HK1043365B - N-(亞氨基甲基)胺衍生物，其製備方法，其作為藥物的用途以及含有該化合物的藥物組合物 - Google Patents

N-(亞氨基甲基)胺衍生物，其製備方法，其作為藥物的用途以及含有該化合物的藥物組合物

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Publication number
HK1043365B
HK1043365B HK02105058.6A HK02105058A HK1043365B HK 1043365 B HK1043365 B HK 1043365B HK 02105058 A HK02105058 A HK 02105058A HK 1043365 B HK1043365 B HK 1043365B
Authority
HK
Hong Kong
Prior art keywords
iminomethyl
medicines
preparation
compositions containing
amine derivatives
Prior art date
Application number
HK02105058.6A
Other languages
English (en)
Other versions
HK1043365A1 (en
Inventor
D‧比戈
P-E‧查波利爾德拉索尼爾
S‧奧溫
J‧哈奈特
G‧尤裡巴利
Original Assignee
Ipsen Pharma Sas
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ipsen Pharma Sas filed Critical Ipsen Pharma Sas
Publication of HK1043365A1 publication Critical patent/HK1043365A1/xx
Publication of HK1043365B publication Critical patent/HK1043365B/zh

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • A—HUMAN NECESSITIES
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D333/40—Thiophene-2-carboxylic acid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

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HK02105058.6A 1998-09-23 2002-07-08 N-(亞氨基甲基)胺衍生物，其製備方法，其作為藥物的用途以及含有該化合物的藥物組合物 HK1043365B (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9811867A FR2784678B1 (fr) 1998-09-23 1998-09-23 Nouveaux derives de n-(iminomethyl)amines, leur preparation, leur application a titre de medicaments et les compositions pharmaceutiques les contenant
PCT/FR1999/002251 WO2000017191A2 (fr) 1998-09-23 1999-09-22 Derives de n-(iminomethyl)amines, leur preparation, leur application a titre de medicaments et les compositions pharmaceutiques les contenant

Publications (2)

Publication Number Publication Date
HK1043365A1 HK1043365A1 (en) 2002-09-13
HK1043365B true HK1043365B (zh) 2005-01-07

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Country Status (26)

Country Link
US (5) US6482822B1 (zh)
EP (1) EP1115720B1 (zh)
JP (1) JP2003517444A (zh)
KR (1) KR100655340B1 (zh)
CN (1) CN1144799C (zh)
AR (1) AR024837A1 (zh)
AT (1) ATE399774T1 (zh)
AU (1) AU759958B2 (zh)
BR (1) BR9913899A (zh)
CA (1) CA2344223A1 (zh)
CZ (1) CZ299664B6 (zh)
DE (1) DE69939021D1 (zh)
DK (1) DK1115720T3 (zh)
ES (1) ES2310045T3 (zh)
FR (1) FR2784678B1 (zh)
HK (1) HK1043365B (zh)
HU (1) HUP0104013A3 (zh)
IL (2) IL141997A0 (zh)
MY (1) MY123219A (zh)
NO (1) NO328466B1 (zh)
NZ (1) NZ511188A (zh)
PL (1) PL347471A1 (zh)
PT (1) PT1115720E (zh)
RU (1) RU2230742C2 (zh)
WO (1) WO2000017191A2 (zh)
ZA (1) ZA200103206B (zh)

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NO328466B1 (no) 2010-02-22
NO20011478D0 (no) 2001-03-22
WO2000017191A3 (fr) 2000-10-26
DK1115720T3 (da) 2008-11-03
JP2003517444A (ja) 2003-05-27
IL141997A (en) 2008-07-08
US20050027009A1 (en) 2005-02-03
IL141997A0 (en) 2002-03-10
US6809090B2 (en) 2004-10-26
US6620840B1 (en) 2003-09-16
NZ511188A (en) 2003-08-29
PT1115720E (pt) 2008-10-08
AU5631599A (en) 2000-04-10
US20050197329A1 (en) 2005-09-08
HUP0104013A3 (en) 2003-01-28
CN1335841A (zh) 2002-02-13
AR024837A1 (es) 2002-10-30
KR100655340B1 (ko) 2006-12-08
ZA200103206B (en) 2002-07-19
FR2784678B1 (fr) 2002-11-29
CA2344223A1 (fr) 2000-03-30
EP1115720B1 (fr) 2008-07-02
CN1144799C (zh) 2004-04-07
ES2310045T3 (es) 2008-12-16
US7186752B2 (en) 2007-03-06
HUP0104013A2 (hu) 2002-04-29
EP1115720A2 (fr) 2001-07-18
KR20010085832A (ko) 2001-09-07
NO20011478L (no) 2001-03-22
ATE399774T1 (de) 2008-07-15
PL347471A1 (en) 2002-04-08
AU759958B2 (en) 2003-05-01
BR9913899A (pt) 2001-07-03
FR2784678A1 (fr) 2000-04-21
CZ20011056A3 (cs) 2002-01-16
CZ299664B6 (cs) 2008-10-08
MY123219A (en) 2006-05-31
US20040097494A1 (en) 2004-05-20
US6482822B1 (en) 2002-11-19
WO2000017191A2 (fr) 2000-03-30
DE69939021D1 (de) 2008-08-14
HK1043365A1 (en) 2002-09-13
RU2230742C2 (ru) 2004-06-20

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