FR2457296A1 - Nouveaux derives de vinyl-3 cephalosporines et leur preparation - Google Patents

Nouveaux derives de vinyl-3 cephalosporines et leur preparation

Info

Publication number
FR2457296A1
FR2457296A1 FR7913096A FR7913096A FR2457296A1 FR 2457296 A1 FR2457296 A1 FR 2457296A1 FR 7913096 A FR7913096 A FR 7913096A FR 7913096 A FR7913096 A FR 7913096A FR 2457296 A1 FR2457296 A1 FR 2457296A1
Authority
FR
France
Prior art keywords
radical
preparation
protector
cephalosporins
eangeloma
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7913096A
Other languages
English (en)
French (fr)
Other versions
FR2457296B1 (US20100170793A1-20100708-C00006.png
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Rhone Poulenc Industries SA
Original Assignee
Rhone Poulenc Industries SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to FR7913096A priority Critical patent/FR2457296A1/fr
Application filed by Rhone Poulenc Industries SA filed Critical Rhone Poulenc Industries SA
Priority to PT71276A priority patent/PT71276A/pt
Priority to US06/152,085 priority patent/US4307233A/en
Priority to AU58595/80A priority patent/AU534806B2/en
Priority to DE19803019462 priority patent/DE3019462A1/de
Priority to SU802926697A priority patent/SU1031409A3/ru
Priority to AT0270980A priority patent/AT369375B/de
Priority to NO801502A priority patent/NO801502L/no
Priority to DD80221272A priority patent/DD150899A5/de
Priority to PL1980224391A priority patent/PL126481B1/pl
Priority to FI801641A priority patent/FI801641A/fi
Priority to DK222080A priority patent/DK222080A/da
Priority to CS803543A priority patent/CS244405B2/cs
Priority to CA000352324A priority patent/CA1144919A/fr
Priority to HU801278A priority patent/HU185890B/hu
Priority to GB8016727A priority patent/GB2051062B/en
Priority to IT22243/80A priority patent/IT1140974B/it
Priority to CH398980A priority patent/CH645379A5/fr
Priority to NZ193799A priority patent/NZ193799A/xx
Priority to YU01368/80A priority patent/YU136880A/xx
Priority to SE8003821A priority patent/SE451072B/sv
Priority to GR62015A priority patent/GR68426B/el
Priority to IE1062/80A priority patent/IE49814B1/en
Priority to ES491687A priority patent/ES491687A0/es
Priority to LU82477A priority patent/LU82477A1/fr
Priority to BE0/200707A priority patent/BE883416A/fr
Priority to ZA00803038A priority patent/ZA803038B/xx
Priority to PH24056A priority patent/PH15946A/en
Priority to IL60139A priority patent/IL60139A/xx
Priority to NL8003023A priority patent/NL8003023A/nl
Priority to JP6800980A priority patent/JPS55154981A/ja
Publication of FR2457296A1 publication Critical patent/FR2457296A1/fr
Application granted granted Critical
Publication of FR2457296B1 publication Critical patent/FR2457296B1/fr
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/02Nutrients, e.g. vitamins, minerals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Nutrition Science (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FR7913096A 1979-05-23 1979-05-23 Nouveaux derives de vinyl-3 cephalosporines et leur preparation Granted FR2457296A1 (fr)

Priority Applications (31)

