GB873049A - Improvements in or relating to penicillin derivatives - Google Patents

Improvements in or relating to penicillin derivatives

Info

Publication number
GB873049A
GB873049A GB31847/58A GB3184758A GB873049A GB 873049 A GB873049 A GB 873049A GB 31847/58 A GB31847/58 A GB 31847/58A GB 3184758 A GB3184758 A GB 3184758A GB 873049 A GB873049 A GB 873049A
Authority
GB
United Kingdom
Prior art keywords
amino
substituted
penicillin
group
acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB31847/58A
Other languages
English (en)
Inventor
Frank Peter Doyle
John Herbert Charles Nayler
Harry Smith
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Beecham Research Laboratories Ltd
Original Assignee
Beecham Research Laboratories Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26251956&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=GB873049(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority to GB31847/58A priority Critical patent/GB873049A/en
Application filed by Beecham Research Laboratories Ltd filed Critical Beecham Research Laboratories Ltd
Priority to ES0252422A priority patent/ES252422A1/es
Priority to FR806723A priority patent/FR246M/fr
Priority to NO133325A priority patent/NO115737B/no
Priority to CH7907859A priority patent/CH387635A/de
Priority to DK356359AA priority patent/DK126118B/da
Priority to CH638961A priority patent/CH407126A/de
Priority to FR863883A priority patent/FR12F/fr
Publication of GB873049A publication Critical patent/GB873049A/en
Priority to CY24262A priority patent/CY242A/xx
Priority to GB4154162A priority patent/GB978178A/en
Priority to MY6200044A priority patent/MY6200044A/xx
Priority to OA50915A priority patent/OA00880A/xx
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/44—Compounds with an amino radical acylated by carboxylic acids, attached in position 6
    • C07D499/48—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical
    • C07D499/58—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical
    • C07D499/64—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by nitrogen atoms
    • C07D499/68—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by nitrogen atoms with aromatic rings as additional substituents on the carbon chain
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/44—Compounds with an amino radical acylated by carboxylic acids, attached in position 6
    • C07D499/48—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
GB31847/58A 1958-10-06 1958-10-06 Improvements in or relating to penicillin derivatives Expired GB873049A (en)

Priority Applications (12)

Application Number Priority Date Filing Date Title
GB31847/58A GB873049A (en) 1958-10-06 1958-10-06 Improvements in or relating to penicillin derivatives
ES0252422A ES252422A1 (es) 1958-10-06 1959-10-02 Proceso para la preparaciën de derivados penicilinicos de la fërmula general:
FR806723A FR246M (xx) 1958-10-06 1959-10-05
NO133325A NO115737B (xx) 1958-10-06 1959-10-05
CH7907859A CH387635A (de) 1958-10-06 1959-10-06 Verfahren zur Herstellung von Penicillinen
DK356359AA DK126118B (da) 1958-10-06 1959-10-06 Fremgangsmåde til fremstilling af 6-aminopenicillansyrederivater eller salte deraf.
CH638961A CH407126A (de) 1958-10-06 1961-06-01 Verfahren zur Herstellung von epimeren a-Amino-benzylpenicillinen
FR863883A FR12F (fr) 1958-10-06 1961-06-05 Dérivés de la pénicilline et leur procédé de préparation.
CY24262A CY242A (en) 1958-10-06 1962-07-03 Improvements in or relating to penicillin derivatives
GB4154162A GB978178A (en) 1958-10-06 1962-11-02 Penicillins
MY6200044A MY6200044A (en) 1958-10-06 1962-12-31 Improvements in or relating to penicillin derivatives
OA50915A OA00880A (fr) 1958-10-06 1964-12-18 Dérivés de la pénicélline et leur procédé de préparation.

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB31847/58A GB873049A (en) 1958-10-06 1958-10-06 Improvements in or relating to penicillin derivatives
GB1630359 1959-05-12

Publications (1)

Publication Number Publication Date
GB873049A true GB873049A (en) 1961-07-19

Family

ID=26251956

Family Applications (1)

Application Number Title Priority Date Filing Date
GB31847/58A Expired GB873049A (en) 1958-10-06 1958-10-06 Improvements in or relating to penicillin derivatives

Country Status (8)

Country Link
CH (1) CH387635A (xx)
CY (1) CY242A (xx)
DK (1) DK126118B (xx)
ES (1) ES252422A1 (xx)
FR (1) FR246M (xx)
GB (1) GB873049A (xx)
NO (1) NO115737B (xx)
OA (1) OA00880A (xx)

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK104060C (da) * 1962-08-18 1966-03-28 Beecham Res Lab Fremgangsmåde til fremstilling af α-aminobenzylpenicillin eller salte deraf.
US3245984A (en) * 1961-09-26 1966-04-12 Lepetit Spa Amino-alpha-phenylalkyl penicillins
DE1296142B (de) * 1962-01-29 1969-05-29 Bristol Myers Co Verfahren zur Herstellung von ª‡-Aminobenzylpenicillin
EP0477639A1 (de) * 1990-09-22 1992-04-01 Bayer Ag Substituierte Aminosäureamid-Derivate deren Herstellung und Verwendung
US5158962A (en) * 1989-11-01 1992-10-27 Bayer Aktiengesellschaft Fungicidal substituted amino acid amides
US5723646A (en) * 1991-01-24 1998-03-03 Bayer Aktiengesellschaft Substituted amino acid amide derivatives their preparation and use as fungicides

Cited By (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3245984A (en) * 1961-09-26 1966-04-12 Lepetit Spa Amino-alpha-phenylalkyl penicillins
DE1296142B (de) * 1962-01-29 1969-05-29 Bristol Myers Co Verfahren zur Herstellung von ª‡-Aminobenzylpenicillin
DK104060C (da) * 1962-08-18 1966-03-28 Beecham Res Lab Fremgangsmåde til fremstilling af α-aminobenzylpenicillin eller salte deraf.
US5158962A (en) * 1989-11-01 1992-10-27 Bayer Aktiengesellschaft Fungicidal substituted amino acid amides
EP0477639A1 (de) * 1990-09-22 1992-04-01 Bayer Ag Substituierte Aminosäureamid-Derivate deren Herstellung und Verwendung
US5723646A (en) * 1991-01-24 1998-03-03 Bayer Aktiengesellschaft Substituted amino acid amide derivatives their preparation and use as fungicides
US5942541A (en) * 1991-01-24 1999-08-24 Bayer Aktiengesellschaft Substituted amino acid amide derivatives their preparation and use as fungicides

Also Published As

Publication number Publication date
OA00880A (fr) 1968-03-22
CY242A (en) 1962-07-03
ES252422A1 (es) 1960-01-01
NO115737B (xx) 1968-11-25
CH387635A (de) 1965-02-15
FR246M (xx) 1900-01-01
DK126118B (da) 1973-06-12

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