GB2045755B - Process and intermediates for penicillanic acid 1,1-dioxide and esters thereof - Google Patents

Process and intermediates for penicillanic acid 1,1-dioxide and esters thereof

Info

Publication number
GB2045755B
GB2045755B GB8007122A GB8007122A GB2045755B GB 2045755 B GB2045755 B GB 2045755B GB 8007122 A GB8007122 A GB 8007122A GB 8007122 A GB8007122 A GB 8007122A GB 2045755 B GB2045755 B GB 2045755B
Authority
GB
United Kingdom
Prior art keywords
intermediates
esters
dioxide
penicillanic acid
penicillanic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB8007122A
Other languages
English (en)
Other versions
GB2045755A (en
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc filed Critical Pfizer Inc
Publication of GB2045755A publication Critical patent/GB2045755A/en
Application granted granted Critical
Publication of GB2045755B publication Critical patent/GB2045755B/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Cosmetics (AREA)
GB8007122A 1979-03-05 1980-03-03 Process and intermediates for penicillanic acid 1,1-dioxide and esters thereof Expired GB2045755B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US1781079A 1979-03-05 1979-03-05
US1780879A 1979-03-05 1979-03-05

Publications (2)

Publication Number Publication Date
GB2045755A GB2045755A (en) 1980-11-05
GB2045755B true GB2045755B (en) 1983-01-26

Family

ID=26690337

Family Applications (1)

Application Number Title Priority Date Filing Date
GB8007122A Expired GB2045755B (en) 1979-03-05 1980-03-03 Process and intermediates for penicillanic acid 1,1-dioxide and esters thereof

Country Status (36)

Country Link
KR (1) KR850001339B1 (nl)
AR (1) AR225031A1 (nl)
AT (1) AT366693B (nl)
AU (1) AU522572B2 (nl)
BG (1) BG33292A3 (nl)
CH (1) CH644608A5 (nl)
CS (1) CS215130B2 (nl)
DD (1) DD149367A5 (nl)
DE (1) DE3008257C2 (nl)
DK (2) DK159852C (nl)
EG (1) EG14437A (nl)
ES (1) ES489185A0 (nl)
FI (1) FI70024C (nl)
FR (1) FR2450836B1 (nl)
GB (1) GB2045755B (nl)
GR (1) GR67234B (nl)
HK (1) HK66587A (nl)
HU (1) HU186304B (nl)
IE (1) IE49535B1 (nl)
IL (1) IL59515A (nl)
IN (1) IN153685B (nl)
IT (1) IT1130300B (nl)
KE (1) KE3464A (nl)
LU (1) LU82215A1 (nl)
MX (1) MX6032E (nl)
MY (1) MY8500319A (nl)
NL (1) NL180317C (nl)
NO (2) NO800618L (nl)
PL (1) PL125197B1 (nl)
PT (1) PT70897A (nl)
RO (1) RO80112A (nl)
SE (2) SE449103B (nl)
SG (1) SG55884G (nl)
SU (1) SU1192626A3 (nl)
UA (1) UA6342A1 (nl)
YU (1) YU42328B (nl)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4419284A (en) * 1981-03-23 1983-12-06 Pfizer Inc. Preparation of halomethyl esters (and related esters) of penicillanic acid 1,1-dioxide
IN159362B (nl) * 1981-03-23 1987-05-09 Pfizer
PT76527B (en) * 1982-04-19 1985-12-09 Gist Brocades Nv A process for the preparation of penicillanic acid 1,1-dioxide and derivatives thereof
IT1190897B (it) * 1982-06-29 1988-02-24 Opos Biochimica Srl Procedimento per la preparazione dell'estere 1-etossicarbonilossietilico dell'acido 6-(d(-)-alfa aminoalfa fenilacetamido)-penicillanico
US4606865A (en) * 1982-09-20 1986-08-19 Astra Lakemedel Aktiebolag Methods for the preparation of α-bromodiethylcarbonate
EP0139047A1 (en) * 1983-10-18 1985-05-02 Gist-Brocades N.V. Process for the preparation of 6,6-dibromopenicillanic acid 1,1-dioxide
EP0139048A1 (en) * 1983-10-18 1985-05-02 Gist-Brocades N.V. Process for the dehalogenation of 6,6-dibromopenicillanic acid 1,1-dioxide
US4596677A (en) * 1984-04-06 1986-06-24 Bristol-Myers Company Anhydropenicillin intermediates

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IN149747B (nl) * 1977-06-07 1982-04-03 Pfizer
CA1158639A (en) * 1978-12-11 1983-12-13 Eric M. Gordon 6-bromopenicillanic acid sulfone
DE3068390D1 (en) * 1979-01-10 1984-08-09 Beecham Group Plc Penicillin derivatives, process for their preparation and pharmaceutical compositions containing certain of these compounds
IE49881B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd B-lactam intermediates

Also Published As

Publication number Publication date
DE3008257A1 (de) 1980-09-11
YU42328B (en) 1988-08-31
FR2450836A1 (fr) 1980-10-03
AU5610480A (en) 1980-09-11
ES8103094A1 (es) 1981-02-16
FR2450836B1 (fr) 1986-03-21
FI800661A (fi) 1980-09-06
PT70897A (en) 1980-04-01
ATA119080A (de) 1981-09-15
SE449103B (sv) 1987-04-06
GB2045755A (en) 1980-11-05
DK159852C (da) 1991-05-06
DD149367A5 (de) 1981-07-08
ES489185A0 (es) 1981-02-16
DK145690D0 (da) 1990-06-14
SU1192626A3 (ru) 1985-11-15
BG33292A3 (en) 1983-01-14
IE800429L (en) 1980-09-05
DK145690A (da) 1990-06-14
PL125197B1 (en) 1983-04-30
UA6342A1 (uk) 1994-12-29
IT8020367A0 (it) 1980-03-05
IT1130300B (it) 1986-06-11
FI70024B (fi) 1986-01-31
KE3464A (en) 1984-10-12
MY8500319A (en) 1985-12-31
PL222448A1 (nl) 1981-01-02
FI70024C (fi) 1986-09-12
AR225031A1 (es) 1982-02-15
NL180317B (nl) 1986-09-01
MX6032E (es) 1984-10-04
CS215130B2 (en) 1982-07-30
KR850001339B1 (ko) 1985-09-19
AU522572B2 (en) 1982-06-17
IL59515A (en) 1983-02-23
SG55884G (en) 1985-03-08
IN153685B (nl) 1984-08-04
DK92680A (da) 1980-09-06
DE3008257C2 (de) 1984-03-01
GR67234B (nl) 1981-06-25
EG14437A (en) 1984-09-30
NL8001285A (nl) 1980-09-09
SE8603309L (sv) 1986-08-04
YU58580A (en) 1983-02-28
IE49535B1 (en) 1985-10-16
AT366693B (de) 1982-04-26
IL59515A0 (en) 1980-06-30
DK166353C (da) 1993-09-06
HK66587A (en) 1987-09-25
DK159852B (da) 1990-12-17
HU186304B (en) 1985-07-29
RO80112A (ro) 1982-10-26
SE8000512L (sv) 1980-09-06
LU82215A1 (fr) 1980-09-24
NL180317C (nl) 1987-02-02
NO823127L (no) 1980-09-08
DK166353B (da) 1993-04-13
CH644608A5 (de) 1984-08-15
NO800618L (no) 1980-09-08
SE8603309D0 (sv) 1986-08-04

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Legal Events

Date Code Title Description
PE20 Patent expired after termination of 20 years

Effective date: 20000302