FR2699921B1 - Dérivés d'acide 2-(thien-2-yl)imidazo[2,1-b]benzothiazole-3-acétique, leur préparation et leur application en thérapeutique. - Google Patents

Dérivés d'acide 2-(thien-2-yl)imidazo[2,1-b]benzothiazole-3-acétique, leur préparation et leur application en thérapeutique.

Info

Publication number
FR2699921B1
FR2699921B1 FR9215889A FR9215889A FR2699921B1 FR 2699921 B1 FR2699921 B1 FR 2699921B1 FR 9215889 A FR9215889 A FR 9215889A FR 9215889 A FR9215889 A FR 9215889A FR 2699921 B1 FR2699921 B1 FR 2699921B1
Authority
FR
France
Prior art keywords
thien
imidazo
benzothiazole
preparation
acetic acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR9215889A
Other languages
English (en)
French (fr)
Other versions
FR2699921A1 (fr
Inventor
Mireille Sevrin
Claude Morel
Pascal George
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Synthelabo SA
Original Assignee
Synthelabo SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo SA filed Critical Synthelabo SA
Priority to FR9215889A priority Critical patent/FR2699921B1/fr
Priority to EP93403137A priority patent/EP0605295A1/fr
Priority to NZ250579A priority patent/NZ250579A/en
Priority to JP5335081A priority patent/JPH06234770A/ja
Priority to US08/175,249 priority patent/US5418248A/en
Priority to PL93301680A priority patent/PL301680A1/xx
Priority to SK1493-93A priority patent/SK149393A3/sk
Priority to CA002112555A priority patent/CA2112555A1/en
Priority to NO934881A priority patent/NO934881L/no
Priority to ZA939760A priority patent/ZA939760B/xx
Priority to FI935915A priority patent/FI935915L/fi
Priority to CZ932918A priority patent/CZ282959B6/cs
Priority to HU9303785A priority patent/HUT70409A/hu
Priority to CN93121519A priority patent/CN1036009C/zh
Priority to TW082111123A priority patent/TW257764B/zh
Priority to KR1019930030792A priority patent/KR0140846B1/ko
Priority to IL108225A priority patent/IL108225A/xx
Priority to AU52762/93A priority patent/AU666790B2/en
Publication of FR2699921A1 publication Critical patent/FR2699921A1/fr
Application granted granted Critical
Publication of FR2699921B1 publication Critical patent/FR2699921B1/fr
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Neurosurgery (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Weting (AREA)
  • Diffracting Gratings Or Hologram Optical Elements (AREA)
FR9215889A 1992-12-30 1992-12-30 Dérivés d'acide 2-(thien-2-yl)imidazo[2,1-b]benzothiazole-3-acétique, leur préparation et leur application en thérapeutique. Expired - Fee Related FR2699921B1 (fr)

Priority Applications (18)

Application Number Priority Date Filing Date Title
FR9215889A FR2699921B1 (fr) 1992-12-30 1992-12-30 Dérivés d'acide 2-(thien-2-yl)imidazo[2,1-b]benzothiazole-3-acétique, leur préparation et leur application en thérapeutique.
EP93403137A EP0605295A1 (fr) 1992-12-30 1993-12-22 Dérivés d'acide 2-thiénylimidazo 2,1-b benzothiazole-3-acétique, leur préparation et leur application en thérapeutique
NZ250579A NZ250579A (en) 1992-12-30 1993-12-23 2-thienylimidazo[2,1-b]benzothiazole-3-acetic acid derivatives, preparation and pharmaceutical compositions thereof
JP5335081A JPH06234770A (ja) 1992-12-30 1993-12-28 ２−チエニルイミダゾ［２，１−ｂ］ベンゾチアゾール−３−酢酸誘導体、それらの製造および医療への応用
CN93121519A CN1036009C (zh) 1992-12-30 1993-12-29 2-噻吩基咪唑并[2，1-b]苯并噻唑-3-乙酸衍生物，其制备方法及其药用
SK1493-93A SK149393A3 (en) 1992-12-30 1993-12-29 2-thienylmidazo/2,1-b/benzothiazole-3-acetic acid derivatives, method of their preparation and their therapeutical using
CA002112555A CA2112555A1 (en) 1992-12-30 1993-12-29 2-thienylimidazo[2,1-b]benzothiazole-3-acetic acid derivatives, their preparation and their use
NO934881A NO934881L (no) 1992-12-30 1993-12-29 Benzotiazolderivater, fremgangsmåte for deres fremstilling og farmasöytisk preparat derav
ZA939760A ZA939760B (en) 1992-12-30 1993-12-29 2-Thienylimidazo(2,1-b)benzothiazole-3-acetic acid derivatives their preparation and their use
FI935915A FI935915L (fi) 1992-12-30 1993-12-29 2-tienyyli-imidatso(2,1-b)bentsotiatsol-3-etikkahappojohdannaiset, niiden valmistus ja terapeuttinen käyttö
US08/175,249 US5418248A (en) 1992-12-30 1993-12-29 2-thienylimidazo[2,1-β]benzothiazole-3-acetic acid derivatives, their preparation and their use
HU9303785A HUT70409A (en) 1992-12-30 1993-12-29 2-thienyl-imidazo[2,1-b]benzothiazol-3-acetic acid derivatives, pharmaceutical compositions containing them and process for preparing them
PL93301680A PL301680A1 (en) 1992-12-30 1993-12-29 Derivatives of 2-thienyl imidazo/2,1-b/benzothiazol-3-acetic acid, their production and application in therapy
TW082111123A TW257764B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1992-12-30 1993-12-29
KR1019930030792A KR0140846B1 (ko) 1992-12-30 1993-12-29 레이저 다이오드의 그레이팅 형성을 위한 습식 식각 방법
IL108225A IL108225A (en) 1992-12-30 1993-12-29 2-THIENYLIMIDAZO £2, 1-b| BENZOTHIAZOLE-3-ACETIC ACID DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
CZ932918A CZ282959B6 (cs) 1992-12-30 1993-12-29 Derivát kyseliny 2-thienylimidazo/2,1-b/benzothiazol-3-octové, způsob jeho přípravy a farmaceutický přípravek tento derivát obsahující
AU52762/93A AU666790B2 (en) 1992-12-30 1993-12-30 2-Thienylimidazo(2,1-b)benzothiazole-3-acetic acid derivatives, their preparation and their use

