GEP19970948B - Method for Production of Imidazolidine - Google Patents

Method for Production of Imidazolidine

Info

Publication number
GEP19970948B
GEP19970948B GEAP19931536A GEAP1993001536A GEP19970948B GE P19970948 B GEP19970948 B GE P19970948B GE AP19931536 A GEAP19931536 A GE AP19931536A GE AP1993001536 A GEAP1993001536 A GE AP1993001536A GE P19970948 B GEP19970948 B GE P19970948B
Authority
GE
Georgia
Prior art keywords
medium
imidazolidine
production
acid
solvent
Prior art date
Application number
GEAP19931536A
Other languages
English (en)
Inventor
Claude Bonne
Pierre Girault
Jacques Perronnet
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of GEP19970948B publication Critical patent/GEP19970948B/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/72—Two oxygen atoms, e.g. hydantoin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/88—Nitrogen atoms, e.g. allantoin

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Electromechanical Clocks (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
GEAP19931536A 1975-10-29 1993-09-09 Method for Production of Imidazolidine GEP19970948B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7533084A FR2329276A1 (fr) 1975-10-29 1975-10-29 Nouvelles imidazolidines substituees, procede de preparation, application comme medicament et compositions les renfermant

Publications (1)

Publication Number Publication Date
GEP19970948B true GEP19970948B (en) 1997-04-18

Family

ID=9161795

Family Applications (1)

Application Number Title Priority Date Filing Date
GEAP19931536A GEP19970948B (en) 1975-10-29 1993-09-09 Method for Production of Imidazolidine

Country Status (18)

Country Link
US (1) US4097578A (cg-RX-API-DMAC7.html)
JP (1) JPS6011701B2 (cg-RX-API-DMAC7.html)
AU (1) AU500542B2 (cg-RX-API-DMAC7.html)
BE (1) BE847742A (cg-RX-API-DMAC7.html)
BG (1) BG60533B2 (cg-RX-API-DMAC7.html)
CA (1) CA1086751A (cg-RX-API-DMAC7.html)
CH (1) CH599164A5 (cg-RX-API-DMAC7.html)
DE (1) DE2649925C2 (cg-RX-API-DMAC7.html)
DK (1) DK152125C (cg-RX-API-DMAC7.html)
ES (1) ES452746A1 (cg-RX-API-DMAC7.html)
FR (1) FR2329276A1 (cg-RX-API-DMAC7.html)
GB (1) GB1518444A (cg-RX-API-DMAC7.html)
GE (1) GEP19970948B (cg-RX-API-DMAC7.html)
IE (1) IE43875B1 (cg-RX-API-DMAC7.html)
LU (2) LU76085A1 (cg-RX-API-DMAC7.html)
NL (2) NL187102C (cg-RX-API-DMAC7.html)
SE (1) SE430502B (cg-RX-API-DMAC7.html)
SU (1) SU596165A3 (cg-RX-API-DMAC7.html)

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USRE35956E (en) * 1991-01-09 1998-11-10 Roussel Uclaf Phenylimidazolidines having antiandrogenic activity
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FR2725206B1 (fr) * 1994-09-29 1996-12-06 Roussel Uclaf Nouvelles imidazolidines substituees par un heterocycle, leur procede et des intermediaires de preparation, leur application comme medicaments et les compositions pharmaceutiques les renfermant
US5656651A (en) * 1995-06-16 1997-08-12 Biophysica Inc. Androgenic directed compositions
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KR20240096623A (ko) 2017-10-16 2024-06-26 아라곤 파마슈티컬스, 인코포레이티드 비-전이성 거세-저항성 전립선암의 치료를 위한 항-안드로겐
KR20220003554A (ko) 2019-04-19 2022-01-10 리간드 파마슈티칼스 인코포레이티드 화합물의 결정질 형태 및 결정질 형태를 제조하는 방법

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Also Published As

Publication number Publication date
FR2329276B1 (cg-RX-API-DMAC7.html) 1979-09-14
ES452746A1 (es) 1977-10-01
JPS6011701B2 (ja) 1985-03-27
GB1518444A (en) 1978-07-19
NL930079I1 (nl) 1993-09-16
NL930079I2 (nl) 1993-10-01
NL7611576A (nl) 1977-05-03
SE7610859L (sv) 1977-04-30
CA1086751A (fr) 1980-09-30
IE43875L (en) 1977-04-29
AU1909576A (en) 1978-05-04
BE847742A (fr) 1977-04-28
IE43875B1 (en) 1981-06-17
LU76085A1 (cg-RX-API-DMAC7.html) 1977-05-31
SE430502B (sv) 1983-11-21
DK152125B (da) 1988-02-01
NL187102B (nl) 1991-01-02
BG60533B2 (bg) 1995-07-28
JPS5257176A (en) 1977-05-11
DK487476A (da) 1977-04-30
DE2649925A1 (de) 1977-05-12
LU88282I2 (fr) 1994-05-04
FR2329276A1 (fr) 1977-05-27
US4097578A (en) 1978-06-27
DE2649925C2 (de) 1986-08-28
CH599164A5 (cg-RX-API-DMAC7.html) 1978-05-12
SU596165A3 (ru) 1978-02-28
NL187102C (nl) 1991-06-03
AU500542B2 (en) 1979-05-24
DK152125C (da) 1988-06-20

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