Application Number Priority Date Filing Date Title
FR7913096A FR2457296A1 (fr) 1979-05-23 1979-05-23 Nouveaux derives de vinyl-3 cephalosporines et leur preparation
NZ193799A NZ193799A (en) 1979-05-23 1980-05-21 3-vinyl-cephalosporin derivatives
AU58595/80A AU534806B2 (en) 1979-05-23 1980-05-21 3-vinyl-cephalosporin derivatives
DE19803019462 DE3019462A1 (de) 1979-05-23 1980-05-21 Neue 3-vinyl-cephalosporin-derivate und verfahren zu deren herstellung
CH398980A CH645379A5 (fr) 1979-05-23 1980-05-21 Derives de vinyl-3 cephalosporines, et leur preparation.
AT0270980A AT369375B (de) 1979-05-23 1980-05-21 Verfahren zur herstellung von neuen 3-vinylcephalosporin-derivaten
NO801502A NO801502L (no) 1979-05-23 1980-05-21 Nye 3-aminovinylcefalosporiner og fremgangsmaate for fremstilling av disse.
US06/152,085 US4307233A (en) 1979-05-23 1980-05-21 3-Vinyl-cephalosporin derivatives
PL1980224391A PL126481B1 (en) 1979-05-23 1980-05-21 Method for producing new derivatives of 3-vinylcephalosporins
YU01368/80A YU136880A (en) 1979-05-23 1980-05-21 Process for obtaining new derivatives of 3-vinyl-cephalosporin
DK222080A DK222080A (da) 1979-05-23 1980-05-21 3-aminovinylcephalosporiner samt fremgangsmaade til fremstilling heraf
CS803543A CS244405B2 (en) 1979-05-23 1980-05-21 3-aminovinyl cephalosporines' new derivatives production method
CA000352324A CA1144919A (fr) 1979-05-23 1980-05-21 Derives de vinyl-3 cephalosporines, et leur preparation
HU801278A HU185890B (en) 1979-05-23 1980-05-21 Process for preparing 7-amino-3-vinyl-cefem-4-carboxylic acid derivatives
GB8016727A GB2051062B (en) 1979-05-23 1980-05-21 3-vinyl-cephalosporin derivatives and their preparation
IT22243/80A IT1140974B (it) 1979-05-23 1980-05-21 Derivati di vinil-3 cefalosporine, e loro preparazione
PT71276A PT71276A (fr) 1979-05-23 1980-05-21 Nouveaux derives de vinyl-3 cephalosporines et leur preparation
DD80221272A DD150899A5 (de) 1979-05-23 1980-05-21 Verfahren zur herstellung eines neuen 3-vinyl-cephalosporinderivates
FI801641A FI801641A (fi) 1979-05-23 1980-05-21 Nya derivat av vinyl-3 kefalosporiner och deras framstaellning
SE8003821A SE451072B (sv) 1979-05-23 1980-05-21 Nya 3-aminovinylcefalosporiner och forfarande for framstellning derav
GR62015A GR68426B (US20100170793A1-20100708-C00006.png) 1979-05-23 1980-05-21
IE1062/80A IE49814B1 (en) 1979-05-23 1980-05-21 Novel 3-vinyl-cephalosporin derivatives and their preparation
ES491687A ES491687A0 (es) 1979-05-23 1980-05-21 Procedimiento para la obtencion de derivados de vinil-3 ce- falosporina
LU82477A LU82477A1 (fr) 1979-05-23 1980-05-21 Nouveaux derives de vinyl-3 cephalosporines,et leur preparation
BE0/200707A BE883416A (fr) 1979-05-23 1980-05-21 Nouveaux derives de vinyl-3 cephalosporines, et leur preparation
ZA00803038A ZA803038B (en) 1979-05-23 1980-05-21 Novel 3-vinyl-cephalosporin derivatives and their preparation
SU802926697A SU1031409A3 (ru) 1979-05-23 1980-05-21 Способ получени производных 3-аминовинилцефалоспорина
PH24056A PH15946A (en) 1979-05-23 1980-05-22 3-vinyl-cephalosporin derivatives
IL60139A IL60139A (en) 1979-05-23 1980-05-22 3-amino vinyl cephalosporin derivatives and their preparation
NL8003023A NL8003023A (nl) 1979-05-23 1980-05-23 3-vinylcefalosporinederivaten en de bereiding van daarvan.
JP6800980A JPS55154981A (en) 1979-05-23 1980-05-23 Novel 33vinyllcephalosporin derivative and its manufacture

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7913096A FR2457296A1 (fr) 1979-05-23 1979-05-23 Nouveaux derives de vinyl-3 cephalosporines et leur preparation

Publications (2)

Publication Number Publication Date
FR2457296A1 true FR2457296A1 (fr) 1980-12-19
FR2457296B1 FR2457296B1 (US20100170793A1-20100708-C00006.png) 1982-02-05

Family

ID=9225762

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7913096A Granted FR2457296A1 (fr) 1979-05-23 1979-05-23 Nouveaux derives de vinyl-3 cephalosporines et leur preparation

Country Status (31)

