FR2435945A1 - Perfectionnements a des compositions contenant de l'etomidate - Google Patents

Perfectionnements a des compositions contenant de l'etomidate

Info

Publication number
FR2435945A1
FR2435945A1 FR7922235A FR7922235A FR2435945A1 FR 2435945 A1 FR2435945 A1 FR 2435945A1 FR 7922235 A FR7922235 A FR 7922235A FR 7922235 A FR7922235 A FR 7922235A FR 2435945 A1 FR2435945 A1 FR 2435945A1
Authority
FR
France
Prior art keywords
etomidate
compositions containing
liquid infusion
containing etomidate
anesthetics
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7922235A
Other languages
English (en)
Other versions
FR2435945B1 (fr
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Janssen Pharmaceutica NV
Original Assignee
Janssen Pharmaceutica NV
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica NV filed Critical Janssen Pharmaceutica NV
Publication of FR2435945A1 publication Critical patent/FR2435945A1/fr
Application granted granted Critical
Publication of FR2435945B1 publication Critical patent/FR2435945B1/fr
Granted legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P23/00Anaesthetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Dermatology (AREA)
  • Anesthesiology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medical Preparation Storing Or Oral Administration Devices (AREA)

Abstract

L'invention concerne une infusion liquide contenant de l'étomidate pour une administration intraveineuse. Selon l'invention, elle se compose d'une infusion liquide physiologiquement acceptable à laquelle a été ajoutée une solution de chlorhydrate ou de bromhydrate d'étomidate dans un milieu qui contient au moins 80 % en poids d'éthanol. L'invention s'applique notamment à la préparation d'anesthésiques.
FR7922235A 1978-09-14 1979-09-05 Perfectionnements a des compositions contenant de l'etomidate Granted FR2435945A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US94223678A 1978-09-14 1978-09-14

Publications (2)

Publication Number Publication Date
FR2435945A1 true FR2435945A1 (fr) 1980-04-11
FR2435945B1 FR2435945B1 (fr) 1983-02-25

Family

ID=25477775

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7922235A Granted FR2435945A1 (fr) 1978-09-14 1979-09-05 Perfectionnements a des compositions contenant de l'etomidate

Country Status (19)

Country Link
US (1) US4289783A (fr)
JP (1) JPS5547858A (fr)
BE (1) BE878709A (fr)
CA (1) CA1140048A (fr)
CH (1) CH651752A5 (fr)
CY (1) CY1254A (fr)
DE (1) DE2937290A1 (fr)
DK (1) DK154926C (fr)
ES (1) ES484160A1 (fr)
FR (1) FR2435945A1 (fr)
GB (1) GB2029700B (fr)
GR (1) GR64915B (fr)
HK (1) HK80984A (fr)
HU (1) HU179989B (fr)
IE (1) IE48689B1 (fr)
IT (1) IT1120537B (fr)
KE (1) KE3426A (fr)
NL (1) NL7906835A (fr)
SE (1) SE447961B (fr)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ225045A (en) * 1987-07-01 1990-06-26 Janssen Pharmaceutica Nv Antiviral pharmaceutical compositions containing cyclodextrin and an antiviral agent
DE19709704C2 (de) 1997-03-10 1999-11-04 Michael Georgieff Verwendung einer flüssigen Präparation von Xenon zur intravenösen Verabreichung bei Einleitung und/oder Aufrechterhaltung der Anaesthesie
US20080268067A1 (en) 2007-03-09 2008-10-30 Llinas Rodolfo R Methods and Compositions for Treating Thalamocortical Dysrhythmia
US8911383B2 (en) 2007-12-20 2014-12-16 Acarix A/S Adhesive patch for monitoring acoustic signals
US8557856B2 (en) 2008-03-31 2013-10-15 The General Hospital Corporation Etomidate analogues with improved pharmacokinetic and pharmacodynamic properties
US8765973B2 (en) 2009-07-10 2014-07-01 The General Hospital Corporation Etomidate analogues that do not inhibit adrenocortical steroid synthesis
SG11201403980VA (en) 2012-01-13 2014-08-28 Gen Hospital Corp Anesthetic compounds and related methods of use
EP3206683A4 (fr) 2014-10-16 2018-06-13 The Board of Trustees of the Leland Stanford Junior University Nouveaux procédés, composés et compositions d'anesthésie

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3354173A (en) * 1964-04-16 1967-11-21 Janssen Pharmaceutica Nv Imidazole carboxylates

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3354173A (en) * 1964-04-16 1967-11-21 Janssen Pharmaceutica Nv Imidazole carboxylates

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
CA1978 *

Also Published As

Publication number Publication date
IE48689B1 (en) 1985-04-17
JPS5547858A (en) 1980-04-05
ES484160A1 (es) 1980-10-01
US4289783A (en) 1981-09-15
JPH0214058B2 (fr) 1990-04-06
SE7907621L (sv) 1980-03-15
SE447961B (sv) 1987-01-12
DE2937290A1 (de) 1980-04-03
HU179989B (en) 1983-01-28
IT1120537B (it) 1986-03-26
NL7906835A (nl) 1980-03-18
IT7950093A0 (it) 1979-08-23
DK154926B (da) 1989-01-09
GB2029700B (en) 1983-03-30
GR64915B (en) 1980-06-09
HK80984A (en) 1984-11-25
CH651752A5 (de) 1985-10-15
GB2029700A (en) 1980-03-26
CA1140048A (fr) 1983-01-25
BE878709A (nl) 1980-03-11
CY1254A (en) 1984-08-31
KE3426A (en) 1984-08-10
IE791741L (en) 1980-03-14
FR2435945B1 (fr) 1983-02-25
DK154926C (da) 1989-05-29
DK384379A (da) 1980-03-15

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Legal Events

Date Code Title Description
CC Supplementary protection certificate (spc) laid open to the public (law of 25 june 1990)

Free format text: 92C0445, 920618

CB Supplementary protection certificate (spc) granted (law of 25 june 1990)

Free format text: 92C0445, 790905

CP Supplementary protection certificate (spc) filed