GT200800253A - Sales y modificaciones del cristal de las mismas - Google Patents

Sales y modificaciones del cristal de las mismas

Info

Publication number
GT200800253A
GT200800253A GT200800253A GT200800253A GT200800253A GT 200800253 A GT200800253 A GT 200800253A GT 200800253 A GT200800253 A GT 200800253A GT 200800253 A GT200800253 A GT 200800253A GT 200800253 A GT200800253 A GT 200800253A
Authority
GT
Guatemala
Prior art keywords
salts
same
crystal
modifications
phenyl
Prior art date
Application number
GT200800253A
Other languages
English (en)
Inventor
Feng Lili
Jiang Xinglong
Karpinski Piortr
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of GT200800253A publication Critical patent/GT200800253A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • A61K31/55131,4-Benzodiazepines, e.g. diazepam or clozapine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Molecular Biology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

LA INVENCIÓN SE REFIERE A SALES DE 1-(2-FLUORO-FENIL)-3-(2-OXO-5-FENIL-2,3-DIHIDRO-1H-BENZO-[E]-[1,4]-DIAZEPIN-3-IL)-UREA, Y A LAS FORMAS CRISTALINAS DE LAS MISMAS, A SU PRODUCCIÓN Y USO, Y A PREPARACIONES FARMACÉUTICAS QUE CONTIENEN ESTAS SALES Y FORMAS CRISTALINAS. T2008
GT200800253A 2006-05-23 2008-11-21 Sales y modificaciones del cristal de las mismas GT200800253A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US80283606P 2006-05-23 2006-05-23

Publications (1)

Publication Number Publication Date
GT200800253A true GT200800253A (es) 2009-04-29

Family

ID=38704747

Family Applications (1)

Application Number Title Priority Date Filing Date
GT200800253A GT200800253A (es) 2006-05-23 2008-11-21 Sales y modificaciones del cristal de las mismas

Country Status (28)

Country Link
US (1) US7977330B2 (es)
EP (1) EP2029556B1 (es)
JP (2) JP2009538330A (es)
KR (1) KR20090009898A (es)
CN (1) CN101448796B (es)
AR (1) AR061056A1 (es)
AT (1) ATE486858T1 (es)
AU (1) AU2007267671A1 (es)
BR (1) BRPI0712556A2 (es)
CA (1) CA2650514A1 (es)
CL (1) CL2007001454A1 (es)
CR (1) CR10431A (es)
DE (1) DE602007010286D1 (es)
EC (1) ECSP088900A (es)
ES (1) ES2355166T3 (es)
GT (1) GT200800253A (es)
IL (1) IL195008A0 (es)
MA (1) MA30482B1 (es)
MX (1) MX2008014836A (es)
NO (1) NO20085000L (es)
PE (1) PE20080261A1 (es)
PL (1) PL2029556T3 (es)
PT (1) PT2029556E (es)
RU (1) RU2008150627A (es)
TN (1) TNSN08477A1 (es)
TW (1) TW200815375A (es)
WO (1) WO2007140154A2 (es)
ZA (1) ZA200809096B (es)

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EA012387B1 (ru) * 2002-09-20 2009-10-30 Эрроу Терапьютикс Лимитед Производные бензодиазепина, содержащие их продукт и фармацевтическая композиция и их применение

Also Published As

Publication number Publication date
IL195008A0 (en) 2009-08-03
ATE486858T1 (de) 2010-11-15
CN101448796A (zh) 2009-06-03
US20090163478A1 (en) 2009-06-25
DE602007010286D1 (de) 2010-12-16
EP2029556A2 (en) 2009-03-04
AR061056A1 (es) 2008-07-30
TNSN08477A1 (en) 2010-04-14
MA30482B1 (fr) 2009-06-01
PE20080261A1 (es) 2008-04-18
CL2007001454A1 (es) 2008-05-16
EP2029556B1 (en) 2010-11-03
CN101448796B (zh) 2012-09-26
WO2007140154A3 (en) 2008-03-20
MX2008014836A (es) 2008-12-01
BRPI0712556A2 (pt) 2013-07-02
AU2007267671A1 (en) 2007-12-06
WO2007140154A2 (en) 2007-12-06
JP2009538330A (ja) 2009-11-05
KR20090009898A (ko) 2009-01-23
JP2013075910A (ja) 2013-04-25
ES2355166T3 (es) 2011-03-23
RU2008150627A (ru) 2010-06-27
CA2650514A1 (en) 2007-12-06
TW200815375A (en) 2008-04-01
NO20085000L (no) 2008-12-23
PL2029556T3 (pl) 2011-04-29
PT2029556E (pt) 2011-01-31
ZA200809096B (en) 2009-11-25
ECSP088900A (es) 2008-12-30
CR10431A (es) 2009-01-07
US7977330B2 (en) 2011-07-12

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