 04103130 A HK04103130 A HK 04103130A HK 04103130 A HK04103130 A HK 04103130A HK 1060129 A1 HK1060129 A1 HK 1060129A1
Authority
HK
Hong Kong
Prior art keywords
same
pharmaceutical compositions
compositions containing
novel
preparing
Prior art date
Application number
HK04103130A
Other languages
English (en)
Inventor
Xavier Emonds-Alt
Vincenzo Proietto
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of HK1060129A1 publication Critical patent/HK1060129A1/xx

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
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  • Biomedical Technology (AREA)
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  • Pain & Pain Management (AREA)
  • Pulmonology (AREA)
  • Diabetes (AREA)
  • Dermatology (AREA)
  • Hematology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Psychiatry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Rheumatology (AREA)
  • Oncology (AREA)
  • Urology & Nephrology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Vascular Medicine (AREA)
  • Psychology (AREA)
  • Obesity (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Molecular Biology (AREA)
  • Emergency Medicine (AREA)
  • Ophthalmology & Optometry (AREA)
HK04103130A 2001-05-21 2004-05-04 Novel piperidinecarboxamide derivatives, method f or preparing same and pharmaceutical compositions containing same. HK1060129A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0106691A FR2824828B1 (fr) 2001-05-21 2001-05-21 Nouveaux derives de piperidinecarboxamide, un procede pour leur preparation et les compositions pharmaceutiques les contenant
PCT/FR2002/001663 WO2002094821A1 (fr) 2001-05-21 2002-05-17 Nouveaux derives de piperidinecarboxamide, un procede pour leur preparation et les compositions pharmaceutiques les contenant

Publications (1)

Publication Number Publication Date
HK1060129A1 true HK1060129A1 (en) 2004-07-30

Family

ID=8863515

Family Applications (1)

Application Number Title Priority Date Filing Date
HK04103130A HK1060129A1 (en) 2001-05-21 2004-05-04 Novel piperidinecarboxamide derivatives, method f or preparing same and pharmaceutical compositions containing same.

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US (2) US20040180890A1 (cs)
EP (1) EP1395582B1 (cs)
JP (1) JP2004529968A (cs)
KR (1) KR20030097886A (cs)
CN (1) CN1249059C (cs)
AR (1) AR035247A1 (cs)
AT (1) ATE294798T1 (cs)
AU (1) AU2002313065B2 (cs)
BG (1) BG108341A (cs)
BR (1) BR0209877A (cs)
CA (1) CA2445631A1 (cs)
CZ (1) CZ20033132A3 (cs)
DE (1) DE60204015T2 (cs)
DK (1) DK1395582T3 (cs)
EA (1) EA006236B1 (cs)
EE (1) EE200300553A (cs)
ES (1) ES2242032T3 (cs)
FR (1) FR2824828B1 (cs)
HK (1) HK1060129A1 (cs)
HR (1) HRP20030923A2 (cs)
HU (1) HUP0401563A2 (cs)
IL (1) IL158660A0 (cs)
IS (1) IS7008A (cs)
MA (1) MA27022A1 (cs)
MX (1) MXPA03010133A (cs)
NO (1) NO20035163D0 (cs)
NZ (1) NZ529206A (cs)
PL (1) PL367341A1 (cs)
PT (1) PT1395582E (cs)
SK (1) SK14192003A3 (cs)
TN (1) TNSN03118A1 (cs)
TW (1) TWI258480B (cs)
UA (1) UA75400C2 (cs)
WO (1) WO2002094821A1 (cs)
YU (1) YU86603A (cs)
ZA (1) ZA200308344B (cs)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2003300911A1 (en) * 2002-12-13 2004-07-09 Smithkline Beecham Corporation Heterocyclic compounds as ccr5 antagonists
FR2873373B1 (fr) 2004-07-23 2006-09-08 Sanofi Synthelabo Derives de 4-arylmorpholin-3-one, leur preparation et leur application en therapeutique
US20070219214A1 (en) * 2006-02-01 2007-09-20 Solvay Pharmaceuticals Gmbh Dual NK2/NK3-antagonists, pharmaceutical compositions comprising them, and processes for their preparation
RU2008135123A (ru) * 2006-02-01 2010-03-10 Зольвай Фармасьютикалз Гмбх (De) Новые двойные антагонисты nk2/nk3, содержащие их фармацевтические композиции и способы их получения
FR2912058A1 (fr) * 2007-02-07 2008-08-08 Sanofi Aventis Sa Utilisation d'un compose antagoniste des recepteurs nk2 de la neurokinine a pour la preparation de medicaments utiles pour la prevention et le traitement des dysfonctions sexuelles
AU2009203874B2 (en) * 2008-01-11 2014-08-21 United Paragon Associates Inc. Fertilized egg isolate and use thereof
US20110152233A1 (en) * 2009-12-18 2011-06-23 Henner Knust Pyrrolidine compounds
CN102884059B (zh) * 2010-03-11 2015-08-26 大日本住友制药株式会社 N-酰基环胺衍生物或其可药用盐
EP3160469B1 (en) 2014-06-25 2021-04-28 Emory University Methods of managing conditioned fear with neurokinin receptor antagonists
EP3881843A4 (en) * 2018-11-15 2022-08-03 Kyushu University, National University Corporation PROPHYLACTIC OR THERAPEUTIC AGENT AND MEDICAL COMPOSITION FOR IL-31 MEDIATED DISEASE