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9215889A FR2699921B1 (fr) 1992-12-30 1992-12-30 Dérivés d'acide 2-(thien-2-yl)imidazo[2,1-b]benzothiazole-3-acétique, leur préparation et leur application en thérapeutique.

Publications (2)

Publication Number Publication Date
FR2699921A1 FR2699921A1 (fr) 1994-07-01
FR2699921B1 true FR2699921B1 (fr) 1995-02-10

Family

ID=9437257

Family Applications (1)

Application Number Title Priority Date Filing Date
FR9215889A Expired - Fee Related FR2699921B1 (fr) 1992-12-30 1992-12-30 Dérivés d'acide 2-(thien-2-yl)imidazo[2,1-b]benzothiazole-3-acétique, leur préparation et leur application en thérapeutique.

Country Status (18)

Country Link
US (1) US5418248A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
EP (1) EP0605295A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
JP (1) JPH06234770A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
KR (1) KR0140846B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CN (1) CN1036009C (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
AU (1) AU666790B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CA (1) CA2112555A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CZ (1) CZ282959B6 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
FI (1) FI935915L (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
FR (1) FR2699921B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
HU (1) HUT70409A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IL (1) IL108225A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NO (1) NO934881L (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NZ (1) NZ250579A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
PL (1) PL301680A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
SK (1) SK149393A3 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
TW (1) TW257764B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
ZA (1) ZA939760B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU3783497A (en) * 1996-08-09 1998-03-06 Yamanouchi Pharmaceutical Co., Ltd. Metabotropic glutamate receptor agonists
EP2218464A1 (en) * 2009-02-11 2010-08-18 Technische Universität München Compounds for non-invasive measurement of aggregates of amyloid peptides

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8724566D0 (en) * 1987-10-20 1987-11-25 Roussel Lab Ltd Chemical compounds
US4896863A (en) * 1988-05-26 1990-01-30 Tim Riplinger System having material dispensing and wind up device with guide
JP2726999B2 (ja) * 1988-06-22 1998-03-11 日研化学株式会社 イミダゾ［２，１−ｂ］ベンゾチアゾール誘導体及び該化合物を有効成分とする抗潰瘍剤
EP0524055A1 (fr) * 1991-07-19 1993-01-20 Synthelabo Dérivés d'imidazo[2,1-b]benzothiazole-3-acétamide, leur préparation et leur application en thérapeutique
DK0630376T3 (da) * 1992-03-12 1999-06-23 Smithkline Beecham Plc Kondenserede indolderivater som 5-HT4-receptorantagonister

Also Published As

Publication number Publication date
NO934881D0 (no) 1993-12-29
AU5276293A (en) 1994-07-14
US5418248A (en) 1995-05-23
IL108225A0 (en) 1994-04-12
ZA939760B (en) 1994-08-18
SK149393A3 (en) 1995-02-08
EP0605295A1 (fr) 1994-07-06
CZ291893A3 (en) 1994-07-13
FI935915A7 (fi) 1994-07-01
HU9303785D0 (en) 1994-04-28
FI935915A0 (fi) 1993-12-29
CA2112555A1 (en) 1994-07-01
FR2699921A1 (fr) 1994-07-01
AU666790B2 (en) 1996-02-22
TW257764B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1995-09-21
CN1036009C (zh) 1997-10-01
PL301680A1 (en) 1994-07-11
FI935915L (fi) 1994-07-01
CN1096029A (zh) 1994-12-07
IL108225A (en) 1997-04-15
HUT70409A (en) 1995-10-30
KR940014415A (ko) 1994-07-18
CZ282959B6 (cs) 1997-11-12
KR0140846B1 (ko) 1998-06-15
NO934881L (no) 1994-07-01
JPH06234770A (ja) 1994-08-23
NZ250579A (en) 1995-07-26

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Legal Events

Date Code Title Description
ST Notification of lapse