GB0229804D0 - Avermection b1 and avermectin b1 monosaccharide derivatives having an alkoxymethyl substituent in the 4"- or 4'-position - Google Patents

Avermection b1 and avermectin b1 monosaccharide derivatives having an alkoxymethyl substituent in the 4"- or 4'-position

Info

Publication number
GB0229804D0
GB0229804D0 GBGB0229804.0A GB0229804A GB0229804D0 GB 0229804 D0 GB0229804 D0 GB 0229804D0 GB 0229804 A GB0229804 A GB 0229804A GB 0229804 D0 GB0229804 D0 GB 0229804D0
Authority
GB
United Kingdom
Prior art keywords
avermection
avermectin
monosaccharide derivatives
alkoxymethyl substituent
alkoxymethyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
GBGB0229804.0A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Syngenta Participations AG
Original Assignee
Syngenta Participations AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Participations AG filed Critical Syngenta Participations AG
Priority to GBGB0229804.0A priority Critical patent/GB0229804D0/en
Publication of GB0229804D0 publication Critical patent/GB0229804D0/en
Priority to PE2003001284A priority patent/PE20040713A1/es
Priority to ARP030104712A priority patent/AR042533A1/es
Priority to TW092135927A priority patent/TW200512214A/zh
Priority to PCT/EP2003/014613 priority patent/WO2004056844A1/en
Priority to CA2507774A priority patent/CA2507774C/en
Priority to AU2003302284A priority patent/AU2003302284B2/en
Priority to JP2004561378A priority patent/JP4851094B2/ja
Priority to BR0317601-0A priority patent/BR0317601A/pt
Priority to MXPA05006036A priority patent/MXPA05006036A/es
Priority to UAA200507209A priority patent/UA81281C2/uk
Priority to US10/539,274 priority patent/US7737261B2/en
Priority to KR1020057011622A priority patent/KR101109500B1/ko
Priority to EP03810843.7A priority patent/EP1581546B1/en
Priority to CN2003801088575A priority patent/CN1738828B/zh
Priority to RU2005122943/04A priority patent/RU2330857C2/ru
Priority to PL377497A priority patent/PL211483B1/pl
Priority to ES03810843T priority patent/ES2742899T3/es
Priority to IL169092A priority patent/IL169092A/en
Priority to MA28349A priority patent/MA27646A1/fr
Priority to CO05059203A priority patent/CO5690647A1/es
Priority to ZA200504353A priority patent/ZA200504353B/en
Priority to US12/768,280 priority patent/US8017589B2/en
Priority to JP2010286151A priority patent/JP5302297B2/ja
Priority to US13/117,292 priority patent/US8263566B2/en
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/02—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms
    • A01N43/04—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom
    • A01N43/22—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom rings with more than six members
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Molecular Biology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Plural Heterocyclic Compounds (AREA)
GBGB0229804.0A 2002-12-20 2002-12-20 Avermection b1 and avermectin b1 monosaccharide derivatives having an alkoxymethyl substituent in the 4"- or 4'-position Ceased GB0229804D0 (en)

Priority Applications (25)

