IT7951070A0 - Composti pirazolo (1,5-c) chinazolinici dotati di attivita' antiallergica e procedimento di preparazione - Google Patents

Composti pirazolo (1,5-c) chinazolinici dotati di attivita' antiallergica e procedimento di preparazione

Info

Publication number
IT7951070A0
IT7951070A0 IT7951070A IT5107079A IT7951070A0 IT 7951070 A0 IT7951070 A0 IT 7951070A0 IT 7951070 A IT7951070 A IT 7951070A IT 5107079 A IT5107079 A IT 5107079A IT 7951070 A0 IT7951070 A0 IT 7951070A0
Authority
IT
Italy
Prior art keywords
pyrazole
preparation procedure
quinazoline compounds
antiallergic activity
antiallergic
Prior art date
Application number
IT7951070A
Other languages
English (en)
Other versions
IT1164093B (it
Inventor
Berthold R Vogt
Ligaya M Simpkins
Original Assignee
Squibb & Sons Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Squibb & Sons Inc filed Critical Squibb & Sons Inc
Publication of IT7951070A0 publication Critical patent/IT7951070A0/it
Application granted granted Critical
Publication of IT1164093B publication Critical patent/IT1164093B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pulmonology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IT51070/79A 1978-12-13 1979-12-12 Composti pirazolo (1,5-c) chinazolinici dotati di attivita' antialler gica e procedimento di preparazione IT1164093B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/969,642 US4198412A (en) 1978-12-13 1978-12-13 Pyrazolo [1,5-C] quinazoline derivatives and their use in treating allergic conditions

Publications (2)

Publication Number Publication Date
IT7951070A0 true IT7951070A0 (it) 1979-12-12
IT1164093B IT1164093B (it) 1987-04-08

Family

ID=25515802

Family Applications (1)

Application Number Title Priority Date Filing Date
IT51070/79A IT1164093B (it) 1978-12-13 1979-12-12 Composti pirazolo (1,5-c) chinazolinici dotati di attivita' antialler gica e procedimento di preparazione

Country Status (15)

Country Link
US (1) US4198412A (it)
JP (1) JPS5583787A (it)
AU (1) AU5359379A (it)
BE (1) BE880607A (it)
CA (1) CA1122215A (it)
DE (1) DE2950234A1 (it)
DK (1) DK529179A (it)
FR (1) FR2444038A1 (it)
GB (1) GB2039896A (it)
IT (1) IT1164093B (it)
LU (1) LU81987A1 (it)
NL (1) NL7908940A (it)
NO (1) NO794064L (it)
SE (1) SE7910255L (it)
ZA (1) ZA796589B (it)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU178523B (en) * 1979-05-18 1982-05-28 Egyt Gyogyszervegyeszeti Gyar Process for preparing new pyrazolo-quinazoline derivatives
CN103130810B (zh) * 2013-03-11 2015-02-25 河南师范大学 一种吡唑并[1,5-c]喹唑啉类化合物的合成方法
CN105408333B (zh) * 2013-07-17 2018-10-16 喜星素材株式会社 含氮多环化合物和使用其的有机发光器件

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3313815A (en) * 1964-05-04 1967-04-11 Sterling Drug Inc 8-chloropyrazolo-[1, 5-c]quinazoline derivatives and methods of preparing same
US3895027A (en) * 1974-04-12 1975-07-15 Lilly Co Eli Process for preparing pyrazole-3-carboxylic acids
US3899508A (en) * 1974-04-12 1975-08-12 Lilly Co Eli 5-(2-Aminophenyl)pyrazole-3-carboxylic acids and esters thereof
US4076818A (en) * 1976-07-02 1978-02-28 E. R. Squibb & Sons, Inc. Pyrazolo [1,5-C]quinazoline derivatives and related compounds
US4129653A (en) * 1977-01-05 1978-12-12 Ortho Pharmaceutical Corporation Substituted pyrrolo [1,2-c] quinazolines and pharmaceutical compositions and methods employing them
US4112098A (en) * 1977-10-17 1978-09-05 E. R. Squibb & Sons, Inc. Pyrazolo[1,5-c]quinazoline derivatives and related compounds
US4110452A (en) * 1977-10-17 1978-08-29 E. R. Squibb & Sons, Inc. Pyrazolo (1,5-c) quinazoline derivatives and related compounds
US4128644A (en) * 1977-07-29 1978-12-05 E. R. Squibb & Sons, Inc. Pyrazolo(1,5-c)quinazoline derivatives and related compounds

Also Published As

Publication number Publication date
JPS5583787A (en) 1980-06-24
DK529179A (da) 1980-06-14
NL7908940A (nl) 1980-06-17
GB2039896A (en) 1980-08-20
ZA796589B (en) 1980-11-26
DE2950234A1 (de) 1980-06-26
IT1164093B (it) 1987-04-08
AU5359379A (en) 1980-06-19
BE880607A (fr) 1980-06-13
US4198412A (en) 1980-04-15
NO794064L (no) 1980-06-16
FR2444038A1 (fr) 1980-07-11
CA1122215A (en) 1982-04-20
SE7910255L (sv) 1980-06-14
LU81987A1 (fr) 1980-04-22

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