GT200600217A - Proceso para la sintesis de compuestos organicos - Google Patents

Proceso para la sintesis de compuestos organicos

Info

Publication number
GT200600217A
GT200600217A GT200600217A GT200600217A GT200600217A GT 200600217 A GT200600217 A GT 200600217A GT 200600217 A GT200600217 A GT 200600217A GT 200600217 A GT200600217 A GT 200600217A GT 200600217 A GT200600217 A GT 200600217A
Authority
GT
Guatemala
Prior art keywords
synthesis
organic compounds
useful
compounds
thyrosines
Prior art date
Application number
GT200600217A
Other languages
English (en)
Spanish (es)
Inventor
Joseph Mckenna
Wen-Chung Shieh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of GT200600217A publication Critical patent/GT200600217A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyridine Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Steroid Compounds (AREA)
GT200600217A 2005-06-09 2006-05-24 Proceso para la sintesis de compuestos organicos GT200600217A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US68897705P 2005-06-09 2005-06-09
US70559005P 2005-08-04 2005-08-04

Publications (1)

Publication Number Publication Date
GT200600217A true GT200600217A (es) 2007-03-28

Family

ID=37091153

Family Applications (1)

Application Number Title Priority Date Filing Date
GT200600217A GT200600217A (es) 2005-06-09 2006-05-24 Proceso para la sintesis de compuestos organicos

Country Status (31)

Country Link
US (2) US8124763B2 (https=)
EP (1) EP1924574B1 (https=)
JP (1) JP5118024B2 (https=)
KR (3) KR101216249B1 (https=)
AR (1) AR053890A1 (https=)
AT (1) ATE487709T1 (https=)
AU (1) AU2006258051B2 (https=)
BR (1) BRPI0611663A2 (https=)
CA (1) CA2610105C (https=)
CY (1) CY1111428T1 (https=)
DE (1) DE602006018156D1 (https=)
DK (1) DK1924574T3 (https=)
EC (1) ECSP077982A (https=)
EG (1) EG25039A (https=)
GT (1) GT200600217A (https=)
IL (1) IL187421A (https=)
JO (1) JO2636B1 (https=)
MA (1) MA29599B1 (https=)
MX (1) MX2007015423A (https=)
MY (1) MY147436A (https=)
NO (1) NO340743B1 (https=)
NZ (1) NZ563740A (https=)
PE (1) PE20070015A1 (https=)
PL (1) PL1924574T3 (https=)
PT (1) PT1924574E (https=)
RU (1) RU2444520C2 (https=)
SA (1) SA06270147B1 (https=)
SI (1) SI1924574T1 (https=)
TN (1) TNSN07463A1 (https=)
TW (1) TWI430999B (https=)
WO (1) WO2006135641A2 (https=)