Application Number Priority Date Filing Date Title
GBGB0229804.0A GB0229804D0 (en) 2002-12-20 2002-12-20 Avermection b1 and avermectin b1 monosaccharide derivatives having an alkoxymethyl substituent in the 4"- or 4'-position
PE2003001284A PE20040713A1 (es) 2002-12-20 2003-12-12 Avermectina b1 y derivados de monosacaridos de avermectina b1 que tienen un sustituyente alcoximetilo en la posicion 4" o 4'
ARP030104712A AR042533A1 (es) 2002-12-20 2003-12-18 Avermectina b1 y derivados de monosacaridos de avermectina b1 que tienen un sustituyente alcoximetilo en la posicion 4' ' o 4'
TW092135927A TW200512214A (en) 2002-12-20 2003-12-18 Avermectin B1 and avermectin B1 monosaccharide derivatives having an alkoxymethyl substituent in the 4"-or 4'-position
ES03810843T ES2742899T3 (es) 2002-12-20 2003-12-19 Derivados de avermectina B1 que tienen un sustituyente alcoximetilo en la posición 4'' o 4'
KR1020057011622A KR101109500B1 (ko) 2002-12-20 2003-12-19 4″- 또는 4′-위치에 알콕시메틸 치환체를 갖는 아버멕틴ｂ1 및 아버멕틴 ｂ1 모노사카라이드 유도체
RU2005122943/04A RU2330857C2 (ru) 2002-12-20 2003-12-19 Производные авермектина в1 и моносахарида авермектина в1, имеющие алкоксиметильный заместитель в положении 4"- или 4'-
AU2003302284A AU2003302284B2 (en) 2002-12-20 2003-12-19 Avermectin B1 and avermectin B1 monosaccharide derivatives having an alkoxymethyl substituent in the 4"- or 4'-position
JP2004561378A JP4851094B2 (ja) 2002-12-20 2003-12-19 アベルメクチンｂ１及び４”位又は４’−位にアルコキシメチル置換基を有するアベルメクチンｂ１モノサッカライド誘導体
BR0317601-0A BR0317601A (pt) 2002-12-20 2003-12-19 Avermectina b1 e derivados de monossacarìdeos da avermectina b1 que possuem um substituinte na posição 4" ou 4'''
MXPA05006036A MXPA05006036A (es) 2002-12-20 2003-12-19 Derivados de avermectina b1 y monosacarido de avermectina b1 que tienen un sustituyente de alcoximetilo en la posicion 4" o 4'.
UAA200507209A UA81281C2 (en) 2002-12-20 2003-12-19 Avermectin derivatives, pesticide composition and method of pest control
US10/539,274 US7737261B2 (en) 2002-12-20 2003-12-19 Avermectin B1 and avermectin B1 monosaccharide derivatives having an alkoxymethyl substituent in the 4″ -or 4′-position
PCT/EP2003/014613 WO2004056844A1 (en) 2002-12-20 2003-12-19 Avermectin b1 and avermectin b1 monosaccharide derivatives having an alkoxymethyl substituent in the 4”- or 4’-position
EP03810843.7A EP1581546B1 (en) 2002-12-20 2003-12-19 Avermectin b1 derivatives having an alkoxymethyl substituent in the 4''- or 4'-position
CN2003801088575A CN1738828B (zh) 2002-12-20 2003-12-19 在4"-或4′-位上有烷氧基甲基取代基的阿维菌素b1和阿维菌素b1单糖衍生物
CA2507774A CA2507774C (en) 2002-12-20 2003-12-19 Avermectin b1 and avermectin b1 monosaccharide derivatives having an alkoxymethyl substituent in the 4"- or 4'-position
PL377497A PL211483B1 (pl) 2002-12-20 2003-12-19 Awermektyna B1 i jej pochodne monosacharydowe, środek do zwalczania szkodników, sposób zwalczania szkodników i zastosowanie kompozycji
IL169092A IL169092A (en) 2002-12-20 2005-06-09 Avermectin b1 derivatives having an alkoxymethyl substituent in the 4" - or 4'-position, use thereof in the preparation of pesticides and pesticides comprising the same
MA28349A MA27646A1 (fr) 2002-12-20 2005-06-17 Derives d'avermectine b1 et d'avermectine b1 monosaccharidique ayant un substituant alcoxymethyle en position 4" ou 4'
CO05059203A CO5690647A1 (es) 2002-12-20 2005-06-17 Avermectina b1 y sus derivados de monosacaridos de avermecti na b1 que tienen un sustituyente alcoximetilo en la posicion 4´ o 4´
ZA200504353A ZA200504353B (en) 2002-12-20 2006-01-06 Avermectin B1 and Avermectin B1 monosaccharide derivatives having an alkoxymethyl substituent in the 4"- or 4'-position
US12/768,280 US8017589B2 (en) 2002-12-20 2010-04-27 Avermectin B1 and avermectin B1 monosaccharide derivatives having an alkoxymethyl substituent in the 4″-or 4′-position
JP2010286151A JP5302297B2 (ja) 2002-12-20 2010-12-22 ４”位又は４’−位にアルコキシメチル置換基を有するアベルメクチンｂ１及びアベルメクチンｂ１単糖誘導体
US13/117,292 US8263566B2 (en) 2002-12-20 2011-05-27 Avermectin B1 and avermectin B1 monosaccharide derivatives having an alkoxymethyl substituent in the 4″-or 4′-position

