HK1056687A1 - Method of treating estrogen receptor positive carcinoma. - Google Patents
Method of treating estrogen receptor positive carcinoma.Info
- Publication number
- HK1056687A1 HK1056687A1 HK03109077A HK03109077A HK1056687A1 HK 1056687 A1 HK1056687 A1 HK 1056687A1 HK 03109077 A HK03109077 A HK 03109077A HK 03109077 A HK03109077 A HK 03109077A HK 1056687 A1 HK1056687 A1 HK 1056687A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- estrogen receptor
- receptor positive
- positive carcinoma
- treating estrogen
- treating
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
- A61K31/4745—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/32—Antioestrogens
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Molecular Biology (AREA)
- Engineering & Computer Science (AREA)
- Endocrinology (AREA)
- Diabetes (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US22432600P | 2000-08-11 | 2000-08-11 | |
PCT/US2001/024615 WO2002013802A2 (fr) | 2000-08-11 | 2001-08-06 | Procede de traitement d'un carcinome a recepteur d'oestrogene |
Publications (1)
Publication Number | Publication Date |
---|---|
HK1056687A1 true HK1056687A1 (en) | 2004-02-27 |
Family
ID=22840171
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HK03109077A HK1056687A1 (en) | 2000-08-11 | 2003-12-12 | Method of treating estrogen receptor positive carcinoma. |
Country Status (15)
Country | Link |
---|---|
US (1) | US6511986B2 (fr) |
EP (1) | EP1318837B1 (fr) |
JP (1) | JP2004507465A (fr) |
CN (1) | CN100448487C (fr) |
AR (1) | AR033555A1 (fr) |
AT (1) | ATE278421T1 (fr) |
AU (1) | AU2001283139A1 (fr) |
CA (1) | CA2416976C (fr) |
DE (1) | DE60106281T2 (fr) |
DK (1) | DK1318837T3 (fr) |
ES (1) | ES2228932T3 (fr) |
HK (1) | HK1056687A1 (fr) |
MX (1) | MXPA03001245A (fr) |
PT (1) | PT1318837E (fr) |
WO (1) | WO2002013802A2 (fr) |
Families Citing this family (74)
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US20030215445A1 (en) | 1997-05-23 | 2003-11-20 | Ginette Serrero | Methods and compositions for inhibiting the growth of hematopoietic malignant cells |
US7091047B2 (en) * | 1997-05-23 | 2006-08-15 | A&G Pharmaceutical, Inc. | Methods and kits for diagnosing tumorigenicity |
US6720159B1 (en) * | 1997-12-16 | 2004-04-13 | A&G Pharmaceutical, Inc. | 88KDA tumorigenic growth factor and antagonists |
US6881548B2 (en) * | 1997-05-23 | 2005-04-19 | A&G Pharmaceutical, Inc. | Methods and kits for diagnosing tumorigenicity and determining resistance to the antineoplastic effects of antiestrogen therapy |
US8512960B2 (en) * | 1997-05-23 | 2013-08-20 | A&G Pharmaceutical, Inc. | 88kDa tumorigenic growth factor and antagonists |
US6309826B1 (en) | 1997-05-23 | 2001-10-30 | Ginette Serrero | 88kDa tumorigenic growth factor and antagonists |
US20100111928A1 (en) * | 1997-05-23 | 2010-05-06 | A & G Pharmaceutical, Inc. | Methods and kits for diagnosis tumorgenicity |
US7617145B1 (en) * | 2000-10-24 | 2009-11-10 | Worldwide Farm Equipment Auctions.Com Ltd. | Adaptive bidding increments in an online auction system |
TWI286074B (en) | 2000-11-15 | 2007-09-01 | Wyeth Corp | Pharmaceutical composition containing CCI-779 as an antineoplastic agent |
EP2269603B1 (fr) * | 2001-02-19 | 2015-05-20 | Novartis AG | Traitement des tumeurs du sein avec un dérivé de la rapamycine en association avec l'exémestane |
AU2016206379B2 (en) * | 2001-02-19 | 2017-09-14 | Novartis Ag | Cancer Treatment |
AU2011226833B9 (en) * | 2001-02-19 | 2014-07-03 | Novartis Ag | Cancer treatment |
