GT200300138A - Moduladores del receptor de glucocorticoides - Google Patents
Moduladores del receptor de glucocorticoidesInfo
- Publication number
- GT200300138A GT200300138A GT200300138A GT200300138A GT200300138A GT 200300138 A GT200300138 A GT 200300138A GT 200300138 A GT200300138 A GT 200300138A GT 200300138 A GT200300138 A GT 200300138A GT 200300138 A GT200300138 A GT 200300138A
- Authority
- GT
- Guatemala
- Prior art keywords
- receptor modulators
- glucocorticoid receptor
- compounds
- modulators
- neoplasic
- Prior art date
Links
- 229940117965 Glucocorticoid receptor modulator Drugs 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 208000017701 Endocrine disease Diseases 0.000 abstract 1
- 102000003676 Glucocorticoid Receptors Human genes 0.000 abstract 1
- 108090000079 Glucocorticoid Receptors Proteins 0.000 abstract 1
- 230000002757 inflammatory effect Effects 0.000 abstract 1
- 230000002914 neoplasic effect Effects 0.000 abstract 1
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- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/28—Radicals substituted by singly-bound oxygen or sulphur atoms
- C07D213/30—Oxygen atoms
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- Pyridine Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Steroid Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
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| US11793787B2 (en) | 2019-10-07 | 2023-10-24 | The Broad Institute, Inc. | Methods and compositions for enhancing anti-tumor immunity by targeting steroidogenesis |
| TW202140550A (zh) | 2020-01-29 | 2021-11-01 | 瑞士商諾華公司 | 使用抗tslp抗體治療炎性或阻塞性氣道疾病之方法 |
| WO2021191875A1 (en) | 2020-03-26 | 2021-09-30 | Glaxosmithkline Intellectual Property Development Limited | Cathepsin inhibitors for preventing or treating viral infections |
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| OA11877A (en) * | 1999-04-30 | 2006-03-29 | Pfizer Prod Inc | Glucocorticoid receptor modulators. |
| CO5271670A1 (es) * | 1999-10-29 | 2003-04-30 | Pfizer Prod Inc | Antagonistas del factor de liberacion de corticitropina y composiciones relacionadas |
| IL180679A0 (en) * | 2000-10-27 | 2009-02-11 | Pfizer Prod Inc | Process for the preparation of non-steroidal glucocorticoid receptor modulators |
| JP2002193911A (ja) * | 2000-10-28 | 2002-07-10 | Pfizer Prod Inc | グルココルチコイドレセプターモジュレーター |
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- 2003-06-25 JP JP2004519100A patent/JP4503436B2/ja not_active Expired - Fee Related
- 2003-06-25 CA CA2491994A patent/CA2491994C/en not_active Expired - Fee Related
- 2003-06-25 MX MXPA05000345A patent/MXPA05000345A/es active IP Right Grant
- 2003-06-25 AU AU2003281355A patent/AU2003281355A1/en not_active Abandoned
- 2003-06-25 DK DK03740911.7T patent/DK1521733T3/da active
- 2003-06-25 SI SI200332380T patent/SI1521733T1/sl unknown
- 2003-06-25 BR BR0312575-0A patent/BR0312575A/pt not_active IP Right Cessation
- 2003-06-25 WO PCT/IB2003/002941 patent/WO2004005229A1/en not_active Ceased
- 2003-06-25 ES ES03740911.7T patent/ES2518940T3/es not_active Expired - Lifetime
- 2003-06-25 PT PT37409117T patent/PT1521733E/pt unknown
- 2003-06-25 EP EP03740911.7A patent/EP1521733B1/en not_active Expired - Lifetime
- 2003-07-04 PA PA20038576901A patent/PA8576901A1/es unknown
- 2003-07-04 PE PE2003000681A patent/PE20040650A1/es not_active Application Discontinuation
- 2003-07-07 GT GT200300138A patent/GT200300138A/es unknown
- 2003-07-07 TW TW095116787A patent/TWI340738B/zh not_active IP Right Cessation
- 2003-07-07 UY UY27884A patent/UY27884A1/es not_active Application Discontinuation
- 2003-07-07 TW TW092118479A patent/TWI336323B/zh not_active IP Right Cessation
- 2003-07-07 HN HN2003000207A patent/HN2003000207A/es unknown
- 2003-07-07 AR ARP030102442A patent/AR041186A1/es unknown
- 2003-07-08 MY MYPI20032555A patent/MY135333A/en unknown
- 2003-07-08 US US10/615,126 patent/US7138406B2/en not_active Expired - Lifetime
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2006
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Also Published As
| Publication number | Publication date |
|---|---|
| SI1521733T1 (sl) | 2014-10-30 |
| TW200409749A (en) | 2004-06-16 |
| US20060247264A1 (en) | 2006-11-02 |
| EP1521733A1 (en) | 2005-04-13 |
| US20040138262A1 (en) | 2004-07-15 |
| AU2003281355A1 (en) | 2004-01-23 |
| PE20040650A1 (es) | 2004-09-18 |
| PT1521733E (pt) | 2014-10-29 |
| US7553877B2 (en) | 2009-06-30 |
| ES2518940T3 (es) | 2014-11-06 |
| CA2491994C (en) | 2013-11-05 |
| MY135333A (en) | 2008-03-31 |
| HN2003000207A (es) | 2004-07-27 |
| AR041186A1 (es) | 2005-05-04 |
| CA2491994A1 (en) | 2004-01-15 |
| PA8576901A1 (es) | 2004-03-10 |
| MXPA05000345A (es) | 2005-03-31 |
| BR0312575A (pt) | 2005-05-03 |
| US7138406B2 (en) | 2006-11-21 |
| DK1521733T3 (da) | 2014-10-13 |
| UY27884A1 (es) | 2004-02-27 |
| EP1521733B1 (en) | 2014-08-20 |
| JP2005532389A (ja) | 2005-10-27 |
| TWI340738B (en) | 2011-04-21 |
| WO2004005229A1 (en) | 2004-01-15 |
| TW200628440A (en) | 2006-08-16 |
| TWI336323B (en) | 2011-01-21 |
| JP4503436B2 (ja) | 2010-07-14 |
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