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0229804.0A GB0229804D0 (en) 2002-12-20 2002-12-20 Avermection b1 and avermectin b1 monosaccharide derivatives having an alkoxymethyl substituent in the 4"- or 4'-position

Publications (1)

Publication Number Publication Date
GB0229804D0 true GB0229804D0 (en) 2003-01-29

Family

ID=9950151

Family Applications (1)

Application Number Title Priority Date Filing Date
GBGB0229804.0A Ceased GB0229804D0 (en) 2002-12-20 2002-12-20 Avermection b1 and avermectin b1 monosaccharide derivatives having an alkoxymethyl substituent in the 4"- or 4'-position

Country Status (22)

Country Link
US (3) US7737261B2 (https=)
EP (1) EP1581546B1 (https=)
JP (2) JP4851094B2 (https=)
KR (1) KR101109500B1 (https=)
CN (1) CN1738828B (https=)
AR (1) AR042533A1 (https=)
AU (1) AU2003302284B2 (https=)
BR (1) BR0317601A (https=)
CA (1) CA2507774C (https=)
CO (1) CO5690647A1 (https=)
ES (1) ES2742899T3 (https=)
GB (1) GB0229804D0 (https=)
IL (1) IL169092A (https=)
MA (1) MA27646A1 (https=)
MX (1) MXPA05006036A (https=)
PE (1) PE20040713A1 (https=)
PL (1) PL211483B1 (https=)
RU (1) RU2330857C2 (https=)
TW (1) TW200512214A (https=)
UA (1) UA81281C2 (https=)
WO (1) WO2004056844A1 (https=)
ZA (1) ZA200504353B (https=)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0229804D0 (en) * 2002-12-20 2003-01-29 Syngenta Participations Ag Avermection b1 and avermectin b1 monosaccharide derivatives having an alkoxymethyl substituent in the 4"- or 4'-position
JP2010006703A (ja) * 2006-11-07 2010-01-14 Hokko Chem Ind Co Ltd アベルメクチンモノ配糖体誘導体
RU2453553C1 (ru) * 2011-05-11 2012-06-20 Игорь Викторович Заварзин 5-о-сукциноилавермектин, способ его получения и антипаразитарное средство на его основе
RU2472801C1 (ru) * 2011-05-11 2013-01-20 Игорь Викторович Заварзин 5-о-производные авермектина, способ их получения и антипаразитарные средства на их основе
CN103613625B (zh) * 2013-12-02 2016-03-02 兰州大学 一种阿维菌素类化合物及其制备方法和在农药中的用途
CN104402953B (zh) * 2014-11-28 2017-07-28 大庆志飞生物化工有限公司 阿维菌素单糖化合物及其制备方法和用途
CN104402954A (zh) * 2014-11-28 2015-03-11 大庆志飞生物化工有限公司 甲胺基阿维菌素单糖化合物及其制备方法和用途
JP6577184B2 (ja) 2014-12-24 2019-09-18 Ntn株式会社 転がり軸受
CN107501368B (zh) * 2017-09-30 2020-02-21 中国科学院成都生物研究所 一种多拉菌素衍生物的合成及其杀虫应用
CN113150053B (zh) * 2020-01-22 2024-10-01 华东理工大学 偶氮苯类阿维菌素衍生物及其制备方法和应用
CN113817008B (zh) * 2021-07-15 2023-05-23 湖州师范学院 新型琥珀酰基十六元大环内酯的制备方法及用途

