FR2372808A1 - Nouveaux derives levogyres de 3-phenoxy n-substitue morphinane, leur preparation et leur application en tant que medicaments - Google Patents

Nouveaux derives levogyres de 3-phenoxy n-substitue morphinane, leur preparation et leur application en tant que medicaments

Info

Publication number
FR2372808A1
FR2372808A1 FR7736745A FR7736745A FR2372808A1 FR 2372808 A1 FR2372808 A1 FR 2372808A1 FR 7736745 A FR7736745 A FR 7736745A FR 7736745 A FR7736745 A FR 7736745A FR 2372808 A1 FR2372808 A1 FR 2372808A1
Authority
FR
France
Prior art keywords
preparation
application
new
levogyrates
morphinane
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7736745A
Other languages
English (en)
French (fr)
Other versions
FR2372808B1 (enExample
Inventor
Ernest Mohacsi
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
F Hoffmann La Roche AG
Original Assignee
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/811,233 external-priority patent/US4113729A/en
Application filed by F Hoffmann La Roche AG filed Critical F Hoffmann La Roche AG
Publication of FR2372808A1 publication Critical patent/FR2372808A1/fr
Application granted granted Critical
Publication of FR2372808B1 publication Critical patent/FR2372808B1/fr
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D217/00Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/12Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring
    • C07D217/18Aralkyl radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D221/00Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/22Bridged ring systems
    • C07D221/28Morphinans

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
FR7736745A 1976-12-06 1977-12-06 Nouveaux derives levogyres de 3-phenoxy n-substitue morphinane, leur preparation et leur application en tant que medicaments Granted FR2372808A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US74802276A 1976-12-06 1976-12-06
US05/811,233 US4113729A (en) 1976-12-06 1977-06-29 3-Phenoxymorphinans and derivatives thereof

Publications (2)

Publication Number Publication Date
FR2372808A1 true FR2372808A1 (fr) 1978-06-30
FR2372808B1 FR2372808B1 (enExample) 1981-07-10

Family

ID=27114858

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7736745A Granted FR2372808A1 (fr) 1976-12-06 1977-12-06 Nouveaux derives levogyres de 3-phenoxy n-substitue morphinane, leur preparation et leur application en tant que medicaments

Country Status (22)

Country Link
JP (1) JPS5392776A (enExample)
AR (1) AR219510A1 (enExample)
AT (1) AT364826B (enExample)
AU (1) AU514827B2 (enExample)
CA (1) CA1088935A (enExample)
DE (1) DE2754062A1 (enExample)
DK (1) DK540977A (enExample)
ES (3) ES464751A1 (enExample)
FI (1) FI773636A7 (enExample)
FR (1) FR2372808A1 (enExample)
GB (1) GB1589792A (enExample)
HU (1) HU177640B (enExample)
IE (1) IE46003B1 (enExample)
IL (1) IL53532A (enExample)
IT (1) IT1143727B (enExample)
LU (1) LU78638A1 (enExample)
MC (1) MC1172A1 (enExample)
NL (1) NL7713432A (enExample)
NO (1) NO774155L (enExample)
NZ (1) NZ185860A (enExample)
PT (1) PT67363B (enExample)
SE (1) SE7713779L (enExample)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4247697A (en) * 1979-09-10 1981-01-27 Hoffmann-La Roche Inc. 3-Phenoxy morphinans and their derivatives
TW264473B (enExample) * 1993-01-06 1995-12-01 Hoffmann La Roche

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1584396A (enExample) * 1967-08-25 1969-12-19
FR2052877A5 (enExample) * 1969-06-24 1971-04-09 Shionogi & Co

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1584396A (enExample) * 1967-08-25 1969-12-19
FR2052877A5 (enExample) * 1969-06-24 1971-04-09 Shionogi & Co

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
CA1963 *
CA1965 *

Also Published As

Publication number Publication date
PT67363A (en) 1978-01-01
IL53532A0 (en) 1978-03-10
NZ185860A (en) 1980-10-24
AT364826B (de) 1981-11-25
PT67363B (en) 1979-12-17
GB1589792A (en) 1981-05-20
ATA869277A (de) 1981-04-15
IT1143727B (it) 1986-10-22
ES464751A1 (es) 1978-12-16
NO774155L (no) 1978-06-07
MC1172A1 (fr) 1978-09-25
AR219510A1 (es) 1980-08-29
DK540977A (da) 1978-06-07
ES472572A1 (es) 1979-02-16
FI773636A7 (fi) 1978-06-07
NL7713432A (nl) 1978-06-08
AU514827B2 (en) 1981-02-26
CA1088935A (en) 1980-11-04
FR2372808B1 (enExample) 1981-07-10
JPS5392776A (en) 1978-08-15
IL53532A (en) 1981-09-13
HU177640B (en) 1981-11-28
IE46003L (en) 1978-06-06
DE2754062A1 (de) 1978-06-08
LU78638A1 (enExample) 1979-02-02
SE7713779L (sv) 1978-06-07
AU3126477A (en) 1979-06-14
ES472573A1 (es) 1979-02-16
IE46003B1 (en) 1983-01-26

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Legal Events

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