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EP2305667A3 (en) 2008-07-17 2011-05-11 Teva Pharmaceutical Industries Ltd. Nilotinib intermediates and preparation thereof
EP2262793B1 (en) 2008-11-05 2012-10-03 Teva Pharmaceutical Industries Ltd. Nilotinib hci crystalline forms
WO2010060074A1 (en) * 2008-11-24 2010-05-27 Teva Pharmaceutical Industries Ltd. Preparation of nilotinib and intermediates thereof
US20110053968A1 (en) 2009-06-09 2011-03-03 Auspex Pharmaceuticals, Inc. Aminopyrimidine inhibitors of tyrosine kinase
JO3634B1 (ar) 2009-11-17 2020-08-27 Novartis Ag طريقة لعلاج اضطرابات تكاثرية وحالات مرضية أخرى متوسطة بنشاط كيناز bcr-abl، c-kit، ddr1، ddr2، أو pdgf-r
EP2691539B1 (en) 2011-03-31 2018-04-25 The Procter and Gamble Company Methods for identifying and evaluating skin-active agents effective for treating dandruff
AR086913A1 (es) * 2011-06-14 2014-01-29 Novartis Ag 4-metil-3-[[4-(3-piridinil)-2-pirimidinil]-amino]-n-[5-(4-metil-1h-imidazol-1-il)-3-(trifluoro-metil)-fenil]-benzamida amorfa, forma de dosificacion que la contiene y metodo para prepararlas
GB2514285B (en) 2012-02-13 2018-07-18 Grindeks Jsc Intermediates for a novel process of preparing imatinib and related tyrosine kinase inhibitors
US9920357B2 (en) 2012-06-06 2018-03-20 The Procter & Gamble Company Systems and methods for identifying cosmetic agents for hair/scalp care compositions
WO2015092624A1 (en) 2013-12-16 2015-06-25 Ranbaxy Laboratories Limited Nilotinib mono-oxalate and its crystalline form
CN103694176B (zh) 2014-01-07 2015-02-18 苏州立新制药有限公司 尼洛替尼中间体的制备方法
EP3095782A1 (en) 2015-05-18 2016-11-23 Esteve Química, S.A. New method for preparing 3-(4-methyl-1h-imidazol-1-yl)-5-(trifluoromethyl)benzenamine
EP3749697A4 (en) 2018-02-05 2021-11-03 Bio-Rad Laboratories, Inc. CHROMATOGRAPHY RESIN WITH LIGAND MIXED MODE ANIONIC / HYDROPHOBIC EXCHANGE
CN113292537B (zh) 2018-06-15 2024-04-05 汉达癌症医药责任有限公司 激酶抑制剂的盐类及其组合物
JP2020007240A (ja) * 2018-07-04 2020-01-16 住友化学株式会社 ベンズアミド化合物の製造方法

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CA2151491A1 (en) 1992-12-24 1994-07-07 Robert J. Kaufman Fluorocarbon emulsions
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US5597829A (en) 1994-05-09 1997-01-28 Bionumerik Pharmaceuticals, Inc. Lactone stable formulation of camptothecin and methods for uses thereof
US5726181A (en) 1995-06-05 1998-03-10 Bionumerik Pharmaceuticals, Inc. Formulations and compositions of poorly water soluble camptothecin derivatives
US6323366B1 (en) 1997-07-29 2001-11-27 Massachusetts Institute Of Technology Arylamine synthesis
AR013261A1 (es) 1997-08-01 2000-12-13 Smithkline Beecham Corp Formulaciones farmaceuticas para analogos de camptotecina en capsula de gelatina
US20030059465A1 (en) 1998-05-11 2003-03-27 Unger Evan C. Stabilized nanoparticle formulations of camptotheca derivatives
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ATE216998T1 (de) 1999-03-09 2002-05-15 Sigma Tau Ind Farmaceuti Camptothecin-derivate mit antitumor-wirkung
IT1306129B1 (it) 1999-04-13 2001-05-30 Sigma Tau Ind Farmaceuti Esteri della l-carnitina o di alcanoil l-carnitine utilizzabili comelipidi cationici per l'immissione intracellulare di composti
DE19926056B4 (de) 1999-06-08 2004-03-25 Gkss-Forschungszentrum Geesthacht Gmbh Einrichtung zur Analyse atomarer und/oder molekularer Elemente mittels wellenlängendispersiver, röntgenspektrometrischer Einrichtungen
GB9918885D0 (en) 1999-08-10 1999-10-13 Pharmacia & Upjohn Spa Pharmaceutical formulations in hydroxypropymethycellulose capsules
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US20040009229A1 (en) 2000-01-05 2004-01-15 Unger Evan Charles Stabilized nanoparticle formulations of camptotheca derivatives
US20020150615A1 (en) 2001-02-12 2002-10-17 Howard Sands Injectable pharmaceutical composition comprising microdroplets of a camptothecin
US6629598B2 (en) 2001-08-10 2003-10-07 Vinod K. Narula Flexible ribbed splint system
US6653319B1 (en) 2001-08-10 2003-11-25 University Of Kentucky Research Foundation Pharmaceutical formulation for poorly water soluble camptothecin analogues
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AU2002353118A1 (en) 2001-12-11 2003-07-24 Dor Biopharma, Inc. Lipid particles and suspensions and uses thereof
JP2003267891A (ja) 2002-03-13 2003-09-25 Mitsubishi-Kagaku Foods Corp W/o/w型エマルション製剤
US7202367B2 (en) 2002-05-31 2007-04-10 Rhodia Chimie Process for arylating or vinylating or alkynating a nucleophilic compound
CZ294371B6 (cs) 2002-06-10 2004-12-15 Pliva - Lachema, A. S. Stabilizovaná farmaceutická kompozice na bázi polyoxyethylovaného ricinového oleje a způsob její přípravy
EP1393719A1 (en) 2002-08-23 2004-03-03 Munich Biotech AG Camptothecin-carboxylate formulations
GB0215676D0 (en) * 2002-07-05 2002-08-14 Novartis Ag Organic compounds
JP4426749B2 (ja) 2002-07-11 2010-03-03 株式会社産学連携機構九州 O/w型エマルション製剤
US20040171560A1 (en) 2002-12-23 2004-09-02 Dabur Research Foundation Stabilized pharmaceutical composition
JP2006199590A (ja) 2003-09-04 2006-08-03 Nano Career Kk 水溶性の塩基性薬物内包ナノ粒子含有組成物
BRPI0415858A (pt) 2003-10-29 2007-01-09 Sonus Pharma Inc compostos de medicamentos terapêuticos modificados por tocoferol
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GT200500310A (es) 2004-11-19 2006-06-19 Compuestos organicos