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US87519A (en) * 1869-03-02 Improvement in furnace-stoves and registers
US18993A (en) * 1857-12-29 Cider-mill
US148520A (en) * 1874-03-10 Improvement in faucets
SE434277B (sv) 1976-04-19 1984-07-16 Merck & Co Inc Sett att framstella nya antihelmintiskt verkande foreningar genom odling av streptomyces avermitilis
US4874749A (en) * 1987-07-31 1989-10-17 Merck & Co., Inc. 4"-Deoxy-4-N-methylamino avermectin Bla/Blb
GB8811037D0 (en) 1988-05-10 1988-06-15 Glaxo Group Ltd Chemical compounds
EP0353959A2 (en) 1988-08-02 1990-02-07 Beecham Group Plc Antihelmintic macrolide antibiotics
SE465605B (sv) * 1990-02-26 1991-10-07 Harry Nilsson Skivfilter
JP2622197B2 (ja) 1990-03-01 1997-06-18 三共株式会社 １３−エーテル置換ミルベマイシン誘導体
US5169839A (en) * 1990-05-11 1992-12-08 Merck & Co., Inc. Derivatives of 3'- and 3"-o-desmethyl avermectin compounds, compositions and methods of treating melmintic and parasitic infections
US5262400A (en) * 1991-06-20 1993-11-16 Merck & Co., Inc. 4α-substituted avermectin derivatives
US5411737A (en) 1991-10-15 1995-05-02 Merck & Co., Inc. Slow release syneresing polymeric drug delivery device
US5602107A (en) 1993-05-10 1997-02-11 Merck & Co., Inc. Pour-on formulations consisting of gylcols, glycerides and avermectin compounds
PL174488B1 (pl) 1993-05-10 1998-08-31 Merck & Co Inc Preparat do zwalczania pasożytów zwierząt oraz sposób wytwarzania preparatu do zwalczania pasożytów zwierząt
CA2168843C (en) * 1993-08-19 2004-10-19 Raymond Cvetovich Thermodynamically stable crystal form of 4"-deoxy-4"-epi-methylamino avermectin b1a/b1b benzoic acid salt and processes for its preparation
US5436355A (en) 1994-02-03 1995-07-25 Merck & Co., Inc. Process for making avermectin/zein compositions
TW327125B (en) 1994-02-07 1998-02-21 Merck & Co Inc Composition and method for protecting against pine exhausted
WO2002012248A1 (en) 2000-08-09 2002-02-14 The Kitasato Institute Avermectin derivatives
JPWO2002012261A1 (ja) 2000-08-09 2004-01-15 社団法人北里研究所 エバーメクチン誘導体
EP1483580A4 (en) * 2002-03-05 2006-10-11 Merck & Co Inc BIOMARKERS FOR THE EFFICACY OF APPETIZERS
GB0229804D0 (en) 2002-12-20 2003-01-29 Syngenta Participations Ag Avermection b1 and avermectin b1 monosaccharide derivatives having an alkoxymethyl substituent in the 4"- or 4'-position

Also Published As

Publication number Publication date
MA27646A1 (fr) 2005-12-01
US7737261B2 (en) 2010-06-15
IL169092A0 (en) 2007-07-04
IL169092A (en) 2010-12-30
AU2003302284B2 (en) 2009-07-23
US20100210574A1 (en) 2010-08-19
US8263566B2 (en) 2012-09-11
KR101109500B1 (ko) 2012-01-31
CA2507774C (en) 2011-06-14
RU2330857C2 (ru) 2008-08-10
WO2004056844A1 (en) 2004-07-08
PE20040713A1 (es) 2004-12-02
PL377497A1 (pl) 2006-02-06
RU2005122943A (ru) 2006-01-20
JP2011102303A (ja) 2011-05-26
CN1738828A (zh) 2006-02-22
AU2003302284A1 (en) 2004-07-14
UA81281C2 (en) 2007-12-25
US20110230429A1 (en) 2011-09-22
US20060148729A1 (en) 2006-07-06
EP1581546A1 (en) 2005-10-05
CN1738828B (zh) 2012-09-05
JP4851094B2 (ja) 2012-01-11
JP5302297B2 (ja) 2013-10-02
CA2507774A1 (en) 2004-07-08
US8017589B2 (en) 2011-09-13
TW200512214A (en) 2005-04-01
AR042533A1 (es) 2005-06-22
EP1581546B1 (en) 2019-03-20
ZA200504353B (en) 2006-03-29
JP2006515849A (ja) 2006-06-08
KR20050088133A (ko) 2005-09-01
PL211483B1 (pl) 2012-05-31
CO5690647A1 (es) 2006-10-31
ES2742899T3 (es) 2020-02-17
MXPA05006036A (es) 2005-08-18
BR0317601A (pt) 2005-11-29

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Legal Events

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