FR2444038A1 - Derives de pyrazolo(1,5-c)quinazoline utiles comme medicaments et leurs procedes de preparation - Google Patents

Derives de pyrazolo(1,5-c)quinazoline utiles comme medicaments et leurs procedes de preparation

Info

Publication number
FR2444038A1
FR2444038A1 FR7930624A FR7930624A FR2444038A1 FR 2444038 A1 FR2444038 A1 FR 2444038A1 FR 7930624 A FR7930624 A FR 7930624A FR 7930624 A FR7930624 A FR 7930624A FR 2444038 A1 FR2444038 A1 FR 2444038A1
Authority
FR
France
Prior art keywords
preparation
pyrazolo
medicaments
processes
derivatives useful
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
FR7930624A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
ER Squibb and Sons LLC
Original Assignee
ER Squibb and Sons LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ER Squibb and Sons LLC filed Critical ER Squibb and Sons LLC
Publication of FR2444038A1 publication Critical patent/FR2444038A1/fr
Withdrawn legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pulmonology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

L'invention concerne des dérivés de pyrazoloØ1,5-cõquinazoline utiles notamment comme médicaments antiallergiques et des procédés de leur préparation. Les composés de l'invention répondent à la formule :
FR7930624A 1978-12-13 1979-12-13 Derives de pyrazolo(1,5-c)quinazoline utiles comme medicaments et leurs procedes de preparation Withdrawn FR2444038A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/969,642 US4198412A (en) 1978-12-13 1978-12-13 Pyrazolo [1,5-C] quinazoline derivatives and their use in treating allergic conditions

Publications (1)

Publication Number Publication Date
FR2444038A1 true FR2444038A1 (fr) 1980-07-11

Family

ID=25515802

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7930624A Withdrawn FR2444038A1 (fr) 1978-12-13 1979-12-13 Derives de pyrazolo(1,5-c)quinazoline utiles comme medicaments et leurs procedes de preparation

Country Status (15)

Country Link
US (1) US4198412A (fr)
JP (1) JPS5583787A (fr)
AU (1) AU5359379A (fr)
BE (1) BE880607A (fr)
CA (1) CA1122215A (fr)
DE (1) DE2950234A1 (fr)
DK (1) DK529179A (fr)
FR (1) FR2444038A1 (fr)
GB (1) GB2039896A (fr)
IT (1) IT1164093B (fr)
LU (1) LU81987A1 (fr)
NL (1) NL7908940A (fr)
NO (1) NO794064L (fr)
SE (1) SE7910255L (fr)
ZA (1) ZA796589B (fr)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU178523B (en) * 1979-05-18 1982-05-28 Egyt Gyogyszervegyeszeti Gyar Process for preparing new pyrazolo-quinazoline derivatives
CN103130810B (zh) * 2013-03-11 2015-02-25 河南师范大学 一种吡唑并[1,5-c]喹唑啉类化合物的合成方法
KR20150010548A (ko) * 2013-07-17 2015-01-28 희성소재 (주) 질소함유 다환고리 화합물 및 이를 이용한 유기발광소자

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3313815A (en) * 1964-05-04 1967-04-11 Sterling Drug Inc 8-chloropyrazolo-[1, 5-c]quinazoline derivatives and methods of preparing same
US3895027A (en) * 1974-04-12 1975-07-15 Lilly Co Eli Process for preparing pyrazole-3-carboxylic acids
US3899508A (en) * 1974-04-12 1975-08-12 Lilly Co Eli 5-(2-Aminophenyl)pyrazole-3-carboxylic acids and esters thereof
US4076818A (en) * 1976-07-02 1978-02-28 E. R. Squibb & Sons, Inc. Pyrazolo [1,5-C]quinazoline derivatives and related compounds
US4129653A (en) * 1977-01-05 1978-12-12 Ortho Pharmaceutical Corporation Substituted pyrrolo [1,2-c] quinazolines and pharmaceutical compositions and methods employing them
US4112098A (en) * 1977-10-17 1978-09-05 E. R. Squibb & Sons, Inc. Pyrazolo[1,5-c]quinazoline derivatives and related compounds
US4128644A (en) * 1977-07-29 1978-12-05 E. R. Squibb & Sons, Inc. Pyrazolo(1,5-c)quinazoline derivatives and related compounds
US4110452A (en) * 1977-10-17 1978-08-29 E. R. Squibb & Sons, Inc. Pyrazolo (1,5-c) quinazoline derivatives and related compounds

Also Published As

Publication number Publication date
IT1164093B (it) 1987-04-08
GB2039896A (en) 1980-08-20
NL7908940A (nl) 1980-06-17
US4198412A (en) 1980-04-15
AU5359379A (en) 1980-06-19
IT7951070A0 (it) 1979-12-12
NO794064L (no) 1980-06-16
CA1122215A (fr) 1982-04-20
JPS5583787A (en) 1980-06-24
LU81987A1 (fr) 1980-04-22
DK529179A (da) 1980-06-14
DE2950234A1 (de) 1980-06-26
SE7910255L (sv) 1980-06-14
BE880607A (fr) 1980-06-13
ZA796589B (en) 1980-11-26

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Legal Events

Date Code Title Description
RE Withdrawal of published application