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5689663A (en) * 1992-06-19 1997-11-18 Microsoft Corporation Remote controller user interface and methods relating thereto
FR2729954B1 (fr) * 1995-01-30 1997-08-01 Sanofi Sa Composes heterocycliques substitues, procede pour leur preparation et compositions pharmaceutiques les contenant
US5780466A (en) * 1995-01-30 1998-07-14 Sanofi Substituted heterocyclic compounds method of preparing them and pharmaceutical compositions in which they are present
FR2738819B1 (fr) * 1995-09-14 1997-12-05 Sanofi Sa Nouveaux composes antagonistes selectifs du recepteur nk3 humain, procede pour leur obtention et compositions pharmaceutiques les contenant
RU2135494C1 (ru) * 1995-12-01 1999-08-27 Санкио Компани Лимитед Гетероциклические соединения и композиция на их основе, проявляющая антагонистическое действие в отношении рецепторов тахикинина
JP3192631B2 (ja) * 1997-05-28 2001-07-30 三共株式会社 飽和複素環化合物からなる医薬
BR9815348A (pt) * 1997-12-04 2000-10-17 Sankyo Co " composto, uso deste ou de um sal farmacologicamente aceitável, éster ou outro derivado do mesmo, medicamento, agentes preventivos ou terapêuticos para asma e/ou bronquite, para rinite, para doença alérgica, e para incontinência urinária, e, processos de prevenção ou tratamento de asma e/ou bronquite, de rinite, de doença alérgica, e de incontinência urinária. "
WO2000034274A1 (fr) * 1998-12-10 2000-06-15 Sankyo Company, Limited Derives de la cyclohexylpiperidine
FR2791346B3 (fr) * 1999-03-25 2001-04-27 Sanofi Sa Nouveaux derives de morpholine, procede pour leur preparation et compositions pharmaceutiques les contenant

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UA75400C2 (en) 2006-04-17
FR2824828B1 (fr) 2005-05-20
DE60204015D1 (de) 2005-06-09
MA27022A1 (fr) 2004-12-20
EP1395582B1 (fr) 2005-05-04
CZ20033132A3 (cs) 2004-02-18
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ATE294798T1 (de) 2005-05-15
JP2004529968A (ja) 2004-09-30
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MXPA03010133A (es) 2005-03-31
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ZA200308344B (en) 2004-10-27
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US20040180890A1 (en) 2004-09-16
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DK1395582T3 (da) 2005-08-29
FR2824828A1 (fr) 2002-11-22
US20080261976A1 (en) 2008-10-23
HUP0401563A2 (hu) 2004-12-28
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