ATE427948T1 (de) | 2001-04-24 | 2009-04-15 | Purdue Research Foundation | Folat-mimetika und deren folatrezeptorbindende konjugate |
CA2453337C (fr) * | 2001-07-09 | 2012-08-28 | Zonagen, Inc. | Methodes et materiaux destines au traitement de la deficience en testosterone chez l'homme |
UA77200C2 (en) | 2001-08-07 | 2006-11-15 | Wyeth Corp | Antineoplastic combination of cci-779 and bkb-569 |
PL216224B1 (pl) | 2002-02-01 | 2014-03-31 | Ariad Pharmaceuticals | Pochodne rapamycyny zawierające fosfor, kompozycja je zawierająca oraz ich zastosowanie |
KR20040106547A (ko) * | 2002-05-15 | 2004-12-17 | 엔도사이트, 인코포레이티드 | 비타민-마이토마이신 공액체 |
US7411045B2 (en) * | 2002-11-19 | 2008-08-12 | A&G Pharmaceutical, Inc. | Autocrine growth factor receptor antibodies and methods |
EP2517730A3 (fr) | 2003-01-27 | 2013-01-02 | Endocyte, Inc. | Conjugués d'administration de médicaments à liaison au récepteur de vitamines |
ES2369695T3 (es) * | 2003-02-26 | 2011-12-05 | A & G PHARMACEUTICAL, INC. | Métodos para incrementar la proliferación de células b. |
UA83484C2 (uk) * | 2003-03-05 | 2008-07-25 | Уайт | Спосіб лікування раку грудей комбінацією похідного рапаміцину і інгібітора ароматази - летрозолу, фармацевтична композиція |
KR20060006058A (ko) * | 2003-04-22 | 2006-01-18 | 와이어쓰 | 항신생물성 배합물 |
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RU2345772C2 (ru) * | 2003-07-25 | 2009-02-10 | Уайт | Лиофилизированные композиции cci-779 |
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JP5558358B2 (ja) | 2007-10-16 | 2014-07-23 | レプロス セラピューティクス インコーポレイティド | メタボリック症候群用のtrans−クロミフェン |
US8022216B2 (en) | 2007-10-17 | 2011-09-20 | Wyeth Llc | Maleate salts of (E)-N-{4-[3-chloro-4-(2-pyridinylmethoxy)anilino]-3-cyano-7-ethoxy-6-quinolinyl}-4-(dimethylamino)-2-butenamide and crystalline forms thereof |
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KR20180128078A (ko) | 2008-06-17 | 2018-11-30 | 와이어쓰 엘엘씨 | Hki-272 및 비노렐빈을 함유하는 항신생물성 조합물 |
NZ590464A (en) | 2008-08-04 | 2012-10-26 | Wyeth Llc | Antineoplastic combinations of the 4-anilino-3-cyanoquinoline neratinib and capecitabine |
HUE061640T2 (hu) | 2009-04-06 | 2023-07-28 | Wyeth Llc | Gyógykezelési rendszer mellrákhoz neratinib alkalmazásával |
ES2627692T3 (es) | 2010-06-10 | 2017-07-31 | Aragon Pharmaceuticals, Inc. | Moduladores de receptores de estrógenos y usos de los mismos |
UA113291C2 (xx) | 2011-08-04 | 2017-01-10 | Метаболіти транскломіфену і їх застосування | |
WO2013090829A1 (fr) | 2011-12-14 | 2013-06-20 | Aragon Pharmaceuticals, Inc. | Modulateurs des récepteurs des œstrogènes et ses utilisations |
US10080805B2 (en) | 2012-02-24 | 2018-09-25 | Purdue Research Foundation | Cholecystokinin B receptor targeting for imaging and therapy |
US20140080175A1 (en) | 2012-03-29 | 2014-03-20 | Endocyte, Inc. | Processes for preparing tubulysin derivatives and conjugates thereof |
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RU2560708C1 (ru) * | 2014-03-24 | 2015-08-20 | Федеральное государственное бюджетное учреждение "Научно-исследовательский институт клинической и экспериментальной лимфологии" Сибирского отделения Российской академии медицинских наук (ФГБУ "НИИКЭЛ" СО РАМН) | Способ воздействия на клетки гепатокарциномы в зависимости от стадии их дифференцировки нанопрепаратами лития |
UA122346C2 (uk) | 2015-10-01 | 2020-10-26 | Олема Фармасьютикалз, Інк. | ТЕТРАГІДРО-1H-ПІРИДО[3,4-b]ІНДОЛЬНІ АНТИЕСТРОГЕННІ ЛІКАРСЬКІ ПРЕПАРАТИ |