Country Link
US (1) US4307233A (US20100170793A1-20100708-C00006.png)
JP (1) JPS55154981A (US20100170793A1-20100708-C00006.png)
AT (1) AT369375B (US20100170793A1-20100708-C00006.png)
AU (1) AU534806B2 (US20100170793A1-20100708-C00006.png)
BE (1) BE883416A (US20100170793A1-20100708-C00006.png)
CA (1) CA1144919A (US20100170793A1-20100708-C00006.png)
CH (1) CH645379A5 (US20100170793A1-20100708-C00006.png)
CS (1) CS244405B2 (US20100170793A1-20100708-C00006.png)
DD (1) DD150899A5 (US20100170793A1-20100708-C00006.png)
DE (1) DE3019462A1 (US20100170793A1-20100708-C00006.png)
DK (1) DK222080A (US20100170793A1-20100708-C00006.png)
ES (1) ES491687A0 (US20100170793A1-20100708-C00006.png)
FI (1) FI801641A (US20100170793A1-20100708-C00006.png)
FR (1) FR2457296A1 (US20100170793A1-20100708-C00006.png)
GB (1) GB2051062B (US20100170793A1-20100708-C00006.png)
GR (1) GR68426B (US20100170793A1-20100708-C00006.png)
HU (1) HU185890B (US20100170793A1-20100708-C00006.png)
IE (1) IE49814B1 (US20100170793A1-20100708-C00006.png)
IL (1) IL60139A (US20100170793A1-20100708-C00006.png)
IT (1) IT1140974B (US20100170793A1-20100708-C00006.png)
LU (1) LU82477A1 (US20100170793A1-20100708-C00006.png)
NL (1) NL8003023A (US20100170793A1-20100708-C00006.png)
NO (1) NO801502L (US20100170793A1-20100708-C00006.png)
NZ (1) NZ193799A (US20100170793A1-20100708-C00006.png)
PH (1) PH15946A (US20100170793A1-20100708-C00006.png)
PL (1) PL126481B1 (US20100170793A1-20100708-C00006.png)
PT (1) PT71276A (US20100170793A1-20100708-C00006.png)
SE (1) SE451072B (US20100170793A1-20100708-C00006.png)
SU (1) SU1031409A3 (US20100170793A1-20100708-C00006.png)
YU (1) YU136880A (US20100170793A1-20100708-C00006.png)
ZA (1) ZA803038B (US20100170793A1-20100708-C00006.png)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0053540A1 (fr) * 1980-11-20 1982-06-09 Rhone-Poulenc Sante Nouveaux dérivés de la céphalosporine et leur préparation
EP0053541A1 (fr) * 1980-11-20 1982-06-09 Rhone-Poulenc Sante Nouvelles oxacéphalosporines et leur préparation
FR2505334A1 (fr) * 1981-05-11 1982-11-12 Rhone Poulenc Sante Nouvelles oxacephalosporines et leur preparation
EP0072757A1 (fr) * 1981-08-17 1983-02-23 Rhone-Poulenc Sante Nouveaux dérivés de la céphalosporine et leur préparation

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL58717A (en) * 1978-11-15 1983-05-15 Glaxo Group Ltd Derivatives of(6r,7r)-7-((z)-2-(2-aminothiazol-4-yl)-2-(carboxy-(lower alkyl or cycloalkyl)oxyimino)acetamido)-3-(2-alkyl-pyrazolium-1-ylmethyl)ceph-3-em-4-carboxylate,process for their preparation and pharmaceutical compositions comprising them
FR2494275A2 (fr) * 1980-11-20 1982-05-21 Rhone Poulenc Ind Nouveaux derives de vinyl-3 cephalosporines et leur preparation
US4486586A (en) * 1983-02-10 1984-12-04 Bristol-Myers Company Cephalosporin derivatives
US4560749A (en) * 1983-11-18 1985-12-24 Eli Lilly And Company Cephem-3-imidates and 3-amidines
US4708955A (en) * 1985-06-24 1987-11-24 Bristol-Myers Company 3-(substituted)propenyl-7-aminothiazol-ylcephalosporanic acids and esters thereof
US4874856A (en) * 1985-06-24 1989-10-17 Bristol-Myers Company 3-(substituted)propenyl-7-(aminothiazolylacetamido) ceph-3-em-4-carboxylic acids and esters thereof
ATE92927T1 (de) * 1986-04-14 1993-08-15 Banyu Pharma Co Ltd 1-carboxy-1-vinyloxyiminoaminothiazolcephalosporin-derivate und deren herstellung.
DK0841339T3 (da) 1996-11-06 2007-07-02 Basilea Pharmaceutica Ag Vinylpyrrolidinon-cephalosporinderivater
WO2009049086A1 (en) 2007-10-09 2009-04-16 Larry Sutton Broad spectrum beta-lactamase inhibitors
JP6403289B2 (ja) 2013-03-12 2018-10-10 グラディウス ファーマシューティカルズ コーポレーションGladius Pharmaceuticals Corporation 誘導体化3−スチリル−セファロスポリン