Also Published As

Publication number Publication date
KR20120066067A (ko) 2012-06-21
IL187421A0 (en) 2008-02-09
KR20130118394A (ko) 2013-10-29
SA06270147B1 (ar) 2009-12-22
ATE487709T1 (de) 2010-11-15
JP5118024B2 (ja) 2013-01-16
US20120116081A1 (en) 2012-05-10
MA29599B1 (fr) 2008-07-01
TWI430999B (zh) 2014-03-21
EP1924574A2 (en) 2008-05-28
NZ563740A (en) 2011-03-31
CA2610105A1 (en) 2006-12-21
KR101514593B1 (ko) 2015-04-22
TNSN07463A1 (en) 2009-03-17
TW200726756A (en) 2007-07-16
CY1111428T1 (el) 2015-08-05
NO20080157L (no) 2008-01-09
KR101216249B1 (ko) 2012-12-28
RU2007148231A (ru) 2009-07-20
US8124763B2 (en) 2012-02-28
AU2006258051B2 (en) 2010-09-09
PT1924574E (pt) 2011-02-08
AU2006258051A1 (en) 2006-12-21
PE20070015A1 (es) 2007-02-06
HK1117524A1 (en) 2009-01-16
JP2008545786A (ja) 2008-12-18
ECSP077982A (es) 2008-01-23
US8946416B2 (en) 2015-02-03
JO2636B1 (en) 2012-06-17
DK1924574T3 (da) 2011-02-14
CA2610105C (en) 2014-03-25
PL1924574T3 (pl) 2011-04-29
AR053890A1 (es) 2007-05-23
MY147436A (en) 2012-12-14
KR20080022093A (ko) 2008-03-10
EP1924574B1 (en) 2010-11-10
DE602006018156D1 (de) 2010-12-23
WO2006135641A3 (en) 2007-03-29
IL187421A (en) 2011-11-30
MX2007015423A (es) 2008-02-21
NO340743B1 (no) 2017-06-12
RU2444520C2 (ru) 2012-03-10
BRPI0611663A2 (pt) 2010-09-28
US20080188656A1 (en) 2008-08-07
SI1924574T1 (sl) 2011-02-28
WO2006135641A2 (en) 2006-12-21
EG25039A (en) 2011-07-06

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