WO2017100715A1 (fr) | 2015-12-09 | 2017-06-15 | The Board Of Trustees Of The University Of Illinois | Composés régulateurs à la baisse des récepteurs des œstrogènes sélectifs à base de benzothiophène |
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JP6892151B2 (ja) | 2016-10-11 | 2021-06-23 | デューク ユニバーシティ | Er+乳がんのラソフォキシフェン処置 |
WO2018081168A2 (fr) | 2016-10-24 | 2018-05-03 | The Board Of Trustees Of The University Of Illinois | Répresseurs du récepteur oestrogénique sélectifs mixtes à base de benzothiophène |
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KR20190117582A (ko) | 2017-02-10 | 2019-10-16 | 쥐원 쎄라퓨틱스, 인크. | 벤조티오펜 에스트로겐 수용체 조정제 |
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EP3773524A4 (fr) | 2018-04-10 | 2021-12-22 | Duke University | Traitement du cancer du sein avec du lasofoxifène |
WO2020132561A1 (fr) | 2018-12-20 | 2020-06-25 | C4 Therapeutics, Inc. | Dégradation ciblée de protéines |
TW202136265A (zh) | 2019-12-20 | 2021-10-01 | 美商C4醫藥公司 | 用於降解egfr的異吲哚啉酮及吲唑化合物 |
TW202146412A (zh) | 2020-03-05 | 2021-12-16 | 美商C4醫藥公司 | 用於標靶降解brd9之化合物 |
GB202116903D0 (en) | 2021-11-18 | 2022-01-05 | Sermonix Pharmaceuticals Inc | Lasofoxifene treatment of aromatase-resistant er+ cancer |
WO2024030968A1 (fr) | 2022-08-03 | 2024-02-08 | Brystol-Myers Squibb Company | Composés pour moduler la protéine ret |
WO2024097980A1 (fr) | 2022-11-04 | 2024-05-10 | Bristol-Myers Squibb Company | Inhibiteurs de protéines ret-ldd |
WO2024097989A1 (fr) | 2022-11-04 | 2024-05-10 | Bristol-Myers Squibb Company | Agents de dégradation de protéine ret-ldd |
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-
2001
- 2001-08-06 PT PT01961914T patent/PT1318837E/pt unknown
- 2001-08-06 AU AU2001283139A patent/AU2001283139A1/en not_active Abandoned
- 2001-08-06 CA CA002416976A patent/CA2416976C/fr not_active Expired - Fee Related
- 2001-08-06 AT AT01961914T patent/ATE278421T1/de not_active IP Right Cessation
- 2001-08-06 ES ES01961914T patent/ES2228932T3/es not_active Expired - Lifetime
- 2001-08-06 EP EP01961914A patent/EP1318837B1/fr not_active Expired - Lifetime
- 2001-08-06 US US09/923,217 patent/US6511986B2/en not_active Expired - Fee Related
- 2001-08-06 CN CNB018137539A patent/CN100448487C/zh not_active Expired - Fee Related
- 2001-08-06 WO PCT/US2001/024615 patent/WO2002013802A2/fr active IP Right Grant
- 2001-08-06 DK DK01961914T patent/DK1318837T3/da active
- 2001-08-06 MX MXPA03001245A patent/MXPA03001245A/es active IP Right Grant
- 2001-08-06 JP JP2002518948A patent/JP2004507465A/ja not_active Withdrawn
- 2001-08-06 DE DE60106281T patent/DE60106281T2/de not_active Expired - Fee Related
- 2001-08-10 AR ARP010103839A patent/AR033555A1/es unknown
-
2003
- 2003-12-12 HK HK03109077A patent/HK1056687A1/xx not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
ES2228932T3 (es) | 2005-04-16 |
DE60106281T2 (de) | 2005-02-24 |
JP2004507465A (ja) | 2004-03-11 |
CN1446106A (zh) | 2003-10-01 |
ATE278421T1 (de) | 2004-10-15 |
AU2001283139A1 (en) | 2002-02-25 |
CA2416976A1 (fr) | 2002-02-21 |
PT1318837E (pt) | 2004-12-31 |
US6511986B2 (en) | 2003-01-28 |
US20020045638A1 (en) | 2002-04-18 |
CN100448487C (zh) | 2009-01-07 |
DK1318837T3 (da) | 2005-01-10 |
WO2002013802A2 (fr) | 2002-02-21 |
EP1318837B1 (fr) | 2004-10-06 |
CA2416976C (fr) | 2008-05-20 |
WO2002013802A3 (fr) | 2003-03-27 |
EP1318837A2 (fr) | 2003-06-18 |
DE60106281D1 (de) | 2004-11-11 |
MXPA03001245A (es) | 2003-05-27 |
AR033555A1 (es) | 2003-12-26 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PC | Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee) |
Effective date: 20080806 |