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4065620A (en) * 1971-06-14 1977-12-27 Eli Lilly And Company 3-(Substituted) vinyl cephalosporins
GB1463077A (en) * 1973-04-19 1977-02-02 Glaxo Lab Ltd 7-substituted-ethyl-cephalosporin derivatives
CH617703A5 (en) * 1973-12-21 1980-06-13 Glaxo Operations Ltd Process for the preparation of the syn-isomer or of a mixture of syn- and anti-isomers of novel antibiotically active 7 beta -acylamino-ceph-3-em-4-carboxylic acids
US4095021A (en) * 1973-12-21 1978-06-13 Glaxo Laboratories Limited 3-Carbamoyloxymethyl or N-methyl-carbamoyloxymethyl-7-[2-carboxymethoxyimino-2-(fur-2-yl or thien-2-yl)acetamido]ceph-3-em-4-carboxylic acids and derivatives thereof
JPS5129492A (en) * 1974-09-04 1976-03-12 Sankyo Co Sefuarosuhorinjudotai no seiho
DK154939C (da) * 1974-12-19 1989-06-12 Takeda Chemical Industries Ltd Analogifremgangsmaade til fremstilling af thiazolylacetamido-cephemforbindelser eller farmaceutisk acceptable salte eller estere deraf
JPS5253890A (en) * 1975-10-14 1977-04-30 Syntex Inc Production of cephalosporin type compound
PT71654B (en) * 1979-08-15 1982-01-22 Merck & Co Inc Process for preparing allylsulfoxide enzyme inhibitor

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0053540A1 (fr) * 1980-11-20 1982-06-09 Rhone-Poulenc Sante Nouveaux dérivés de la céphalosporine et leur préparation
EP0053541A1 (fr) * 1980-11-20 1982-06-09 Rhone-Poulenc Sante Nouvelles oxacéphalosporines et leur préparation
FR2505334A1 (fr) * 1981-05-11 1982-11-12 Rhone Poulenc Sante Nouvelles oxacephalosporines et leur preparation
EP0072757A1 (fr) * 1981-08-17 1983-02-23 Rhone-Poulenc Sante Nouveaux dérivés de la céphalosporine et leur préparation

Also Published As

Publication number Publication date
GB2051062B (en) 1983-10-12
NZ193799A (en) 1983-03-15
AT369375B (de) 1982-12-27
ES8102136A1 (es) 1980-12-16
SE8003821L (sv) 1980-11-24
DE3019462A1 (de) 1980-12-04
YU136880A (en) 1983-04-30
CS244405B2 (en) 1986-07-17
ZA803038B (en) 1981-05-27
IT8022243A0 (it) 1980-05-21
GB2051062A (en) 1981-01-14
PT71276A (fr) 1980-06-01
PL126481B1 (en) 1983-08-31
JPH0246595B2 (US20100170793A1-20100708-C00006.png) 1990-10-16
IT1140974B (it) 1986-10-10
JPS55154981A (en) 1980-12-02
SE451072B (sv) 1987-08-31
HU185890B (en) 1985-04-28
NL8003023A (nl) 1980-11-25
AU5859580A (en) 1980-11-27
CS354380A2 (US20100170793A1-20100708-C00006.png) 1985-09-17
NO801502L (no) 1980-11-24
IL60139A0 (en) 1980-07-31
SU1031409A3 (ru) 1983-07-23
PH15946A (en) 1983-04-29
BE883416A (fr) 1980-11-21
CH645379A5 (fr) 1984-09-28
PL224391A1 (US20100170793A1-20100708-C00006.png) 1981-02-13
IE49814B1 (en) 1985-12-25
AU534806B2 (en) 1984-02-16
IL60139A (en) 1984-04-30
DK222080A (da) 1980-11-24
LU82477A1 (fr) 1980-12-16
FR2457296B1 (US20100170793A1-20100708-C00006.png) 1982-02-05
FI801641A (fi) 1980-11-24
ATA270980A (de) 1982-05-15
US4307233A (en) 1981-12-22
DD150899A5 (de) 1981-09-23
GR68426B (US20100170793A1-20100708-C00006.png) 1981-12-30
ES491687A0 (es) 1980-12-16
CA1144919A (fr) 1983-04-19
IE801062L (en) 1980-11-23

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